Works matching IS 18607179 AND DT 2020 AND VI 15 AND IP 16

Results: 14

Cover Feature: Synthesis and Antibacterial Activity of New N‐Alkylammonium and Carbonate‐Triazole Derivatives within Desosamine of 14‐ and 15‐Membered Lactone Macrolides (ChemMedChem 16/2020).

Published in:

ChemMedChem, 2020, v. 15, n. 16, p. 1498, doi. 10.1002/cmdc.202000578

By:

Janas, Anna;
Pecyna, Paulina;
Gajecka, Marzena;
Bartl, Franz;
Przybylski, Piotr

Publication type:

Article

Front Cover: Pentathiepins: A Novel Class of Glutathione Peroxidase 1 Inhibitors that Induce Oxidative Stress, Loss of Mitochondrial Membrane Potential and Apoptosis in Human Cancer Cells (ChemMedChem 16/2020).

Published in:

ChemMedChem, 2020, v. 15, n. 16, p. 1497, doi. 10.1002/cmdc.202000577

By:

Behnisch‐Cornwell, Steven;
Bandaru, Siva Sankar Murthy;
Napierkowski, Martin;
Wolff, Lisa;
Zubair, Muhammad;
Urbainsky, Claudia;
Lillig, Christopher;
Schulzke, Carola;
Bednarski, Patrick J.

Publication type:

Article

Exploring Proprotein Convertase Subtilisin/Kexin 9 (PCSK9) Autoproteolysis Process by Molecular Simulations: Hints for Drug Design.

Published in:

ChemMedChem, 2020, v. 15, n. 16, p. 1601, doi. 10.1002/cmdc.202000431

By:

Sgrignani, Jacopo;
Fassi, Enrico M. A.;
Lammi, Carmen;
Roda, Gabriella;
Grazioso, Giovanni

Publication type:

Article

Peptidyl Vinyl Ketone Irreversible Inhibitors of Rhodesain: Modifications of the P2 Fragment.

Published in:

ChemMedChem, 2020, v. 15, n. 16, p. 1552, doi. 10.1002/cmdc.202000360

By:

Maiorana, Santina;
Ettari, Roberta;
Previti, Santo;
Amendola, Giorgio;
Wagner, Annika;
Cosconati, Sandro;
Hellmich, Ute A.;
Schirmeister, Tanja;
Zappalà, Maria

Publication type:

Article

A Primary Evaluation of Potential Small‐Molecule Inhibitors of the Astacin Metalloproteinase Ovastacin, a Novel Drug Target in Female Infertility Treatment.

Published in:

ChemMedChem, 2020, v. 15, n. 16, p. 1499, doi. 10.1002/cmdc.202000397

By:

Körschgen, Hagen;
Jäger, Christian;
Tan, Kathrin;
Buchholz, Mirko;
Stöcker, Walter;
Ramsbeck, Daniel

Publication type:

Article

First‐Generation Bispidine Chelators for <sup>213</sup>Bi<sup>III</sup> Radiopharmaceutical Applications.

Published in:

ChemMedChem, 2020, v. 15, n. 16, p. 1591, doi. 10.1002/cmdc.202000361

By:

Bruchertseifer, Frank;
Comba, Peter;
Martin, Bodo;
Morgenstern, Alfred;
Notni, Johannes;
Starke, Miriam;
Wadepohl, Hubert

Publication type:

Article

Short Photoswitchable Antibacterial Peptides.

Published in:

ChemMedChem, 2020, v. 15, n. 16, p. 1505, doi. 10.1002/cmdc.202000280

By:

Yeoh, Yuan Qi;
Horsley, John R.;
Yu, Jingxian;
Polyak, Steven W.;
Jovcevski, Blagojce;
Abell, Andrew D.

Publication type:

Article

Synthesis and Antibacterial Activity of New N‐Alkylammonium and Carbonate‐Triazole Derivatives within Desosamine of 14‐ and 15‐Membered Lactone Macrolides.

Published in:

ChemMedChem, 2020, v. 15, n. 16, p. 1529, doi. 10.1002/cmdc.202000273

By:

Janas, Anna;
Pecyna, Paulina;
Gajecka, Marzena;
Bartl, Franz;
Przybylski, Piotr

Publication type:

Article

Synthesis and Anticancer Properties of Oxazepines Related to Azaisoerianin and IsoCoQuines.

Published in:

ChemMedChem, 2020, v. 15, n. 16, p. 1571, doi. 10.1002/cmdc.202000197

By:

Khelifi, Ilhem;
Pecnard, Shannon;
Bernadat, Guillaume;
Bignon, Jérome;
Levaique, Hélène;
Dubois, Joëlle;
Provot, Olivier;
Alami, Mouad

Publication type:

Article

A Dual Inhibitor of DYRK1A and GSK3β for β‐Cell Proliferation: Aminopyrazine Derivative GNF4877.

Published in:

ChemMedChem, 2020, v. 15, n. 16, p. 1562, doi. 10.1002/cmdc.202000183

By:

Liu, Yahu A.;
Jin, Qihui;
Ding, Qiang;
Hao, Xueshi;
Mo, Tingting;
Yan, Shanshan;
Zou, Yefen;
Huang, Zhihong;
Zhang, Xiaoyue;
Gao, Wenqi;
Wu, Tom Y.‐H.;
Li, Chun;
Bursalaya, Badry;
Di Donato, Michael;
Zhang, You‐Qing;
Deaton, Lisa;
Shen, Weijun;
Taylor, Brandon;
Kamireddy, Anwesh;
Harb, George

Publication type:

Article

Discovery of an Orally Active and Long‐Acting DPP‐IV Inhibitor through Property‐Based Optimization with an in Silico Biotransformation Prediction Tool.

Published in:

ChemMedChem, 2020, v. 15, n. 16, p. 1608, doi. 10.1002/cmdc.202000175

By:

Zeng, Shaogao;
Dou, Wenyuan;
Li, Manna;
Zhou, Yang;
Guo, Jiehuang;
Zhao, Nan;
Huang, Hong;
Zhou, Qiaoli;
Hu, Wenhui;
Ma, Yanfang;
Zhao, Xin;
Xie, Hui

Publication type:

Article

Design, Synthesis, Radiosynthesis and Biological Evaluation of Fenretinide Analogues as Anticancer and Metabolic Syndrome‐Preventive Agents.

Published in:

ChemMedChem, 2020, v. 15, n. 16, p. 1579, doi. 10.1002/cmdc.202000143

By:

Patruno, Ilaria;
Thompson, Dawn;
Dall'Angelo, Sergio;
Windhorst, Albert D.;
Vugts, Danielle J.;
Poot, Alex J.;
Mody, Nimesh;
Zanda, Matteo

Publication type:

Article

Pentathiepins: A Novel Class of Glutathione Peroxidase 1 Inhibitors that Induce Oxidative Stress, Loss of Mitochondrial Membrane Potential and Apoptosis in Human Cancer Cells.

Published in:

ChemMedChem, 2020, v. 15, n. 16, p. 1515, doi. 10.1002/cmdc.202000160

By:

Behnisch‐Cornwell, Steven;
Bandaru, Siva Sankar Murthy;
Napierkowski, Martin;
Wolff, Lisa;
Zubair, Muhammad;
Urbainsky, Claudia;
Lillig, Christopher;
Schulzke, Carola;
Bednarski, Patrick J.

Publication type:

Article

Synthesis of N‐Aryl‐ and N‐alkyl‐Substituted Imidazolium Silver Complexes: Cytotoxic Screening by Using Human Cell Lines Modelling Acute Myeloid Leukaemia.

Published in:

ChemMedChem, 2020, v. 15, n. 16, p. 1509, doi. 10.1002/cmdc.202000138

By:

Alme, Eirin;
Törnroos, Karl Wilhelm;
Gjertsen, Bjørn Tore;
Bjørsvik, Hans‐René

Publication type:

Article