Works matching IS 18607179 AND DT 2020 AND VI 15 AND IP 13

Results: 14

Front Cover: Synthetic Peroxides Promote Apoptosis of Cancer Cells by Inhibiting P‐Glycoprotein ABCB5 (ChemMedChem 13/2020).

Published in:

ChemMedChem, 2020, v. 15, n. 13, p. 1101, doi. 10.1002/cmdc.202000413

By:

Yaremenko, Ivan A.;
Coghi, Paolo;
Prommana, Parichat;
Qiu, Congling;
Radulov, Peter S.;
Qu, Yuanqing;
Belyakova, Yulia Yu.;
Zanforlin, Enrico;
Kokorekin, Vladimir A.;
Wu, Yuki Yu Jun;
Fleury, Fabrice;
Uthaipibull, Chairat;
Wong, Vincent Kam Wai;
Terent'ev, Alexander O.

Publication type:

Article

Design, Synthesis, and Characterization of Novel CXCR4 Antagonists Featuring Cyclic Amines.

Published in:

ChemMedChem, 2020, v. 15, n. 13, p. 1150, doi. 10.1002/cmdc.202000268

By:

Lin, Yu;
Li, Zhanhui;
Ma, Haikuo;
Wang, Yujie;
Wang, Xu;
Song, Shiwei;
Zhao, Li;
Wu, Shuwei;
Tian, Sheng;
Fu, Chunyan;
Luo, Lusong;
Zhu, Fang;
He, Sudan;
Zheng, Jiyue;
Zhang, Xiaohu

Publication type:

Article

Macrocyclic Iminopeptides Diversify To Better Target Proteins.

Published in:

ChemMedChem, 2020, v. 15, n. 13, p. 1111, doi. 10.1002/cmdc.202000261

By:

Reguera, Leslie;
Rivera, Daniel G.

Publication type:

Article

The Synthesis and Anti‐tumour Properties of Poly Ethoxy Ethyl Glycinamide (PEE−G) Scaffolds with Multiple PD‐1 Peptides Attached.

Published in:

ChemMedChem, 2020, v. 15, n. 13, p. 1128, doi. 10.1002/cmdc.202000221

By:

Shrestha, Rinu;
Petley, Emma V.;
Farrand, Kathryn J.;
Jamieson, Sam A.;
Jiao, Wanting;
Teesdale‐Spittle, Paul H.;
Mace, Peter D.;
Hermans, Ian F.;
Rendle, Phillip M.

Publication type:

Article

Sulfonylguanidine Derivatives as Potential Antimelanoma Agents.

Published in:

ChemMedChem, 2020, v. 15, n. 13, p. 1113, doi. 10.1002/cmdc.202000218

By:

Baladi, Tom;
Hamouda‐Tekaya, Nedra;
Gonçalves, Leticia Christina Pires;
Rocchi, Stéphane;
Ronco, Cyril;
Benhida, Rachid

Publication type:

Article

Synthesis, Radiosynthesis and Biological Evaluation of Buprenorphine‐Derived Phenylazocarboxamides as Novel μ‐Opioid Receptor Ligands.

Published in:

ChemMedChem, 2020, v. 15, n. 13, p. 1175, doi. 10.1002/cmdc.202000180

By:

Krüll, Jasmin;
Fehler, Stefanie K.;
Hofmann, Laura;
Nebel, Natascha;
Maschauer, Simone;
Prante, Olaf;
Gmeiner, Peter;
Lanig, Harald;
Hübner, Harald;
Heinrich, Markus R.

Publication type:

Article

Physicochemical Properties of Zwitterionic Drugs in Therapy.

Published in:

ChemMedChem, 2020, v. 15, n. 13, p. 1102, doi. 10.1002/cmdc.202000164

By:

Mazák, Károly;
Noszál, Béla

Publication type:

Article

Design and Synthesis of Dihydroxamic Acids as HDAC6/8/10 Inhibitors.

Published in:

ChemMedChem, 2020, v. 15, n. 13, p. 1163, doi. 10.1002/cmdc.202000149

By:

Morgen, Michael;
Steimbach, Raphael R.;
Géraldy, Magalie;
Hellweg, Lars;
Sehr, Peter;
Ridinger, Johannes;
Witt, Olaf;
Oehme, Ina;
Herbst‐Gervasoni, Corey J.;
Osko, Jeremy D.;
Porter, Nicholas J.;
Christianson, David W.;
Gunkel, Nikolas;
Miller, Aubry K.

Publication type:

Article

Targeting the Water Network in Cyclin G‐Associated Kinase (GAK) with 4‐Anilino‐quin(az)oline Inhibitors.

Published in:

ChemMedChem, 2020, v. 15, n. 13, p. 1200, doi. 10.1002/cmdc.202000150

By:

Asquith, Christopher R. M.;
Tizzard, Graham J.;
Bennett, James M.;
Wells, Carrow I.;
Elkins, Jonathan M.;
Willson, Timothy M.;
Poso, Antti;
Laitinen, Tuomo

Publication type:

Article

Synthesis of Novel Pyridine‐Carboxylates as Small‐Molecule Inhibitors of Human Aspartate/Asparagine‐β‐Hydroxylase.

Published in:

ChemMedChem, 2020, v. 15, n. 13, p. 1139, doi. 10.1002/cmdc.202000147

By:

Brewitz, Lennart;
Tumber, Anthony;
Thalhammer, Armin;
Salah, Eidarus;
Christensen, Kirsten E.;
Schofield, Christopher J.

Publication type:

Article

Synthetic Guaiacol Derivatives as Promising Myeloperoxidase Inhibitors Targeting Atherosclerotic Cardiovascular Disease.

Published in:

ChemMedChem, 2020, v. 15, n. 13, p. 1187, doi. 10.1002/cmdc.202000084

By:

Premkumar, Jayaraj;
Sampath, Parthasarathy;
Sanjay, Rajagopalan;
Chandrakala, Aluganti;
Rajagopal, Desikan

Publication type:

Article

A Library of Thiazolidin‐4‐one Derivatives as Protein Tyrosine Phosphatase 1B (PTP1B) Inhibitors: An Attempt To Discover Novel Antidiabetic Agents.

Published in:

ChemMedChem, 2020, v. 15, n. 13, p. 1229, doi. 10.1002/cmdc.202000055

By:

Patel, Ashish D.;
Pasha, Thopallada Y.;
Lunagariya, Paras;
Shah, Umang;
Bhambharoliya, Tushar;
Tripathi, Rati K. P.

Publication type:

Article

Design, Synthesis, Structure‐Activity Relationship and Docking Studies of Novel Functionalized Arylvinyl‐1,2,4‐Trioxanes as Potent Antiplasmodial as well as Anticancer Agents.

Published in:

ChemMedChem, 2020, v. 15, n. 13, p. 1216, doi. 10.1002/cmdc.202000045

By:

Tiwari, Mohit K.;
Coghi, Paolo;
Agrawal, Prakhar;
Shyamlal, Bharti Rajesh K.;
Jun Yang, Li;
Yadav, Lalit;
Peng, Yuzhong;
Sharma, Richa;
Yadav, Dharmendra K.;
Sahal, Dinkar;
Kam Wai Wong, Vincent;
Chaudhary, Sandeep

Publication type:

Article

Synthetic Peroxides Promote Apoptosis of Cancer Cells by Inhibiting P‐Glycoprotein ABCB5.

Published in:

ChemMedChem, 2020, v. 15, n. 13, p. 1118, doi. 10.1002/cmdc.202000042

By:

Yaremenko, Ivan A.;
Coghi, Paolo;
Prommana, Parichat;
Qiu, Congling;
Radulov, Peter S.;
Qu, Yuanqing;
Belyakova, Yulia Yu.;
Zanforlin, Enrico;
Kokorekin, Vladimir A.;
Wu, Yuki Yu Jun;
Fleury, Fabrice;
Uthaipibull, Chairat;
Wong, Vincent Kam Wai;
Terent'ev, Alexander O.

Publication type:

Article