Works matching IS 18607179 AND DT 2020 AND VI 15 AND IP 24

Results: 23

Cover Feature: Memoirs of the First 50 Years of the European Federation for Medicinal Chemistry (EFMC) (ChemMedChem 24/2020).

Published in:

ChemMedChem, 2020, v. 15, n. 24, p. 2333, doi. 10.1002/cmdc.202000910

By:

Timmerman, Henk

Publication type:

Article

Front Cover: Evaluation of 5H‐Thiazolo[3,2‐α]pyrimidin‐5‐ones as Potential GluN2A PET Tracers (ChemMedChem 24/2020).

Published in:

ChemMedChem, 2020, v. 15, n. 24, p. 2332, doi. 10.1002/cmdc.202000909

By:

He, Yingfang;
Whitehead, David M.;
Briard, Emmanuelle;
Numao, Shin;
Mu, Linjing;
Schibli, Roger;
Ametamey, Simon M.;
Auberson, Yves P.

Publication type:

Article

Trends in Drug Discovery over Five Decades – The European Federation for Medicinal Chemistry International Symposium on Medicinal Chemistry (EFMC−ISMC).

Published in:

ChemMedChem, 2020, v. 15, n. 24, p. 2352, doi. 10.1002/cmdc.202000840

By:

Differding, Edmond

Publication type:

Article

The Young Scientists Network: How the European Federation for Medicinal Chemistry (EFMC) Became Young Again.

Published in:

ChemMedChem, 2020, v. 15, n. 24, p. 2359, doi. 10.1002/cmdc.202000794

By:

Goncharenko, Kristina;
Mari, Michele;
Auberson, Yves P.;
Matagne, Brieuc

Publication type:

Article

50 Years European Federation for Medicinal Chemistry (EFMC) – The Ascent of Medicinal Chemistry in Europe.

Published in:

ChemMedChem, 2020, v. 15, n. 24, p. 2338, doi. 10.1002/cmdc.202000691

By:

Differding, Edmond

Publication type:

Article

Benzylaminoethylureido‐Tailed Benzenesulfonamides Show Potent Inhibitory Activity against Bacterial Carbonic Anhydrases.

Published in:

ChemMedChem, 2020, v. 15, n. 24, p. 2444, doi. 10.1002/cmdc.202000680

By:

Ali, Majid;
Angeli, Andrea;
Bozdag, Murat;
Carta, Fabrizio;
Capasso, Clemente;
Farooq, Umar;
Supuran, Claudiu T.

Publication type:

Article

Co‐staining of KCa3.1 Channels in NSCLC Cells with a Small‐Molecule Fluorescent Probe and Antibody‐Based Indirect Immunofluorescence.

Published in:

ChemMedChem, 2020, v. 15, n. 24, p. 2462, doi. 10.1002/cmdc.202000652

By:

Brömmel, Kathrin;
Maskri, Sarah;
Bulk, Etmar;
Pethő, Zoltan;
Rieke, Marius;
Budde, Thomas;
Koch, Oliver;
Schwab, Albrecht;
Wünsch, Bernhard

Publication type:

Article

The European Federation for Medicinal Chemistry (EFMC) Best Practice Initiative: Validating Chemical Probes.

Published in:

ChemMedChem, 2020, v. 15, n. 24, p. 2388, doi. 10.1002/cmdc.202000597

By:

Quancard, Jean;
Cox, Brian;
Finsinger, Dirk;
Guéret, Stéphanie M.;
Hartung, Ingo V.;
Koolman, Hannes F.;
Messinger, Josef;
Sbardella, Gianluca;
Laufer, Stefan

Publication type:

Article

Activating Effect of 3‐Benzylidene Oxindoles on AMPK: From Computer Simulation to High‐Content Screening.

Published in:

ChemMedChem, 2020, v. 15, n. 24, p. 2521, doi. 10.1002/cmdc.202000579

By:

Novikova, Daria S.;
Grigoreva, Tatyana A.;
Ivanov, Gleb S.;
Melino, Gerry;
Barlev, Nickolai A.;
Tribulovich, Vyacheslav G.

Publication type:

Article

Memoirs of the First 50 Years of the European Federation for Medicinal Chemistry (EFMC).

Published in:

ChemMedChem, 2020, v. 15, n. 24, p. 2363, doi. 10.1002/cmdc.202000576

By:

Timmerman, Henk

Publication type:

Article

Targeted Protein Degradation as a Promising Tool for Epigenetic Upregulation of Fetal Hemoglobin.

Published in:

ChemMedChem, 2020, v. 15, n. 24, p. 2436, doi. 10.1002/cmdc.202000574

By:

J. Verheul, Thijs C.;
Trinh, Van Tuan;
Vázquez, Olalla;
Philipsen, Sjaak

Publication type:

Article

Deliberately Losing Control of C−H Activation Processes in the Design of Small‐Molecule‐Fragment Arrays Targeting Peroxisomal Metabolism.

Published in:

ChemMedChem, 2020, v. 15, n. 24, p. 2513, doi. 10.1002/cmdc.202000543

By:

Khan Tareque, Raysa;
Hassell‐Hart, Storm;
Krojer, Tobias;
Bradley, Anthony;
Velupillai, Srikannathasan;
Talon, Romain;
Fairhead, Michael;
Day, Iain J.;
Bala, Kamlesh;
Felix, Robert;
Kemmitt, Paul D.;
Brennan, Paul;
Delft, Frank;
Díaz Sáez, Laura;
Huber, Kilian;
Spencer, John

Publication type:

Article

Alternating Cationic‐Hydrophobic Peptide/Peptoid Hybrids: Influence of Hydrophobicity on Antibacterial Activity and Cell Selectivity.

Published in:

ChemMedChem, 2020, v. 15, n. 24, p. 2544, doi. 10.1002/cmdc.202000526

By:

Frederiksen, Nicki;
Hansen, Paul R.;
Zabicka, Dorota;
Tomczak, Magdalena;
Urbas, Malgorzata;
Domraceva, Ilona;
Björkling, Fredrik;
Franzyk, Henrik

Publication type:

Article

Rational Design of Azastatin as a Potential ADC Payload with Reduced Bystander Killing.

Published in:

ChemMedChem, 2020, v. 15, n. 24, p. 2500, doi. 10.1002/cmdc.202000497

By:

Hartmann, Rafael W.;
Fahrner, Raphael;
Shevshenko, Denys;
Fyrknäs, Mårten;
Larsson, Rolf;
Lehmann, Fredrik;
Odell, Luke R.

Publication type:

Article

Broad‐Spectrum Flavivirus Inhibitors: a Medicinal Chemistry Point of View.

Published in:

ChemMedChem, 2020, v. 15, n. 24, p. 2391, doi. 10.1002/cmdc.202000464

By:

Felicetti, Tommaso;
Manfroni, Giuseppe;
Cecchetti, Violetta;
Cannalire, Rolando

Publication type:

Article

MedChemTrain e‐School 2020: Event Highlights and Insights into Virtual Symposium Organization.

Published in:

ChemMedChem, 2020, v. 15, n. 24, p. 2562, doi. 10.1002/cmdc.202000450

By:

Ramilo‐Gomes, Filipa;
António, João P. M.;
Mendes, Maria Inês P.;
Gomes, Rafael F. A.

Publication type:

Article

Synthesis of Novel Nitroxoline Analogs with Potent Cathepsin B Exopeptidase Inhibitory Activity.

Published in:

ChemMedChem, 2020, v. 15, n. 24, p. 2477, doi. 10.1002/cmdc.202000402

By:

Van de Walle, Tim;
Briand, Marina;
Mitrović, Ana;
Sosič, Izidor;
Gobec, Stanislav;
Kos, Janko;
Persoons, Leentje;
Daelemans, Dirk;
De Jonghe, Steven;
Ubiparip, Zorica;
Desmet, Tom;
Van Hecke, Kristof;
Mangelinckx, Sven;
D'hooghe, Matthias

Publication type:

Article

Radiosynthesis and Preclinical Investigation of 11C‐Labelled 3‐(4,5‐Diphenyl‐1,3‐oxazol‐2‐yl)propanal Oxime ([11C]SZV 1287).

Published in:

ChemMedChem, 2020, v. 15, n. 24, p. 2470, doi. 10.1002/cmdc.202000389

By:

Forgács, Viktória;
Németh, Enikő;
Gyuricza, Barbara;
Kis, Adrienn;
Szabó, Judit P.;
Mikecz, Pál;
Mátyus, Péter;
Helyes, Zsuzsanna;
Horváth, Ádám István;
Kálai, Tamás;
Trencsényi, György;
Fekete, Anikó;
Szikra, Dezső

Publication type:

Article

Evaluation of 5H‐Thiazolo[3,2‐α]pyrimidin‐5‐ones as Potential GluN2A PET Tracers.

Published in:

ChemMedChem, 2020, v. 15, n. 24, p. 2448, doi. 10.1002/cmdc.202000340

By:

He, Yingfang;
Whitehead, David M.;
Briard, Emmanuelle;
Numao, Shin;
Mu, Linjing;
Schibli, Roger;
Ametamey, Simon M.;
Auberson, Yves P.

Publication type:

Article

Recent Advancement in the Search of Innovative Antiprotozoal Agents Targeting Trypanothione Metabolism.

Published in:

ChemMedChem, 2020, v. 15, n. 24, p. 2420, doi. 10.1002/cmdc.202000325

By:

Saccoliti, Francesco;
Di Santo, Roberto;
Costi, Roberta

Publication type:

Article

Concise Synthesis of 1,4‐Benzoquinone‐Based Natural Products as Mitochondrial Complex I Substrates and Substrate‐Based Inhibitors.

Published in:

ChemMedChem, 2020, v. 15, n. 24, p. 2491, doi. 10.1002/cmdc.202000307

By:

Han, Zhenyu;
Angerer, Heike;
Bischoff, Iris;
Qin, Yihan;
Stegmann, Dennis;
Tuz, Karina;
Fritz, Günter;
Juarez, Oscar;
Fürst, Robert;
Lashley, Dana;
Nasiri, Hamid R.

Publication type:

Article

Design, Synthesis, and in vitro Evaluation of P2X7 Antagonists.

Published in:

ChemMedChem, 2020, v. 15, n. 24, p. 2530, doi. 10.1002/cmdc.202000303

By:

T. Pournara, Dimitra;
Durner, Anna;
Kritsi, Eftichia;
Papakostas, Alexios;
Zoumpoulakis, Panagiotis;
Nicke, Annette;
Koufaki, Maria

Publication type:

Article

EFMC, Medicinal Chemistry and Chemical Biology in Europe.

Published in:

ChemMedChem, 2020, v. 15, n. 24, p. 2334, doi. 10.1002/cmdc.202000178

By:

Auberson, Yves P.

Publication type:

Article

Works matching IS 18607179 AND DT 2020 AND VI 15 AND IP 24

Cover Feature: Memoirs of the First 50 Years of the European Federation for Medicinal Chemistry (EFMC) (ChemMedChem 24/2020).

Front Cover: Evaluation of 5H‐Thiazolo[3,2‐α]pyrimidin‐5‐ones as Potential GluN2A PET Tracers (ChemMedChem 24/2020).

Trends in Drug Discovery over Five Decades – The European Federation for Medicinal Chemistry International Symposium on Medicinal Chemistry (EFMC−ISMC).

The Young Scientists Network: How the European Federation for Medicinal Chemistry (EFMC) Became Young Again.

50 Years European Federation for Medicinal Chemistry (EFMC) – The Ascent of Medicinal Chemistry in Europe.

Benzylaminoethylureido‐Tailed Benzenesulfonamides Show Potent Inhibitory Activity against Bacterial Carbonic Anhydrases.

Co‐staining of K<sub>Ca</sub>3.1 Channels in NSCLC Cells with a Small‐Molecule Fluorescent Probe and Antibody‐Based Indirect Immunofluorescence.

The European Federation for Medicinal Chemistry (EFMC) Best Practice Initiative: Validating Chemical Probes.

Activating Effect of 3‐Benzylidene Oxindoles on AMPK: From Computer Simulation to High‐Content Screening.

Memoirs of the First 50 Years of the European Federation for Medicinal Chemistry (EFMC).

Targeted Protein Degradation as a Promising Tool for Epigenetic Upregulation of Fetal Hemoglobin.

Deliberately Losing Control of C−H Activation Processes in the Design of Small‐Molecule‐Fragment Arrays Targeting Peroxisomal Metabolism.

Alternating Cationic‐Hydrophobic Peptide/Peptoid Hybrids: Influence of Hydrophobicity on Antibacterial Activity and Cell Selectivity.

Rational Design of Azastatin as a Potential ADC Payload with Reduced Bystander Killing.

Broad‐Spectrum Flavivirus Inhibitors: a Medicinal Chemistry Point of View.

MedChemTrain e‐School 2020: Event Highlights and Insights into Virtual Symposium Organization.

Synthesis of Novel Nitroxoline Analogs with Potent Cathepsin B Exopeptidase Inhibitory Activity.

Radiosynthesis and Preclinical Investigation of <sup>11</sup>C‐Labelled 3‐(4,5‐Diphenyl‐1,3‐oxazol‐2‐yl)propanal Oxime ([<sup>11</sup>C]SZV 1287).

Evaluation of 5H‐Thiazolo[3,2‐α]pyrimidin‐5‐ones as Potential GluN2A PET Tracers.

Recent Advancement in the Search of Innovative Antiprotozoal Agents Targeting Trypanothione Metabolism.

Concise Synthesis of 1,4‐Benzoquinone‐Based Natural Products as Mitochondrial Complex I Substrates and Substrate‐Based Inhibitors.

Design, Synthesis, and in vitro Evaluation of P2X7 Antagonists.

EFMC, Medicinal Chemistry and Chemical Biology in Europe.