Works matching IS 18607179 AND DT 2020 AND VI 15 AND IP 18

Results: 11

Synthesis of 2‐Organylchalcogenopheno[2,3‐b]pyridines from Elemental Chalcogen and NaBH4/PEG‐400 as a Reducing System: Antioxidant and Antinociceptive Properties.

Published in:

ChemMedChem, 2020, v. 15, n. 18, p. 1741, doi. 10.1002/cmdc.202000358

By:

Peglow, Thiago J.;
Bartz, Ricardo H.;
Martins, Carolina C.;
Belladona, Andrei L.;
Luchese, Cristiane;
Wilhelm, Ethel A.;
Schumacher, Ricardo F.;
Perin, Gelson

Publication type:

Article

A Potent Mimetic of the Siglec‐8 Ligand 6'‐Sulfo‐Sialyl Lewisx.

Published in:

ChemMedChem, 2020, v. 15, n. 18, p. 1680, doi. 10.1002/cmdc.202000649

By:

Kroezen, Blijke S.;
Conti, Gabriele;
Girardi, Benedetta;
Cramer, Jonathan;
Jiang, Xiaohua;
Rabbani, Said;
Müller, Jennifer;
Kokot, Maja;
Luisoni, Enrico;
Ricklin, Daniel;
Schwardt, Oliver;
Ernst, Beat

Publication type:

Article

Selective Fragments for the CREBBP Bromodomain Identified from an Encoded Self‐assembly Chemical Library.

Published in:

ChemMedChem, 2020, v. 15, n. 18, p. 1752, doi. 10.1002/cmdc.202000528

By:

Catalano, Marco;
Moroglu, Mustafa;
Balbi, Petra;
Mazzieri, Federica;
Clayton, James;
Andrews, Katrina H.;
Bigatti, Martina;
Scheuermann, Jörg;
Conway, Stuart J.;
Neri, Dario

Publication type:

Article

A Potent Mimetic of the Siglec‐8 Ligand 6'‐Sulfo‐Sialyl Lewisx.

Published in:

ChemMedChem, 2020, v. 15, n. 18, p. 1706, doi. 10.1002/cmdc.202000417

By:

Kroezen, Blijke S.;
Conti, Gabriele;
Girardi, Benedetta;
Cramer, Jonathan;
Jiang, Xiaohua;
Rabbani, Said;
Müller, Jennifer;
Kokot, Maja;
Luisoni, Enrico;
Ricklin, Daniel;
Schwardt, Oliver;
Ernst, Beat

Publication type:

Article

ACE2, the Receptor that Enables Infection by SARS‐CoV‐2: Biochemistry, Structure, Allostery and Evaluation of the Potential Development of ACE2 Modulators.

Published in:

ChemMedChem, 2020, v. 15, n. 18, p. 1682, doi. 10.1002/cmdc.202000368

By:

Gross, Lissy Z. F.;
Sacerdoti, Mariana;
Piiper, Albrecht;
Zeuzem, Stefan;
Leroux, Alejandro E.;
Biondi, Ricardo M.

Publication type:

Article

Structural Consequences of the 1,2,3‐Triazole as an Amide Bioisostere in Analogues of the Cystic Fibrosis Drugs VX‐809 and VX‐770.

Published in:

ChemMedChem, 2020, v. 15, n. 18, p. 1681, doi. 10.1002/cmdc.202000650

By:

Doiron, Jake E.;
Le, Christina A.;
Bacsa, John;
Breton, Gary W.;
Martin, Kenneth L.;
Aller, Stephen G.;
Turlington, Mark

Publication type:

Article

Kiss1R Identification and Biodistribution Analysis Employing a Western Ligand Blot and Ligand‐Derivative Stain with a FITC‐Kisspeptin Derivative.

Published in:

ChemMedChem, 2020, v. 15, n. 18, p. 1699, doi. 10.1002/cmdc.202000356

By:

Hasegawa, Koki;
Maedomari, Rika;
Sato, Younosuke;
Gotoh, Kumiko;
Kudoh, Shinji;
Kojima, Akihiro;
Okada, Seiji;
Ito, Takaaki

Publication type:

Article

Optimization of 4‐Substituted Benzenesulfonamide Scaffold To Reverse Acinetobacter baumannii Serum‐Adaptive Efflux Associated Antibiotic Tolerance.

Published in:

ChemMedChem, 2020, v. 15, n. 18, p. 1731, doi. 10.1002/cmdc.202000328

By:

Chojnacki, Michaelle;
Cao, Xufeng;
Young, Mikaeel;
Fritz, Rebecca N.;
Dunman, Paul M.;
Flaherty, Daniel P.

Publication type:

Article

Rationally Designed Polypharmacology: α‐Helix Mimetics as Dual Inhibitors of the Oncoproteins Mcl‐1 and HDM2.

Published in:

ChemMedChem, 2020, v. 15, n. 18, p. 1691, doi. 10.1002/cmdc.202000278

By:

Conlon, Ivie L.;
Drennen, Brandon;
Lanning, Maryanna E.;
Hughes, Samuel;
Rothhaas, Rebecca;
Wilder, Paul T.;
MacKerell, Alexander D.;
Fletcher, Steven

Publication type:

Article

Structural Consequences of the 1,2,3‐Triazole as an Amide Bioisostere in Analogues of the Cystic Fibrosis Drugs VX‐809 and VX‐770.

Published in:

ChemMedChem, 2020, v. 15, n. 18, p. 1720, doi. 10.1002/cmdc.202000220

By:

Doiron, Jake E.;
Le, Christina A.;
Bacsa, John;
Breton, Gary W.;
Martin, Kenneth L.;
Aller, Stephen G.;
Turlington, Mark

Publication type:

Article

4‐Fluorobenzylpiperazine‐Containing Derivatives as Efficient Inhibitors of Mushroom Tyrosinase.

Published in:

ChemMedChem, 2020, v. 15, n. 18, p. 1757, doi. 10.1002/cmdc.202000125

By:

Vittorio, Serena;
Ielo, Laura;
Mirabile, Salvatore;
Gitto, Rosaria;
Fais, Antonella;
Floris, Sonia;
Rapisarda, Antonio;
Germanò, Maria Paola;
De Luca, Laura

Publication type:

Article

Works matching IS 18607179 AND DT 2020 AND VI 15 AND IP 18

Synthesis of 2‐Organylchalcogenopheno[2,3‐b]pyridines from Elemental Chalcogen and NaBH<sub>4</sub>/PEG‐400 as a Reducing System: Antioxidant and Antinociceptive Properties.

A Potent Mimetic of the Siglec‐8 Ligand 6'‐Sulfo‐Sialyl Lewis<sup>x</sup>.

Selective Fragments for the CREBBP Bromodomain Identified from an Encoded Self‐assembly Chemical Library.

A Potent Mimetic of the Siglec‐8 Ligand 6'‐Sulfo‐Sialyl Lewis<sup>x</sup>.

ACE2, the Receptor that Enables Infection by SARS‐CoV‐2: Biochemistry, Structure, Allostery and Evaluation of the Potential Development of ACE2 Modulators.

Structural Consequences of the 1,2,3‐Triazole as an Amide Bioisostere in Analogues of the Cystic Fibrosis Drugs VX‐809 and VX‐770.

Kiss1R Identification and Biodistribution Analysis Employing a Western Ligand Blot and Ligand‐Derivative Stain with a FITC‐Kisspeptin Derivative.

Optimization of 4‐Substituted Benzenesulfonamide Scaffold To Reverse Acinetobacter baumannii Serum‐Adaptive Efflux Associated Antibiotic Tolerance.

Rationally Designed Polypharmacology: α‐Helix Mimetics as Dual Inhibitors of the Oncoproteins Mcl‐1 and HDM2.

Structural Consequences of the 1,2,3‐Triazole as an Amide Bioisostere in Analogues of the Cystic Fibrosis Drugs VX‐809 and VX‐770.

4‐Fluorobenzylpiperazine‐Containing Derivatives as Efficient Inhibitors of Mushroom Tyrosinase.