Works matching IS 18607179 AND DT 2022 AND VI 17 AND IP 10

Results: 17

Front Cover: Covalent Allosteric Inhibitors of Akt Generated Using a Click Fragment Approach (ChemMedChem 10/2022).

Published in:

ChemMedChem, 2022, v. 17, n. 10, p. 1, doi. 10.1002/cmdc.202200252

By:

van der Westhuizen, Leandi;
Weisner, Jörn;
Taher, Abu;
Landel, Ina;
Quambusch, Lena;
Lindemann, Marius;
Uhlenbrock, Niklas;
Müller, Matthias P.;
Green, Ivan R.;
Pelly, Stephen C.;
Rauh, Daniel;
van Otterlo, Willem A. L.

Publication type:

Article

Adsorption to the Surface of Hemozoin Crystals: Structure‐Based Design and Synthesis of Amino‐Phenoxazine β‐Hematin Inhibitors.

Published in:

ChemMedChem, 2022, v. 17, n. 10, p. 1, doi. 10.1002/cmdc.202200139

By:

Olivier, Tania;
Loots, Leigh;
Kok, Michélle;
de Villiers, Marianne;
Reader, Janette;
Birkholtz, Lyn‐Marié;
Arnott, Gareth E.;
de Villiers, Katherine A.

Publication type:

Article

Engineered Exosomes as a Photosensitizer Delivery Platform for Cancer Photodynamic Therapy.

Published in:

ChemMedChem, 2022, v. 17, n. 10, p. 1, doi. 10.1002/cmdc.202200119

By:

Dao, Anyi;
Kushwaha, Rajesh;
Kumar, Ashish;
Huang, Huaiyi;
Banerjee, Samya

Publication type:

Article

Jumping from Fragment to Drug via Smart Scaffolds.

Published in:

ChemMedChem, 2022, v. 17, n. 10, p. 1, doi. 10.1002/cmdc.202200092

By:

Farahani, Majid D.;
França, Tanos C. C.;
Alapour, Saba;
Shahout, Fatma;
Boulon, Richard;
Iddir, Mustapha;
Maddalena, Michael;
Ayotte, Yann;
LaPlante, Steven R.

Publication type:

Article

Conjugates of Tacrine with Salicylamide as Promising Multitarget Agents for Alzheimer's Disease.

Published in:

ChemMedChem, 2022, v. 17, n. 10, p. 1, doi. 10.1002/cmdc.202200080

By:

Grishchenko, Maria V.;
Makhaeva, Galina F.;
Burgart, Yanina V.;
Rudakova, Elena V.;
Boltneva, Natalia P.;
Kovaleva, Nadezhda V.;
Serebryakova, Olga G.;
Lushchekina, Sofya V.;
Astakhova, Tatiana Y.;
Zhilina, Ekaterina F.;
Shchegolkov, Evgeny V.;
Richardson, Rudy J.;
Saloutin, Victor I.

Publication type:

Article

Disrupting Transcription and Folate Biosynthesis Leads to Synergistic Suppression of Escherichia coli Growth.

Published in:

ChemMedChem, 2022, v. 17, n. 10, p. 1, doi. 10.1002/cmdc.202200075

By:

Chen, Pei‐Hsin;
Sung, Li‐Kang;
Hegemann, Julian D.;
Chu, John

Publication type:

Article

2‐Amino‐4‐aryl‐5‐oxo‐4,5‐dihydropyrano[3,2‐c]chromene‐3‐carbonitriles with Microtubule‐Disruptive, Centrosome‐Declustering, and Antiangiogenic Effects in vitro and in vivo

Published in:

ChemMedChem, 2022, v. 17, n. 10, p. 1, doi. 10.1002/cmdc.202200064

By:

Köhler, Leonhard H. F.;
Reich, Sebastian;
Begemann, Gerrit;
Schobert, Rainer;
Biersack, Bernhard

Publication type:

Article

A Series of Thiadiazolyl‐Benzenesulfonamides Incorporating an Aromatic Tail as Isoform‐Selective, Potent Carbonic Anhydrase II/XII Inhibitors.

Published in:

ChemMedChem, 2022, v. 17, n. 10, p. 1, doi. 10.1002/cmdc.202200056

By:

Banoglu, Erden;
Ercanlı, Taner;
Gür Maz, Tuğçe;
Vullo, Daniela;
Bonardi, Alessandro;
Gratteri, Paola;
Supuran, Claudiu T.

Publication type:

Article

Anthracene‐Walled Acyclic CB[n] Receptors: in vitro and in vivo Binding Properties toward Drugs of Abuse.

Published in:

ChemMedChem, 2022, v. 17, n. 10, p. 1, doi. 10.1002/cmdc.202200046

By:

DiMaggio, Delaney;
Brockett, Adam T.;
Shuster, Michael;
Murkli, Steven;
Zhai, Canjia;
King, David;
O'Dowd, Brona;
Cheng, Ming;
Brady, Kimberly;
Briken, Volker;
Roesch, Matthew R.;
Isaacs, Lyle

Publication type:

Article

Rational Optimization of Dihydropyrimidinone‐Quinoline Hybrids as Plasmodium falciparum Glutathione Reductase Inhibitors.

Published in:

ChemMedChem, 2022, v. 17, n. 10, p. 1, doi. 10.1002/cmdc.202200034

By:

Adigun, Rasheed A.;
Malan, Frederick P.;
Balogun, Mohammed O.;
October, Natasha

Publication type:

Article

Synthesis, in vitro Antileishmanial Efficacy and Hit/Lead Identification of Nitrofurantoin‐Triazole Hybrids.

Published in:

ChemMedChem, 2022, v. 17, n. 10, p. 1, doi. 10.1002/cmdc.202200023

By:

Zuma, Nonkululeko H.;
Aucamp, Janine;
Viljoen, Maryna;
N'Da, David D.

Publication type:

Article

Recent Developments in Porous Silicon Nanovectors with Various Imaging Modalities in the Framework of Theranostics.

Published in:

ChemMedChem, 2022, v. 17, n. 10, p. 1, doi. 10.1002/cmdc.202200004

By:

Qian, Jing;
Wen, Huang;
Tamarov, Konstantin;
Xu, Wujun;
Lehto, Vesa‐Pekka

Publication type:

Article

Design, Synthesis, and Characterization of a Novel Fluoroprobe for Live Human Islet Cell Imaging of Serotonin 5‐HT<sub>1A</sub> Receptor.

Published in:

ChemMedChem, 2022, v. 17, n. 10, p. 1, doi. 10.1002/cmdc.202100759

By:

Garvey, Robert W.;
Lacivita, Enza;
Niso, Mauro;
Duszyńska, Beata;
Harris, Paul E.;
Leopoldo, Marcello

Publication type:

Article

Liraglutide‐Loaded Milk Exosomes Lower Blood Glucose When Given by Sublingual Route.

Published in:

ChemMedChem, 2022, v. 17, n. 10, p. 1, doi. 10.1002/cmdc.202100758

By:

Xu, Mingzhi;
Chen, Gang;
Dong, Yanan;
Yang, Jing;
Liu, Yongxue;
Song, Haijing;
Song, Haifeng;
Wang, Yi

Publication type:

Article

Corrigendum: Self‐Foaming Metal‐Organic Gels Based on Phytic Acid and Their Mechanical, Moldable, and Load‐Bearing Properties.

Published in:

ChemMedChem, 2022, v. 17, n. 10, p. 1, doi. 10.1002/cmdc.202100738

By:

Xiao, Yali;
Gong, Xi;
Zhang, Jianyong

Publication type:

Article

Corrigendum: Design of Trehalose‐Based Amide/Sulfonamide C‐type Lectin Receptor Signaling Compounds.

Published in:

ChemMedChem, 2022, v. 17, n. 10, p. 1, doi. 10.1002/cmdc.202100376

By:

Rasheed, Omer K.;
Buhl, Cassandra;
Evans, Jay T.;
Ryter, Kendal T.

Publication type:

Article

Covalent Allosteric Inhibitors of Akt Generated Using a Click Fragment Approach.

Published in:

ChemMedChem, 2022, v. 17, n. 10, p. 1, doi. 10.1002/cmdc.202100776

By:

van der Westhuizen, Leandi;
Weisner, Jörn;
Taher, Abu;
Landel, Ina;
Quambusch, Lena;
Lindemann, Marius;
Uhlenbrock, Niklas;
Müller, Matthias P.;
Green, Ivan R.;
Pelly, Stephen C.;
Rauh, Daniel;
van Otterlo, Willem A. L.

Publication type:

Article