Works matching AU Zappalà, Maria
Results: 34
Non-covalent immunoproteasome inhibitors induce cell cycle arrest in multiple myeloma MM.1R cells.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 1307, doi. 10.1080/14756366.2019.1594802
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- Article
Synthesis and biological evaluation of novel peptidomimetics as rhodesain inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, n. 6, p. 1184, doi. 10.3109/14756366.2015.1108972
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- Article
Synthesis and Antitumour Activity of 1 H,3 H-Thiazolo[3,4- a]benzimidazole Derivatives.
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- Archiv der Pharmazie, 2001, v. 334, n. 6, p. 203, doi. 10.1002/1521-4184(200106)334:6<203::AID-ARDP203>3.0.CO;2-L
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- Article
Enantioseparation, absolute configuration determination, and anticonvulsant activity of (±)‐1‐(4‐aminophenyl)‐7,8‐methylenedioxy‐1,2,3,5‐tetrahydro‐4H‐2,3‐benzodiazepin‐4‐oneCrystallographic data for the structure reported in this paper have been deposited with the Cambridge Crystallographic Data Centre (CCDC 189745).
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- Chirality, 2007, v. 19, n. 1, p. 16
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- Article
Drug combination studies of PS-1 and quercetin against rhodesain of Trypanosoma brucei rhodesiense.
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- Natural Product Research, 2022, v. 36, n. 16, p. 4282, doi. 10.1080/14786419.2021.1978993
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- Article
Evaluation of curcumin irreversibility.
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- 2020
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- Letter
Drug combination studies of curcumin and genistein against rhodesain of Trypanosoma brucei rhodesiense.
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- Natural Product Research, 2019, v. 33, n. 24, p. 3577, doi. 10.1080/14786419.2018.1483927
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- Article
Synthesis of Novel 3-(Alkylcarbamoyl)-2-aryl-1,2-dihydro-6,7-(methylenedioxy)-3 H-quinazolin-4-ones as Anticonvulsant Agents.
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- Chemistry & Biodiversity, 2006, v. 3, n. 3, p. 304, doi. 10.1002/cbdv.200690033
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- Article
Peptidyl Vinyl Ketone Irreversible Inhibitors of Rhodesain: Modifications of the P2 Fragment.
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- ChemMedChem, 2020, v. 15, n. 16, p. 1552, doi. 10.1002/cmdc.202000360
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- Article
Development of Novel Benzodiazepine‐Based Peptidomimetics as Inhibitors of Rhodesain from Trypanosoma brucei rhodesiense.
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- ChemMedChem, 2020, v. 15, n. 11, p. 995, doi. 10.1002/cmdc.202000158
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- Article
Development of Novel Amides as Noncovalent Inhibitors of Immunoproteasomes.
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- ChemMedChem, 2019, v. 14, n. 8, p. 842, doi. 10.1002/cmdc.201900028
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- Article
Development of Novel Selective Peptidomimetics Containing a Boronic Acid Moiety, Targeting the 20S Proteasome as Anticancer Agents.
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- ChemMedChem, 2014, v. 9, n. 8, p. 1801, doi. 10.1002/cmdc.201402075
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- Article
Synthesis and Biological Evaluation of Papain-Family Cathepsin L-Like Cysteine Protease Inhibitors Containing a 1,4-Benzodiazepine Scaffold as Antiprotozoal Agents.
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- ChemMedChem, 2014, v. 9, n. 8, p. 1817, doi. 10.1002/cmdc.201402079
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- Article
Synthesis and Molecular Modeling Studies of Derivatives of a Highly Potent Peptidomimetic Vinyl Ester as Falcipain-2 Inhibitors.
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- ChemMedChem, 2012, v. 7, n. 9, p. 1594, doi. 10.1002/cmdc.201200274
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- Article
Development of Novel Peptidomimetics Containing a Vinyl Sulfone Moiety as Proteasome Inhibitors.
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- ChemMedChem, 2011, v. 6, n. 7, p. 1228, doi. 10.1002/cmdc.201100093
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- Article
Synthesis, Chiral Resolution and Pharmacological Evaluation of a 2,3-Benzodiazepine-Derived Noncompetitive AMPA Receptor Antagonist.
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- ChemMedChem, 2009, v. 4, n. 3, p. 415, doi. 10.1002/cmdc.200800341
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- Article
Nonpeptidic Vinyl and Allyl Phosphonates as Falcipain-2 Inhibitors.
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- ChemMedChem, 2008, v. 3, n. 7, p. 1030, doi. 10.1002/cmdc.200800050
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- Article
Development of Novel Peptidyl Nitriles Targeting Rhodesain and Falcipain-2 for the Treatment of Sleeping Sickness and Malaria.
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- International Journal of Molecular Sciences, 2024, v. 25, n. 8, p. 4410, doi. 10.3390/ijms25084410
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- Article
The Inhibition of NS2B/NS3 Protease: A New Therapeutic Opportunity to Treat Dengue and Zika Virus Infection.
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- International Journal of Molecular Sciences, 2024, v. 25, n. 8, p. 4376, doi. 10.3390/ijms25084376
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- Article
Blunting Neuroinflammation by Targeting the Immunoproteasome with Novel Amide Derivatives.
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- International Journal of Molecular Sciences, 2023, v. 24, n. 13, p. 10732, doi. 10.3390/ijms241310732
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- Article
Virtual Screening Strategy and In Vitro Tests to Identify New Inhibitors of the Immunoproteasome.
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- International Journal of Molecular Sciences, 2023, v. 24, n. 13, p. 10504, doi. 10.3390/ijms241310504
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- Article
Dipeptide Nitrile CD34 with Curcumin: A New Improved Combination Strategy to Synergistically Inhibit Rhodesain of Trypanosoma brucei rhodesiense.
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- International Journal of Molecular Sciences, 2023, v. 24, n. 10, p. 8477, doi. 10.3390/ijms24108477
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- Article
Monoclonal Antibodies: The Greatest Resource to Treat Multiple Myeloma.
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- 2023
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- Literature Review
Drug Combination Studies of the Dipeptide Nitrile CD24 with Curcumin: A New Strategy to Synergistically Inhibit Rhodesain of Trypanosoma brucei rhodesiense.
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- International Journal of Molecular Sciences, 2022, v. 23, n. 22, p. 14470, doi. 10.3390/ijms232214470
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- Article
Development of Reduced Peptide Bond Pseudopeptide Michael Acceptors for the Treatment of Human African Trypanosomiasis.
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- Molecules, 2022, v. 27, n. 12, p. 3765, doi. 10.3390/molecules27123765
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- Article
Immunoproteasome and Non-Covalent Inhibition: Exploration by Advanced Molecular Dynamics and Docking Methods.
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- Molecules, 2021, v. 26, n. 13, p. 4046, doi. 10.3390/molecules26134046
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- Article
Exploring the SARS-CoV-2 Proteome in the Search of Potential Inhibitors via Structure-Based Pharmacophore Modeling/Docking Approach.
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- Computation, 2020, v. 8, n. 3, p. 77, doi. 10.3390/computation8030077
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- Article
Synthesis and Cytotoxicity of Diarylpentanoids against Sensitive CCRF‐CEM and Multidrug‐Resistant CEM/ADR5000 Leukemia Cells.
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- Chemistry & Biodiversity, 2022, v. 19, n. 2, p. 1, doi. 10.1002/cbdv.202100451
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- Article
Drug Combination Studies of Isoquinolinone AM12 with Curcumin or Quercetin: A New Combination Strategy to Synergistically Inhibit 20S Proteasome.
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- International Journal of Molecular Sciences, 2024, v. 25, n. 19, p. 10708, doi. 10.3390/ijms251910708
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- Article
Ethnobotanical studies on the Tyrrhenian side of the Aspromonte Massif (Calabria, Southern Italy).
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- Plant Biosystems, 2024, v. 158, n. 3, p. 545, doi. 10.1080/11263504.2024.2336601
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- Article
Peptide-Based Proteasome Inhibitors in Anticancer Drug Design.
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- Medicinal Research Reviews, 2014, v. 34, n. 5, p. 1001, doi. 10.1002/med.21312
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- Article
Falcipain-2 inhibitors.
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- Medicinal Research Reviews, 2010, v. 30, n. 1, p. 136, doi. 10.1002/med.20163
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- Article
A SIMPLE AND EFFICIENT SYNTHESIS OF GYKI 52466 AND GYKI 52895.
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- Synthetic Communications, 2002, v. 32, n. 4, p. 527, doi. 10.1081/SCC-120002397
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- Article
Synthesis and stereochemistry of novel [1,2,4]oxadiazolo[4,5- a][1,5]benzodiazepine derivatives.
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- Journal of Heterocyclic Chemistry, 1990, v. 27, n. 2, p. 371, doi. 10.1002/jhet.5570270250
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- Article