Works matching IS 18607179 AND DT 2013 AND VI 8 AND IP 7

Results: 20

Graphical Abstract: ChemMedChem 7/2013.

Published in:: ChemMedChem, 2013, v. 8, n. 7, p. 1023, doi. 10.1002/cmdc.201390027
Publication type:: Article

Water-Soluble Nitric-Oxide-Releasing Acetylsalicylic Acid (ASA) Prodrugs.

Published in:

ChemMedChem, 2013, v. 8, n. 7, p. 1199, doi. 10.1002/cmdc.201300105

By:

Rolando, Barbara;
Lazzarato, Loretta;
Donnola, Monica;
Marini, Elisabetta;
Joseph, Sony;
Morini, Giuseppina;
Pozzoli, Cristina;
Fruttero, Roberta;
Gasco, Alberto

Publication type:

Article

Synthesis of an <sup>11</sup>C-Labeled Antiprion GN8 Derivative and Evaluation of Its Brain Uptake by Positron Emission Tomography.

Published in:

ChemMedChem, 2013, v. 8, n. 7, p. 1035, doi. 10.1002/cmdc.201300167

By:

Kimura, Tsutomu;
Sako, Takeo;
Siqin;
Hosokawa‐Muto, Junji;
Cui, Yi Long;
Wada, Yasuhiro;
Kataoka, Yosky;
Doi, Hisashi;
Sakaguchi, Suehiro;
Suzuki, Masaaki;
Watanabe, Yasuyoshi;
Kuwata, Kazuo

Publication type:

Article

Adamantyl Arotinoids That Inhibit IκB Kinase α and IκB Kinase β.

Published in:

ChemMedChem, 2013, v. 8, n. 7, p. 1184, doi. 10.1002/cmdc.201300100

By:

Lorenzo, Paula;
Ortiz, María A.;
Álvarez, Rosana;
Piedrafita, F. Javier;
de Lera, Ángel R.

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 7/2013.

Published in:: ChemMedChem, 2013, v. 8, n. 7, p. 1032, doi. 10.1002/cmdc.201390028
Publication type:: Article

Back Cover: From On-Target to Off-Target Activity: Identification and Optimisation of Trypanosoma brucei GSK3 Inhibitors and Their Characterisation as Anti- Trypanosoma brucei Drug Discovery Lead Molecules (ChemMedChem 7/2013).

Published in:

ChemMedChem, 2013, v. 8, n. 7, p. 1228, doi. 10.1002/cmdc.201390029

By:

Woodland, Andrew;
Grimaldi, Raffaella;
Luksch, Torsten;
Cleghorn, Laura A. T.;
Ojo, Kayode K.;
Van Voorhis, Wesley C.;
Brenk, Ruth;
Frearson, Julie A.;
Gilbert, Ian H.;
Wyatt, Paul G.

Publication type:

Article

Design, Synthesis, and Structure-Activity Relationships of 3,4,5-Trisubstituted 4,5-Dihydro-1,2,4-oxadiazoles as TGR5 Agonists.

Published in:

ChemMedChem, 2013, v. 8, n. 7, p. 1210, doi. 10.1002/cmdc.201300144

By:

Zhu, Junjie;
Ye, Yangliang;
Ning, Mengmeng;
Mándi, Attila;
Feng, Ying;
Zou, Qingan;
Kurtán, Tibor;
Leng, Ying;
Shen, Jianhua

Publication type:

Article

Probing the Structural Properties of DNA/RNA Grooves with Sterically Restricted Phosphonium Dyes: Screening of Dye Cytotoxicity and Uptake.

Published in:

ChemMedChem, 2013, v. 8, n. 7, p. 1093, doi. 10.1002/cmdc.201300085

By:

Crnolatac, Ivo;
Tumir, Lidija‐Marija;
Lesev, Nedyalko Y.;
Vasilev, Aleksey A.;
Deligeorgiev, Todor G.;
Mišković, Katarina;
Glavaš‐Obrovac, Ljubica;
Vugrek, Oliver;
Piantanida, Ivo

Publication type:

Article

The Lab Oddity Prevails: Discovery of Pan-CDK Inhibitor ( R)- S-Cyclopropyl- S-(4-{[4-{[(1 R,2 R)-2-hydroxy-1-methylpropyl]oxy}-5-(trifluoromethyl)pyrimidin-2-yl]amino}phenyl)sulfoximide (BAY 1000394) for the Treatment of Cancer.

Published in:

ChemMedChem, 2013, v. 8, n. 7, p. 1067, doi. 10.1002/cmdc.201300096

By:

Lücking, Ulrich;
Jautelat, Rolf;
Krüger, Martin;
Brumby, Thomas;
Lienau, Philip;
Schäfer, Martina;
Briem, Hans;
Schulze, Julia;
Hillisch, Alexander;
Reichel, Andreas;
Wengner, Antje Margret;
Siemeister, Gerhard

Publication type:

Article

Alzheimer's Disease: Identification and Development of β-Secretase (BACE-1) Binding Fragments and Inhibitors by Dynamic Ligation Screening (DLS).

Published in:

ChemMedChem, 2013, v. 8, n. 7, p. 1041, doi. 10.1002/cmdc.201300078

By:

Fernández‐Bachiller, María Isabel;
Horatscheck, André;
Lisurek, Michael;
Rademann, Jörg

Publication type:

Article

Design and Synthesis of 4-(2,4,5-Trifluorophenyl)butane-1,3-diamines as Dipeptidyl Peptidase IV Inhibitors.

Published in:

ChemMedChem, 2013, v. 8, n. 7, p. 1104, doi. 10.1002/cmdc.201300104

By:

Zhu, Linrong;
Li, Yuanyuan;
Qiu, Ling;
Su, Mingbo;
Wang, Xin;
Xia, Chunmei;
Qu, Yi;
Li, Jingya;
Li, Jia;
Xiong, Bing;
Shen, Jingkang

Publication type:

Article

Rational Design of Angiotensin-I-Converting Enzyme Inhibitory Peptides by Integrating in silico Modeling and an in vitro Assay.

Published in:

ChemMedChem, 2013, v. 8, n. 7, p. 1057, doi. 10.1002/cmdc.201300132

By:

Jing, Tao;
Feng, Jian;
Li, De;
Liu, Jianping;
He, Guoxiang

Publication type:

Article

Inhibition of Leishmania infantum Trypanothione Reductase by Azole-Based Compounds: a Comparative Analysis with Its Physiological Substrate by X-ray Crystallography.

Published in:

ChemMedChem, 2013, v. 8, n. 7, p. 1175, doi. 10.1002/cmdc.201300176

By:

Baiocco, Paola;
Poce, Giovanna;
Alfonso, Salvatore;
Cocozza, Martina;
Porretta, Giulio Cesare;
Colotti, Gianni;
Biava, Mariangela;
Moraca, Francesca;
Botta, Maurizio;
Yardley, Vanessa;
Fiorillo, Annarita;
Lantella, Antonella;
Malatesta, Francesco;
Ilari, Andrea

Publication type:

Article

Aquaporin Inhibition by Gold(III) Compounds: New Insights.

Published in:

ChemMedChem, 2013, v. 8, n. 7, p. 1086, doi. 10.1002/cmdc.201300107

By:

Martins, Ana Paula;
Ciancetta, Antonella;
de Almeida, Andreia;
Marrone, Alessandro;
Re, Nazzareno;
Soveral, Graça;
Casini, Angela

Publication type:

Article

5′-Trityl-Substituted Thymidine Derivatives as a Novel Class of Antileishmanial Agents: Leishmania infantum EndoG as a Potential Target.

Published in:

ChemMedChem, 2013, v. 8, n. 7, p. 1161, doi. 10.1002/cmdc.201300129

By:

Casanova, Elena;
Moreno, David;
Gigante, Alba;
Rico, Eva;
Genes, Carlos Mario;
Oliva, Cristina;
Camarasa, María‐José;
Gago, Federico;
Jiménez‐Ruiz, Antonio;
Pérez‐Pérez, María‐Jesús

Publication type:

Article

Inside Cover: Alzheimer's Disease: Identification and Development of β-Secretase (BACE-1) Binding Fragments and Inhibitors by Dynamic Ligation Screening (DLS) (ChemMedChem 7/2013).

Published in:

ChemMedChem, 2013, v. 8, n. 7, p. 1022, doi. 10.1002/cmdc.201390026

By:

Fernández‐Bachiller, María Isabel;
Horatscheck, André;
Lisurek, Michael;
Rademann, Jörg

Publication type:

Article

From On-Target to Off-Target Activity: Identification and Optimisation of Trypanosoma brucei GSK3 Inhibitors and Their Characterisation as Anti- Trypanosoma brucei Drug Discovery Lead Molecules.

Published in:

ChemMedChem, 2013, v. 8, n. 7, p. 1127, doi. 10.1002/cmdc.201300072

By:

Woodland, Andrew;
Grimaldi, Raffaella;
Luksch, Torsten;
Cleghorn, Laura A. T.;
Ojo, Kayode K.;
Van Voorhis, Wesley C.;
Brenk, Ruth;
Frearson, Julie A.;
Gilbert, Ian H.;
Wyatt, Paul G.

Publication type:

Article

Cover Picture: The Lab Oddity Prevails: Discovery of Pan-CDK Inhibitor ( R)- S-Cyclopropyl- S-(4-{[4-{[(1 R,2 R)-2-hydroxy-1-methylpropyl]oxy}-5-(trifluoromethyl)pyrimidin-2-yl]amino}phenyl)sulfoximide (BAY 1000394) for the Treatment of Cancer (ChemMedChem 7/2013)

Published in:

ChemMedChem, 2013, v. 8, n. 7, p. 1021, doi. 10.1002/cmdc.201390025

By:

Lücking, Ulrich;
Jautelat, Rolf;
Krüger, Martin;
Brumby, Thomas;
Lienau, Philip;
Schäfer, Martina;
Briem, Hans;
Schulze, Julia;
Hillisch, Alexander;
Reichel, Andreas;
Wengner, Antje Margret;
Siemeister, Gerhard

Publication type:

Article

Discovery of Piperidine-Linked Pyridine Analogues as Potent Non-nucleoside HIV-1 Reverse Transcriptase Inhibitors.

Published in:

ChemMedChem, 2013, v. 8, n. 7, p. 1117, doi. 10.1002/cmdc.201300130

By:

Chen, Xuwang;
Li, Yuanyuan;
Ding, Shufang;
Balzarini, Jan;
Pannecouque, Christophe;
De Clercq, Erik;
Liu, Huiqing;
Liu, Xinyong

Publication type:

Article

Modification of Triclosan Scaffold in Search of Improved Inhibitors for Enoyl-Acyl Carrier Protein (ACP) Reductase in Toxoplasma gondii.

Published in:

ChemMedChem, 2013, v. 8, n. 7, p. 1138, doi. 10.1002/cmdc.201300050

By:

Stec, Jozef;
Fomovska, Alina;
Afanador, Gustavo A.;
Muench, Stephen P.;
Zhou, Ying;
Lai, Bo‐Shiun;
El Bissati, Kamal;
Hickman, Mark R.;
Lee, Patty J.;
Leed, Susan E.;
Auschwitz, Jennifer M.;
Sommervile, Caroline;
Woods, Stuart;
Roberts, Craig W.;
Rice, David;
Prigge, Sean T.;
McLeod, Rima;
Kozikowski, Alan P.

Publication type:

Article