Works matching IS 18607179 AND DT 2023 AND VI 18 AND IP 8

Results: 9

Front Cover: Facile, Single‐Step Synthesis of a Series of D‐Ring Ethisterones Substituted with 1,4‐1,2,3‐Triazoles: Preliminary Evaluation of Cytotoxic Activities (ChemMedChem 8/2023).

Published in:

ChemMedChem, 2023, v. 18, n. 8, p. 1, doi. 10.1002/cmdc.202300190

By:

Canseco‐González, Daniel;
Rodríguez‐Victoria, Isaac;
Apan‐Ramírez, Teresa;
Viviano‐Posadas, Alejandro O.;
Serrano‐García, Juan S.;
Arenaza‐Corona, Antonino;
Orjuela, Adrian L.;
Alí‐Torres, Jorge;
Dorazco‐González, Alejandro;
Morales‐Morales, David

Publication type:

Article

Discovery of SI 1/20 and SI 1/22 as Mutual Prodrugs of 5‐Fluorouracil and Imidazole‐Based Heme Oxygenase 1 Inhibitor with Improved Cytotoxicity in DU145 Prostate Cancer Cells.

Published in:

ChemMedChem, 2023, v. 18, n. 8, p. 1, doi. 10.1002/cmdc.202300047

By:

Salerno, Loredana;
Sorrenti, Valeria;
Pittalà, Valeria;
Consoli, Valeria;
Modica, Maria N.;
Romeo, Giuseppe;
Marrazzo, Agostino;
Giuliano, Michela;
Zajdel, Paweł;
Vanella, Luca;
Intagliata, Sebastiano

Publication type:

Article

Design of OSMI‐4 Analogs Using Scaffold Hopping: Investigating the Importance of the Uridine Mimic in the Binding of OGT Inhibitors.

Published in:

ChemMedChem, 2023, v. 18, n. 8, p. 1, doi. 10.1002/cmdc.202300001

By:

Balsollier, Cyril;
Tomašič, Tihomir;
Yasini, Daniel;
Bijkerk, Simon;
Anderluh, Marko;
Pieters, Roland J.

Publication type:

Article

Imidazo[1,2‐a]pyridine Derivatives as AMPK Activators: Synthesis, Structure–Activity Relationships, and Regulation of Reactive Oxygen Species in Renal Fibroblasts.

Published in:

ChemMedChem, 2023, v. 18, n. 8, p. 1, doi. 10.1002/cmdc.202200696

By:

Wu, Siming;
Xiao, Zhihong;
Wei, Junling;
Zhang, Lei;
Cao, Yuanyuan;
Chen., Zhuo;
Li, Qianbin;
Hu, Gaoyun

Publication type:

Article

Exploration of the Binding Modes of Toll‐Like Receptor 4 Competitive Inhibitors: A Combined Ligand‐Based and Target‐Based Approach.

Published in:

ChemMedChem, 2023, v. 18, n. 8, p. 1, doi. 10.1002/cmdc.202200690

By:

Dang, Wen;
Meng, Churen;
Wang, Jian;
Zhou, Di;
Chen, Gang;
Li, Ning

Publication type:

Article

Recent Development of Copper (II) Complexes of Polypyridyl Ligands in Chemotherapy and Photodynamic Therapy.

Published in:

ChemMedChem, 2023, v. 18, n. 8, p. 1, doi. 10.1002/cmdc.202200652

By:

Rani J, Jansi;
Roy, Sovan

Publication type:

Article

Anticancer Activities of Tetrasubstituted Imidazole‐Pyrimidine‐Sulfonamide Hybrids as Inhibitors of EGFR Mutants.

Published in:

ChemMedChem, 2023, v. 18, n. 8, p. 1, doi. 10.1002/cmdc.202200641

By:

Alghamdi, Eman M.;
Alamshany, Zahra M.;
El Hamd, Mohamed A.;
Taher, Ehab S.;
Farrag El‐Behairy, Mohammed;
Norcott, Philip L.;
Marzouk, Adel A.

Publication type:

Article

Systematic Potency and Property Assessment of VHL Ligands and Implications on PROTAC Design.

Published in:

ChemMedChem, 2023, v. 18, n. 8, p. 1, doi. 10.1002/cmdc.202200615

By:

Krieger, Johannes;
Sorrell, Fiona J.;
Wegener, Ansgar A.;
Leuthner, Birgitta;
Machrouhi‐Porcher, Fouzia;
Hecht, Martin;
Leibrock, Eva M.;
Müller, Juliane E.;
Eisert, Jonathan;
Hartung, Ingo V.;
Schlesiger, Sarah

Publication type:

Article

Facile, Single‐Step Synthesis of a Series of D‐Ring Ethisterones Substituted with 1,4‐1,2,3‐Triazoles: Preliminary Evaluation of Cytotoxic Activities.

Published in:

ChemMedChem, 2023, v. 18, n. 8, p. 1, doi. 10.1002/cmdc.202200659

By:

Canseco‐González, Daniel;
Rodríguez‐Victoria, Isaac;
Apan‐Ramírez, Teresa;
Viviano‐Posadas, Alejandro O.;
Serrano‐García, Juan S.;
Arenaza‐Corona, Antonino;
Orjuela, Adrian L.;
Alí‐Torres, Jorge;
Dorazco‐González, Alejandro;
Morales‐Morales, David

Publication type:

Article