Works matching IS 18607179 AND DT 2022 AND VI 17 AND IP 9

Results: 17

Front Cover: Balancing Histone Deacetylase (HDAC) Inhibition and Drug‐likeness: Biological and Physicochemical Evaluation of Class I Selective HDAC Inhibitors (ChemMedChem 9/2022).

Published in:

ChemMedChem, 2022, v. 17, n. 9, p. 1, doi. 10.1002/cmdc.202200210

By:

Schäker‐Hübner, Linda;
Haschemi, Reza;
Büch, Thomas;
Kraft, Fabian B.;
Brumme, Birke;
Schöler, Andrea;
Jenke, Robert;
Meiler, Jens;
Aigner, Achim;
Bendas, Gerd;
Hansen, Finn K.

Publication type:

Article

Puckering the Planar Landscape of Fragments: Design and Synthesis of a 3D Cyclobutane Fragment Library.

Published in:

ChemMedChem, 2022, v. 17, n. 9, p. 1, doi. 10.1002/cmdc.202200113

By:

Hamilton, David J.;
Beemsterboer, Marieke;
Carter, Caroline M.;
Elsayed, Jasmina;
Huiberts, Rilana E. M.;
Klein, Hanna F.;
O'Brien, Peter;
de Esch, Iwan J. P.;
Wijtmans, Maikel

Publication type:

Article

Effect of meso Positioned Substituents on the Stability and Photodynamic Activity of Lipid‐Membrane‐Incorporated Porphyrin Derivatives.

Published in:

ChemMedChem, 2022, v. 17, n. 9, p. 1, doi. 10.1002/cmdc.202200070

By:

Nishimura, Kotaro;
Shimada, Risako;
Yamana, Keita;
Kawasaki, Riku;
Nakaya, Toshimi;
Ikeda, Atsushi

Publication type:

Article

Multidrug Idebenone/Naproxen Co‐loaded Aspasomes for Significant in vivo Anti‐inflammatory Activity.

Published in:

ChemMedChem, 2022, v. 17, n. 9, p. 1, doi. 10.1002/cmdc.202200067

By:

d'Avanzo, Nicola;
Cristiano, Maria Chiara;
Di Marzio, Luisa;
Bruno, Maria Chiara;
Paolino, Donatella;
Celia, Christian;
Fresta, Massimo

Publication type:

Article

Design, Synthesis and X‐Ray Structural Studies of Potent HIV‐1 Protease Inhibitors Containing C‐4 Substituted Tricyclic Hexahydro‐Furofuran Derivatives as P2 Ligands.

Published in:

ChemMedChem, 2022, v. 17, n. 9, p. 1, doi. 10.1002/cmdc.202200058

By:

Ghosh, Arun K.;
Kovela, Satish;
Sharma, Ashish;
Shahabi, Dana;
Ghosh, Ajay K.;
Hopkins, Denver R.;
Yadav, Monika;
Johnson, Megan E.;
Agniswamy, Johnson;
Wang, Yuan‐Fang;
Hattori, Shin‐Ichiro;
Higashi‐Kuwata, Nobuyo;
Aoki, Manabu;
Amano, Masayuki;
Weber, Irene T.;
Mitsuya, Hiroaki

Publication type:

Article

Desorption Electrospray Ionization Mass Spectrometry Assay for Label‐Free Characterization of SULT2B1b Enzyme Kinetics.

Published in:

ChemMedChem, 2022, v. 17, n. 9, p. 1, doi. 10.1002/cmdc.202200043

By:

Kulathunga, Samadhi C.;
Morato, Nicolás M.;
Zhou, Qing;
Cooks, R. Graham;
Mesecar, Andrew D.

Publication type:

Article

Cyclobutanes in Small‐Molecule Drug Candidates.

Published in:

ChemMedChem, 2022, v. 17, n. 9, p. 1, doi. 10.1002/cmdc.202200020

By:

van der Kolk, Marnix R.;
Janssen, Mathilde A. C. H.;
Rutjes, Floris P. J. T.;
Blanco‐Ania, Daniel

Publication type:

Article

Synthesis and in vitro Study of Artemisinin/Synthetic Peroxide‐Based Hybrid Compounds against SARS‐CoV‐2 and Cancer.

Published in:

ChemMedChem, 2022, v. 17, n. 9, p. 1, doi. 10.1002/cmdc.202200005

By:

Herrmann, Lars;
Yaremenko, Ivan A.;
Çapcı, Aysun;
Struwe, Julia;
Tailor, Dhanir;
Dheeraj, Arpit;
Hodek, Jan;
Belyakova, Yulia Yu.;
Radulov, Peter S.;
Weber, Jan;
Malhotra, Sanjay V.;
Terent'ev, Alexander O.;
Ackermann, Lutz;
Tsogoeva, Svetlana B.

Publication type:

Article

Mass Spectrometric Assays Reveal Discrepancies in Inhibition Profiles for the SARS‐CoV‐2 Papain‐Like Protease.

Published in:

ChemMedChem, 2022, v. 17, n. 9, p. 1, doi. 10.1002/cmdc.202200016

By:

Brewitz, Lennart;
Kamps, Jos J. A. G.;
Lukacik, Petra;
Strain‐Damerell, Claire;
Zhao, Yilin;
Tumber, Anthony;
Malla, Tika R.;
Orville, Allen M.;
Walsh, Martin A.;
Schofield, Christopher J.

Publication type:

Article

Modification of Biphenolic Anti‐Bacterial to Achieve Broad‐Spectrum Activity.

Published in:

ChemMedChem, 2022, v. 17, n. 9, p. 1, doi. 10.1002/cmdc.202100783

By:

Ochoa, Cristian;
Roenfanz, Hanna F.;
Kozlowski, Marisa C.

Publication type:

Article

Near‐Infrared Fluorescent Heptamethine Cyanine Dyes for COX‐2 Targeted Photodynamic Cancer Therapy.

Published in:

ChemMedChem, 2022, v. 17, n. 9, p. 1, doi. 10.1002/cmdc.202100780

By:

Wangngae, Sirilak;
Siriwibool, Siriwalee;
Chansaenpak, Kantapat;
Wet‐osot, Sirawit;
Lai, Rung‐Yi;
Kamkaew, Anyanee

Publication type:

Article

Nanoparticles‐Mediated CRISPR/Cas Gene Editing Delivery System.

Published in:

ChemMedChem, 2022, v. 17, n. 9, p. 1, doi. 10.1002/cmdc.202100777

By:

Saw, Phei Er;
Cui, Guo‐hui;
Xu, Xiaoding

Publication type:

Article

Hexafluoroisopropyl Carbamates as Selective MAGL and Dual MAGL/FAAH Inhibitors: Biochemical and Physicochemical Properties.

Published in:

ChemMedChem, 2022, v. 17, n. 9, p. 1, doi. 10.1002/cmdc.202100757

By:

Barth, Maximilian;
Rudolph, Stefan;
Kampschulze, Jan;
Meyer zu Vilsendorf, Imke;
Hanekamp, Walburga;
Mulac, Dennis;
Langer, Klaus;
Lehr, Matthias

Publication type:

Article

Balancing Histone Deacetylase (HDAC) Inhibition and Drug‐likeness: Biological and Physicochemical Evaluation of Class I Selective HDAC Inhibitors.

Published in:

ChemMedChem, 2022, v. 17, n. 9, p. 1, doi. 10.1002/cmdc.202100755

By:

Schäker‐Hübner, Linda;
Haschemi, Reza;
Büch, Thomas;
Kraft, Fabian B.;
Brumme, Birke;
Schöler, Andrea;
Jenke, Robert;
Meiler, Jens;
Aigner, Achim;
Bendas, Gerd;
Hansen, Finn K.

Publication type:

Article

Solid State Development and Processing of Pharmaceutical Molecules: Salts, Cocrystals, and Polymorphism. Edited by Michael Gruss.

Published in:: ChemMedChem, 2022, v. 17, n. 9, p. 1, doi. 10.1002/cmdc.202100711
Publication type:: Article

Successful Drug Discovery, Volume 5. Edited by János Fischer, Christian Klein, and Wayne E. Childers.

Published in:

ChemMedChem, 2022, v. 17, n. 9, p. 1, doi. 10.1002/cmdc.202100705

By:

Langer, Thierry;
Bryant, Sharon D.

Publication type:

Article

Synthesis and Evaluation of a Class of Compounds Inhibiting the Growth of Stromal Antigen 2 (STAG2)‐Mutant Ewing Sarcoma Cells.

Published in:

ChemMedChem, 2022, v. 17, n. 9, p. 1, doi. 10.1002/cmdc.202100653

By:

Zhang, Nenggang;
Lin, Keng‐Fu;
Yang, Christian;
Peruski, Scott;
Pati, Debananda;
Gilbertson, Scott R.

Publication type:

Article