Works matching IS 18607179 AND DT 2019 AND VI 14 AND IP 13

Results: 10

Front Cover: The Discovery of LML134, a Histamine H3 Receptor Inverse Agonist for the Clinical Treatment of Excessive Sleep Disorders (ChemMedChem 13/2019).

Published in:

ChemMedChem, 2019, v. 14, n. 13, p. 1226, doi. 10.1002/cmdc.201900365

By:

Troxler, Thomas;
Feuerbach, Dominik;
Zhang, Xuechun;
Yang, Charles R.;
Lagu, Bharat;
Perrone, Mark;
Wang, Tie‐Lin;
Briner, Karin;
Bock, Mark G.;
Auberson, Yves P.

Publication type:

Article

Biomolecular Simulations in Structure‐Based Drug Discovery. Edited by Francesco L. Gervasio and Vojtech Spiwock.

Published in:

ChemMedChem, 2019, v. 14, n. 13, p. 1303, doi. 10.1002/cmdc.201900291

By:

Bronowska, Agnieszka K.

Publication type:

Article

Oxadiazole Derivatives as Dual Orexin Receptor Antagonists: Synthesis, Structure–Activity Relationships, and Sleep‐Promoting Properties in Rats.

Published in:

ChemMedChem, 2019, v. 14, n. 13, p. 1257, doi. 10.1002/cmdc.201900242

By:

Brotschi, Christine;
Roch, Catherine;
Gatfield, John;
Treiber, Alexander;
Williams, Jodi T.;
Sifferlen, Thierry;
Heidmann, Bibia;
Jenck, Francois;
Bolli, Martin H.;
Boss, Christoph

Publication type:

Article

The Outcomes of Decorated Prolines in the Discovery of Antimicrobial Peptides from Temporin‐L.

Published in:

ChemMedChem, 2019, v. 14, n. 13, p. 1283, doi. 10.1002/cmdc.201900221

By:

Buommino, Elisabetta;
Carotenuto, Alfonso;
Antignano, Ignazio;
Bellavita, Rosa;
Casciaro, Bruno;
Loffredo, Maria Rosa;
Merlino, Francesco;
Novellino, Ettore;
Mangoni, Maria Luisa;
Nocera, Francesca Paola;
Brancaccio, Diego;
Punzi, Pasqualina;
Roversi, Daniela;
Ingenito, Raffaele;
Bianchi, Elisabetta;
Grieco, Paolo

Publication type:

Article

Discovery of 6‐Arylurea‐2‐arylbenzoxazole and 6‐Arylurea‐2‐arylbenzimidazole Derivatives as Angiogenesis Inhibitors: Design, Synthesis and in vitro Biological Evaluation.

Published in:

ChemMedChem, 2019, v. 14, n. 13, p. 1291, doi. 10.1002/cmdc.201900216

By:

Zi, Mengli;
Liu, Feifei;
Wu, Di;
Li, Ke;
Zhang, Da;
Zhu, Changcheng;
Zhang, Zhiyun;
Li, Linghua;
Zhang, Conghai;
Xie, Mingjin;
Lin, Jun;
Zhang, Jihong;
Jin, Yi

Publication type:

Article

Development of Tetrahydroindazole‐Based Potent and Selective Sigma‐2 Receptor Ligands.

Published in:

ChemMedChem, 2019, v. 14, n. 13, p. 1248, doi. 10.1002/cmdc.201900203

By:

Iyamu, Iredia D.;
Lv, Wei;
Malik, Neha;
Mishra, Rama K.;
Schiltz, Gary E.

Publication type:

Article

The Discovery of LML134, a Histamine H3 Receptor Inverse Agonist for the Clinical Treatment of Excessive Sleep Disorders.

Published in:

ChemMedChem, 2019, v. 14, n. 13, p. 1238, doi. 10.1002/cmdc.201900176

By:

Troxler, Thomas;
Feuerbach, Dominik;
Zhang, Xuechun;
Yang, Charles R.;
Lagu, Bharat;
Perrone, Mark;
Wang, Tie‐Lin;
Briner, Karin;
Bock, Mark G.;
Auberson, Yves P.

Publication type:

Article

Investigation of Dipicolinic Acid Isosteres for the Inhibition of Metallo‐β‐Lactamases.

Published in:

ChemMedChem, 2019, v. 14, n. 13, p. 1271, doi. 10.1002/cmdc.201900172

By:

Chen, Allie Y.;
Thomas, Pei W.;
Cheng, Zishuo;
Xu, Nasa Y.;
Tierney, David L.;
Crowder, Michael W.;
Fast, Walter;
Cohen, Seth M.

Publication type:

Article

Synthesis and Evaluation of Nifurtimox–Adamantane Adducts with Trypanocidal Activity.

Published in:

ChemMedChem, 2019, v. 14, n. 13, p. 1227, doi. 10.1002/cmdc.201900165

By:

Foscolos, Angeliki‐Sofia;
Papanastasiou, Ioannis;
Tsotinis, Andrew;
Taylor, Martin C.;
Kelly, John M.

Publication type:

Article

Synthesis and Antibacterial Evaluation of Bis‐thiazolium, Bis‐imidazolium, and Bis‐triazolium Derivatives.

Published in:

ChemMedChem, 2019, v. 14, n. 13, p. 1232, doi. 10.1002/cmdc.201900151

By:

Thomas, Benoît;
Duval, Raphaël E.;
Fontanay, Stéphane;
Varbanov, Mihayl;
Boisbrun, Michel

Publication type:

Article