Works matching IS 18607179 AND DT 2014 AND VI 9 AND IP 11

Results: 20

Natural Products in Medicinal Chemistry.

Published in:

ChemMedChem, 2014, v. 9, n. 11, p. 2602, doi. 10.1002/cmdc.201402297

By:

Sarker, Satyajit D.

Publication type:

Article

Biological Evaluation of Potent Triclosan-Derived Inhibitors of the Enoyl-Acyl Carrier Protein Reductase InhA in Drug-Sensitive and Drug-Resistant Strains of Mycobacterium tuberculosis.

Published in:

ChemMedChem, 2014, v. 9, n. 11, p. 2528, doi. 10.1002/cmdc.201402255

By:

Stec, Jozef;
Vilchèze, Catherine;
Lun, Shichun;
Perryman, Alexander L.;
Wang, Xin;
Freundlich, Joel S.;
Bishai, William;
Jacobs, William R.;
Kozikowski, Alan P.

Publication type:

Article

Synthesis and Structure-Activity Relationship Studies of 2-(1,3,4-Oxadiazole-2(3H)-thione)-3-amino-5-arylthieno[2,3-b]pyridines as Inhibitors of DRAK2.

Published in:

ChemMedChem, 2014, v. 9, n. 11, p. 2587, doi. 10.1002/cmdc.201402234

By:

Leonczak, Piotr;
Gao, Ling‐Jie;
Ramadori, Anna Teresa;
Lescrinier, Eveline;
Rozenski, Jef;
De Jonghe, Steven;
Herdewijn, Piet

Publication type:

Article

Design and Synthesis of Aminostilbene-Arylpropenones as Tubulin Polymerization Inhibitors.

Published in:

ChemMedChem, 2014, v. 9, n. 11, p. 2565, doi. 10.1002/cmdc.201402256

By:

Kamal, Ahmed;
Kumar, G. Bharath;
Polepalli, Sowjanya;
Shaik, Anver Basha;
Reddy, Vangala Santhosh;
Reddy, M. Kashi;
Reddy, Ch. Ratna;
Mahesh, Rasala;
Kapure, Jeevak Sopanrao;
Jain, Nishant

Publication type:

Article

α-Keto Phenylamides as P1'-Extended Proteasome Inhibitors.

Published in:

ChemMedChem, 2014, v. 9, n. 11, p. 2557, doi. 10.1002/cmdc.201402244

By:

Voss, Constantin;
Scholz, Christoph;
Knorr, Sabine;
Beck, Philipp;
Stein, Martin L.;
Zall, Andrea;
Kuckelkorn, Ulrike;
Kloetzel, Peter‐Michael;
Groll, Michael;
Hamacher, Kay;
Schmidt, Boris

Publication type:

Article

Non-natural Acetogenin Analogues as Potent Trypanosoma brucei Inhibitors.

Published in:

ChemMedChem, 2014, v. 9, n. 11, p. 2548, doi. 10.1002/cmdc.201402272

By:

Florence, Gordon J.;
Fraser, Andrew L.;
Gould, Eoin R.;
King, Elizabeth F. B.;
Menzies, Stefanie K.;
Morris, Joanne C.;
Tulloch, Lindsay B.;
Smith, Terry K.

Publication type:

Article

Structure-Guided Design of Thiazolidine Derivatives as Mycobacterium tuberculosis Pantothenate Synthetase Inhibitors.

Published in:

ChemMedChem, 2014, v. 9, n. 11, p. 2538, doi. 10.1002/cmdc.201402171

By:

Devi, Parthiban Brindha;
Samala, Ganesh;
Sridevi, Jonnalagadda Padma;
Saxena, Shalini;
Alvala, Mallika;
Salina, Elena G.;
Sriram, Dharmarajan;
Yogeeswari, Perumal

Publication type:

Article

Molecular Mechanism of Action of 2-Ferrocenyl-1,1-diphenylbut-1-ene on HL-60 Leukemia Cells.

Published in:

ChemMedChem, 2014, v. 9, n. 11, p. 2580, doi. 10.1002/cmdc.201402219

By:

de Oliveira, Alane Cabral;
da Silva, Emanuella Gomes;
Rocha, Danilo Damasceno;
Hillard, Elizabeth A.;
Pigeon, Pascal;
Jaouen, Gérard;
Rodrigues, Felipe A. R.;
de Abreu, Fabiane C.;
da Rocha Ferreira, Fabrícia;
Goulart, Marilia O. F.;
Costa‐Lotufo, Letícia V.

Publication type:

Article

Novel Hinge-Binding Motifs for Janus Kinase 3 Inhibitors: A Comprehensive Structure-Activity Relationship Study on Tofacitinib Bioisosteres.

Published in:

ChemMedChem, 2014, v. 9, n. 11, p. 2516, doi. 10.1002/cmdc.201402252

By:

Gehringer, Matthias;
Forster, Michael;
Pfaffenrot, Ellen;
Bauer, Silke M.;
Laufer, Stefan A.

Publication type:

Article

Drug Screening Boosted by Hyperpolarized Long-Lived States in NMR.

Published in:

ChemMedChem, 2014, v. 9, n. 11, p. 2509, doi. 10.1002/cmdc.201402214

By:

Buratto, Roberto;
Bornet, Aurélien;
Milani, Jonas;
Mammoli, Daniele;
Vuichoud, Basile;
Salvi, Nicola;
Singh, Maninder;
Laguerre, Aurélien;
Passemard, Solène;
Gerber‐Lemaire, Sandrine;
Jannin, Sami;
Bodenhausen , Geoffrey

Publication type:

Article

Are 1,4- and 1,5-Disubstituted 1,2,3-Triazoles Good Pharmacophoric Groups?

Published in:

ChemMedChem, 2014, v. 9, n. 11, p. 2497, doi. 10.1002/cmdc.201402233

By:

Massarotti, Alberto;
Aprile, Silvio;
Mercalli, Valentina;
Del Grosso, Erika;
Grosa, Giorgio;
Sorba, Giovanni;
Tron, Gian Cesare

Publication type:

Article

Structure-Activity Relationship, Biological, and Pharmacological Characterization of the Proline Sulfonamide ACT-462206: a Potent, Brain-Penetrant Dual Orexin 1/Orexin 2 Receptor Antagonist.

Published in:

ChemMedChem, 2014, v. 9, n. 11, p. 2486, doi. 10.1002/cmdc.201402258

By:

Boss, Christoph;
Roch‐Brisbare, Catherine;
Steiner, Michel A.;
Treiber, Alexander;
Dietrich, Hendrik;
Jenck, Francois;
von Raumer, Markus;
Sifferlen, Thierry;
Brotschi, Christine;
Heidmann, Bibia;
Williams, Jodi T.;
Aissaoui, Hamed;
Siegrist, Romain;
Gatfield, John

Publication type:

Article

5-(Piperidin-4-yl)-3-Hydroxypyrazole: A Novel Scaffold for Probing the Orthosteric γ-Aminobutyric Acid Type A Receptor Binding Site.

Published in:

ChemMedChem, 2014, v. 9, n. 11, p. 2475, doi. 10.1002/cmdc.201402248

By:

Krall, Jacob;
Kongstad, Kenneth T.;
Nielsen, Birgitte;
Sørensen, Troels E.;
Balle, Thomas;
Jensen, Anders A.;
Frølund, Bente

Publication type:

Article

Position and Length of Fatty Acids Strongly Affect Receptor Selectivity Pattern of Human Pancreatic Polypeptide Analogues.

Published in:

ChemMedChem, 2014, v. 9, n. 11, p. 2463, doi. 10.1002/cmdc.201402235

By:

Mäde, Veronika;
Bellmann‐Sickert, Kathrin;
Kaiser, Anette;
Meiler, Jens;
Beck‐Sickinger, Annette G.

Publication type:

Article

Small Molecules that Target the Toxic RNA in Myotonic Dystrophy Type 2.

Published in:

ChemMedChem, 2014, v. 9, n. 11, p. 2455, doi. 10.1002/cmdc.201402095

By:

Nguyen, Lien;
Lee, JuYeon;
Wong, Chun‐Ho;
Zimmerman, Steven C.

Publication type:

Article

Amphiphilic Bicyclic Peptides as Cellular Delivery Agents.

Published in:

ChemMedChem, 2014, v. 9, n. 11, p. 2449, doi. 10.1002/cmdc.201402230

By:

Oh, Donghoon;
Darwish, Shaban Anwar;
Shirazi, Amir Nasrolahi;
Tiwari, Rakesh Kumar;
Parang, Keykavous

Publication type:

Article

Diaryl-Substituted Azolylthioacetamides: Inhibitor Discovery of New Delhi Metallo-β-Lactamase-1 (NDM-1).

Published in:

ChemMedChem, 2014, v. 9, n. 11, p. 2445, doi. 10.1002/cmdc.201402249

By:

Zhang, Yi‐Lin;
Yang, Ke‐Wu;
Zhou, Ya‐Jun;
LaCuran, Alecander E.;
Oelschlaeger, Peter;
Crowder, Michael W.

Publication type:

Article

In Vitro Antiamoebic Activity Evaluation and Docking Studies of Metronidazole-Triazole Hybrids.

Published in:

ChemMedChem, 2014, v. 9, n. 11, p. 2439, doi. 10.1002/cmdc.201402240

By:

Negi, Beena;
Raj, K. Kranthi;
Siddiqui, Shadab Miyan;
Ramachandran, Dittakavi;
Azam, Amir;
Rawat, Diwan S.

Publication type:

Article

Recent Advances in The Discovery of N-Myristoyltransferase Inhibitors.

Published in:

ChemMedChem, 2014, v. 9, n. 11, p. 2425, doi. 10.1002/cmdc.201402174

By:

Zhao, Can;
Ma, Shutao

Publication type:

Article

Therapeutic Strategies for Metabolic Diseases: Small-Molecule Diacylglycerol Acyltransferase (DGAT) Inhibitors.

Published in:

ChemMedChem, 2014, v. 9, n. 11, p. 2410, doi. 10.1002/cmdc.201402069

By:

Naik, Ravi;
Obiang‐Obounou, Brice W.;
Kim, Minkyoung;
Choi, Yongseok;
Lee, Hyun Sun;
Lee, Kyeong

Publication type:

Article