Works matching IS 18607179 AND DT 2020 AND VI 15 AND IP 14

Results: 14

Front Cover: Synthesis and Biological Screening of New Lawson Derivatives as Selective Substrate‐Based Inhibitors of Cytochrome bo<sub>3</sub> Ubiquinol Oxidase from Escherichia coli (ChemMedChem 14/2020).

Published in:

ChemMedChem, 2020, v. 15, n. 14, p. 1243, doi. 10.1002/cmdc.202000481

By:

Elamri, Isam;
Radloff, Melanie;
Hohmann, Katharina F.;
Nimbarte, Vijaykumar D.;
Nasiri, Hamid R.;
Bolte, Michael;
Safarian, Schara;
Michel, Hartmut;
Schwalbe, Harald

Publication type:

Article

Small‐Molecule Inhibitors Targeting Sterol 14α‐Demethylase (CYP51): Synthesis, Molecular Modelling and Evaluation Against Candida albicans.

Published in:

ChemMedChem, 2020, v. 15, n. 14, p. 1294, doi. 10.1002/cmdc.202000250

By:

Binjubair, Faizah A.;
Parker, Josie E.;
Warrilow, Andrew G.;
Puri, Kalika;
Braidley, Peter J.;
Tatar, Esra;
Kelly, Steven L.;
Kelly, Diane E.;
Simons, Claire

Publication type:

Article

Pharmacological Profile and Molecular Modeling of Cyclic Opioid Analogues Incorporating Various Phenylalanine Derivatives.

Published in:

ChemMedChem, 2020, v. 15, n. 14, p. 1322, doi. 10.1002/cmdc.202000248

By:

Adamska‐Bartłomiejczyk, Anna;
Lipiński, Piotr F. J.;
Piekielna‐Ciesielska, Justyna;
Kluczyk, Alicja;
Janecka, Anna

Publication type:

Article

Controlling PROTACs with Light.

Published in:

ChemMedChem, 2020, v. 15, n. 14, p. 1258, doi. 10.1002/cmdc.202000249

By:

Verma, Shreya;
Manna, Debasish

Publication type:

Article

Divergent Synthesis of Novel Cylindrocyclophanes that Inhibit Methicillin‐Resistant Staphylococcus aureus (MRSA).

Published in:

ChemMedChem, 2020, v. 15, n. 14, p. 1289, doi. 10.1002/cmdc.202000179

By:

Freudenreich, Julien J.;
Bartlett, Sean;
Robertson, Naomi S.;
Kidd, Sarah L.;
Forrest, Suzie;
Sore, Hannah F.;
Galloway, Warren R. J. D.;
Welch, Martin;
Spring, David R.

Publication type:

Article

Plumbagin‐Serum Albumin Interaction: Spectral, Electrochemical, Structure‐Binding Analysis, Antiproliferative and Cell Signaling Aspects with Implications for Anticancer Therapy.

Published in:

ChemMedChem, 2020, v. 15, n. 14, p. 1338, doi. 10.1002/cmdc.202000157

By:

Chrastina, Adrian;
Welsh, John;
Rondeau, Gaelle;
Abedinpour, Parisa;
Borgström, Per;
Baron, Véronique T.

Publication type:

Article

Design, Synthesis and Biological Evaluation of Highly Potent Simplified Archazolids.

Published in:

ChemMedChem, 2020, v. 15, n. 14, p. 1348, doi. 10.1002/cmdc.202000154

By:

Rivière, Solenne;
Vielmuth, Christin;
Ennenbach, Christiane;
Abdelrahman, Aliaa;
Lemke, Carina;
Gütschow, Michael;
Müller, Christa E.;
Menche, Dirk

Publication type:

Article

Structure‐Activity Relationship of Phenylpyrazolones against Trypanosoma cruzi.

Published in:

ChemMedChem, 2020, v. 15, n. 14, p. 1310, doi. 10.1002/cmdc.202000136

By:

Sijm, Maarten;
Sterk, Geert Jan;
Caljon, Guy;
Maes, Louis;
Esch, Iwan J. P.;
Leurs, Rob

Publication type:

Article

Design and Synthesis of Fluorescent Methylphenidate Analogues for a FRET‐Based Assay of Synapsin III Binding.

Published in:

ChemMedChem, 2020, v. 15, n. 14, p. 1330, doi. 10.1002/cmdc.202000128

By:

Casiraghi, Andrea;
Longhena, Francesca;
Straniero, Valentina;
Faustini, Gaia;
Newman, Amy H.;
Bellucci, Arianna;
Valoti, Ermanno

Publication type:

Article

α‐Triazolylboronic Acids: A Promising Scaffold for Effective Inhibitors of KPCs.

Published in:

ChemMedChem, 2020, v. 15, n. 14, p. 1283, doi. 10.1002/cmdc.202000126

By:

Introvigne, Maria Luisa;
Taracila, Magdalena A.;
Prati, Fabio;
Caselli, Emilia;
Bonomo, Robert A.

Publication type:

Article

Iminodiacetic Acid as a Novel Metal‐Binding Pharmacophore for New Delhi Metallo‐β‐lactamase Inhibitor Development.

Published in:

ChemMedChem, 2020, v. 15, n. 14, p. 1272, doi. 10.1002/cmdc.202000123

By:

Chen, Allie Y.;
Thomas, Caitlyn A.;
Thomas, Pei W.;
Yang, Kundi;
Cheng, Zishuo;
Fast, Walter;
Crowder, Michael W.;
Cohen, Seth M.

Publication type:

Article

O‐GlcNAcase: Emerging Mechanism, Substrate Recognition and Small‐Molecule Inhibitors.

Published in:

ChemMedChem, 2020, v. 15, n. 14, p. 1244, doi. 10.1002/cmdc.202000077

By:

Elbatrawy, Ahmed A.;
Kim, Eun Ju;
Nam, Ghilsoo

Publication type:

Article

Biological Characterization, Mechanistic Investigation and Structure‐Activity Relationships of Chemically Stable TLR2 Antagonists.

Published in:

ChemMedChem, 2020, v. 15, n. 14, p. 1364, doi. 10.1002/cmdc.202000060

By:

Bermudez, Marcel;
Grabowski, Maria;
Murgueitio, Manuela S.;
Tiemann, Markus;
Varga, Péter;
Rudolf, Thomas;
Wolber, Gerhard;
Weindl, Günther;
Rademann, Jörg

Publication type:

Article

Synthesis and Biological Screening of New Lawson Derivatives as Selective Substrate‐Based Inhibitors of Cytochrome bo<sub>3</sub> Ubiquinol Oxidase from Escherichia coli.

Published in:

ChemMedChem, 2020, v. 15, n. 14, p. 1262, doi. 10.1002/cmdc.201900707

By:

Elamri, Isam;
Radloff, Melanie;
Hohmann, Katharina F.;
Nimbarte, Vijaykumar D.;
Nasiri, Hamid R.;
Bolte, Michael;
Safarian, Schara;
Michel, Hartmut;
Schwalbe, Harald

Publication type:

Article