Works matching IS 18607179 AND DT 2022 AND VI 17 AND IP 1

Results: 20

Front Cover: MPI8 is Potent against SARS‐CoV‐2 by Inhibiting Dually and Selectively the SARS‐CoV‐2 Main Protease and the Host Cathepsin L (ChemMedChem 1/2022).

Published in:

ChemMedChem, 2022, v. 17, n. 1, p. 1, doi. 10.1002/cmdc.202100769

By:

Ma, Xinyu R.;
Alugubelli, Yugendar R.;
Ma, Yuying;
Vatansever, Erol C.;
Scott, Danielle A.;
Qiao, Yuchen;
Yu, Ge;
Xu, Shiqing;
Liu, Wenshe Ray

Publication type:

Article

Something New in 22!

Published in:: ChemMedChem, 2022, v. 17, n. 1, p. 1, doi. 10.1002/cmdc.202100768
Publication type:: Article

A Bivalent Supramolecular GCP Ligand Enables Blocking of the Taspase1/Importin α Interaction.

Published in:

ChemMedChem, 2022, v. 17, n. 1, p. 1, doi. 10.1002/cmdc.202100640

By:

Höing, Alexander;
Zimmermann, Alexander;
Moews, Lisa;
Killa, Matthias;
Heimann, Marius;
Hensel, Astrid;
Voskuhl, Jens;
Knauer, Shirley K.

Publication type:

Article

Stimuli‐Responsive DNA Origami Nanodevices and Their Biological Applications.

Published in:

ChemMedChem, 2022, v. 17, n. 1, p. 1, doi. 10.1002/cmdc.202100635

By:

Pitikultham, Piyawat;
Wang, Zhaoran;
Wang, Yiming;
Shang, Yingxu;
Jiang, Qiao;
Ding, Baoquan

Publication type:

Article

Prodrugs of E‐selectin Antagonists with Enhanced Pharmacokinetic Properties.

Published in:

ChemMedChem, 2022, v. 17, n. 1, p. 1, doi. 10.1002/cmdc.202100634

By:

Dätwyler, Philipp;
Jiang, Xiaohua;
Wagner, Beatrice;
Varga, Norbert;
Mühlethaler, Tobias;
Hostettler, Katja;
Rabbani, Said;
Schwardt, Oliver;
Ernst, Beat

Publication type:

Article

Borcalein: a Carborane‐Based Analogue of Baicalein with 12‐Lipoxygenase‐Independent Toxicity.

Published in:

ChemMedChem, 2022, v. 17, n. 1, p. 1, doi. 10.1002/cmdc.202100588

By:

Kuhnert, Robert;
Kuhnert, Lydia;
Sárosi, Menyhárt‐B.;
George, Sven;
Draca, Dijana;
Paskas, Svetlana;
Hofmann, Bettina;
Steinhilber, Dieter;
Honscha, Walther;
Mijatović, Sanja;
Maksimović‐Ivanić, Danijela;
Hey‐Hawkins, Evamarie

Publication type:

Article

Interaction of Copper Trafficking Proteins with the Platinum Anticancer Drug Kiteplatin.

Published in:

ChemMedChem, 2022, v. 17, n. 1, p. 1, doi. 10.1002/cmdc.202100593

By:

Barbanente, Alessandra;
Galliani, Angela;
Iacobazzi, Rosa Maria;
Lasorsa, Alessia;
Nardella, Maria Incoronata;
Pennetta, Antonio;
Margiotta, Nicola;
Arnesano, Fabio

Publication type:

Article

A Patent Review on SARS Coronavirus Main Protease (3CL<sup>pro</sup>) Inhibitors.

Published in:

ChemMedChem, 2022, v. 17, n. 1, p. 1, doi. 10.1002/cmdc.202100576

By:

Chia, C. S. Brian;
Xu, Weijun;
Shuyi Ng, Pearly

Publication type:

Article

Halogen‐Dance‐Based Synthesis of Phosphonomethoxyethyl (PME) Substituted 2‐Aminothiazoles as Potent Inhibitors of Bacterial Adenylate Cyclases.

Published in:

ChemMedChem, 2022, v. 17, n. 1, p. 1, doi. 10.1002/cmdc.202100568

By:

Česnek, Michal;
Šafránek, Michal;
Dračínský, Martin;
Tloušťová, Eva;
Mertlíková‐Kaiserová, Helena;
Hayes, Michael P.;
Watts, Val J.;
Janeba, Zlatko

Publication type:

Article

Pyrimidyn‐Based Dynamin Inhibitors as Novel Cytotoxic Agents.

Published in:

ChemMedChem, 2022, v. 17, n. 1, p. 1, doi. 10.1002/cmdc.202100560

By:

Odell, Luke R.;
Chau, Ngoc;
Russell, Cecilia C.;
Young, Kelly A.;
Gilbert, Jayne;
Robinson, Phillip J.;
Sakoff, Jennette A.;
McCluskey, Adam

Publication type:

Article

Discovery of Isatin‐Based Carbohydrazones as Potential Dual Inhibitors of Fatty Acid Amide Hydrolase and Monoacylglycerol Lipase.

Published in:

ChemMedChem, 2022, v. 17, n. 1, p. 1, doi. 10.1002/cmdc.202100559

By:

Jaiswal, Shivani;
Ayyannan, Senthil Raja

Publication type:

Article

Synthesis, Binding Affinity Analysis, and <sup>18</sup>F Radiosynthesis of Small‐Molecular‐Weight HIF‐1α‐Binding Compounds.

Published in:

ChemMedChem, 2022, v. 17, n. 1, p. 1, doi. 10.1002/cmdc.202100544

By:

Dawn Woodfield, Jenilee;
Bhardwaj, Atul;
Bergman, Cody;
Wuest, Frank

Publication type:

Article

Recent Advances in the Prediction of Pharmacokinetics Properties in Drug Design Studies: A Review.

Published in:

ChemMedChem, 2022, v. 17, n. 1, p. 1, doi. 10.1002/cmdc.202100542

By:

Pantaleão, Simone Q.;
Fernandes, Philipe O.;
Gonçalves, José Eduardo;
Maltarollo, Vinícius G.;
Honorio, Kathia Maria

Publication type:

Article

Revisiting the Molecular Interactions between the Tumor Protein TCTP and the Drugs Sertraline/Thioridazine.

Published in:

ChemMedChem, 2022, v. 17, n. 1, p. 1, doi. 10.1002/cmdc.202100528

By:

Malard, Florian;
Jacquet, Eric;
Nhiri, Naima;
Sizun, Christina;
Chabrier, Amélie;
Messaoudi, Samir;
Dejeu, Jérôme;
Betzi, Stéphane;
Zhang, Xu;
Thureau, Aurélien;
Lescop, Ewen

Publication type:

Article

MPI8 is Potent against SARS‐CoV‐2 by Inhibiting Dually and Selectively the SARS‐CoV‐2 Main Protease and the Host Cathepsin L**.

Published in:

ChemMedChem, 2022, v. 17, n. 1, p. 1, doi. 10.1002/cmdc.202100456

By:

Ma, Xinyu R.;
Alugubelli, Yugendar R.;
Ma, Yuying;
Vatansever, Erol C.;
Scott, Danielle A.;
Qiao, Yuchen;
Yu, Ge;
Xu, Shiqing;
Liu, Wenshe Ray

Publication type:

Article

Drug Repurposing for the SARS‐CoV‐2 Papain‐Like Protease.

Published in:

ChemMedChem, 2022, v. 17, n. 1, p. 1, doi. 10.1002/cmdc.202100455

By:

Cho, Chia‐Chuan;
Li, Shuhua G.;
Lalonde, Tyler J.;
Yang, Kai S.;
Yu, Ge;
Qiao, Yuchen;
Xu, Shiqing;
Ray Liu, Wenshe

Publication type:

Article

Sophoridine Derivatives Induce Apoptosis and Autophagy to Suppress the Growth of Triple‐Negative Breast Cancer through Inhibition of mTOR Signaling.

Published in:

ChemMedChem, 2022, v. 17, n. 1, p. 1, doi. 10.1002/cmdc.202100434

By:

Dai, Linlin;
Wang, Luyao;
Tan, Cheng;
Cai, Jun;
Shen, Hongsheng;
Zhang, Ting;
Zhi, Shuang;
Yang, Zibo;
Hu, Yunhui;
Zhao, Xiumei;
Li, Dongdong

Publication type:

Article

Emerging Nitric Oxide and Hydrogen Sulfide Releasing Carriers for Skin Wound Healing Therapy.

Published in:

ChemMedChem, 2022, v. 17, n. 1, p. 1, doi. 10.1002/cmdc.202100429

By:

Pinto, Rosana V.;
Carvalho, Sílvia;
Antunes, Fernando;
Pires, João;
Pinto, Moisés L.

Publication type:

Article

Dihydropyridine Lactam Analogs Targeting BET Bromodomains.

Published in:

ChemMedChem, 2022, v. 17, n. 1, p. 1, doi. 10.1002/cmdc.202100407

By:

Jiang, Jiewei;
Sigua, Logan H.;
Chan, Alice;
Kalra, Prakriti;
Pomerantz, William C.K.;
Schönbrunn, Ernst;
Qi, Jun;
Georg, Gunda I.

Publication type:

Article

Inhibition of JMJD6 by 2‐Oxoglutarate Mimics.

Published in:

ChemMedChem, 2022, v. 17, n. 1, p. 1, doi. 10.1002/cmdc.202100398

By:

Islam, Md. Sailful;
Thinnes, Cyrille C.;
Holt‐Martyn, James P.;
Chowdhury, Rasheduzzaman;
McDonough, Michael A.;
Schofield, Christopher J.

Publication type:

Article