Works matching IS 18607179 AND DT 2010 AND VI 5 AND IP 11

Results: 24

Preview: ChemMedChem 12/2010.

Published in:: ChemMedChem, 2010, v. 5, n. 11, p. 1955, doi. 10.1002/cmdc.201090053
Publication type:: Article

Hypoxia-Selective Growth Inhibition of Cancer Cells by Furospinosulin-1, a Furanosesterterpene Isolated from an Indonesian Marine Sponge.

Published in:

ChemMedChem, 2010, v. 5, n. 11, p. 1919, doi. 10.1002/cmdc.201000302

By:

Arai, Masayoshi;
Kawachi, Takashi;
Setiawan, Andi;
Kobayashi, Motomasa

Publication type:

Article

Fusion Intermediates of HIV-1 gp41 as Targets for Antibody Production: Design, Synthesis, and HR1-HR2 Complex Purification and Characterization of Generated Antibodies.

Published in:

ChemMedChem, 2010, v. 5, n. 11, p. 1907, doi. 10.1002/cmdc.201000313

By:

Mzoughi, Olfa;
Gaston, Fabrice;
Granados, Giovana C.;
Lakhdar-Ghazal, Faouzi;
Giralt, Ernest;
Bahraoui, Elmostafa

Publication type:

Article

Synthesis of Imidazothiazole-Chalcone Derivatives as Anticancer and Apoptosis Inducing Agents.

Published in:

ChemMedChem, 2010, v. 5, n. 11, p. 1937, doi. 10.1002/cmdc.201000346

By:

Kamal, Ahmed;
Dastagiri, D.;
Ramaiah, M. Janaki;
Reddy, J. Surendranadha;
Bharathi, E. Vijaya;
Srinivas, Chatla;
Pushpavalli, S. N. C. V. L.;
Pal, Dhananjaya;
Pal-Bhadra, Manika

Publication type:

Article

Feeding the Antimalarial Pipeline.

Published in:

ChemMedChem, 2010, v. 5, n. 11, p. 1837, doi. 10.1002/cmdc.201000341

By:

Schlitzer, Martin;
Ortmann, Regina

Publication type:

Article

Synthesis, In Vitro and In Vivo Release Kinetics, and Anti-HIV Activity of A Sustained-Release Prodrug (mPEG-AZT) of 3′-Azido-3′-deoxythymidine (AZT, Zidovudine).

Published in:

ChemMedChem, 2010, v. 5, n. 11, p. 1893, doi. 10.1002/cmdc.201000352

By:

Li, Wenjun;
Chang, Yu;
Zhan, Peng;
Zhang, Na;
Liu, Xinyong;
Pannecouque, Christophe;
De Clercq, Erik

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 11/2010.

Published in:: ChemMedChem, 2010, v. 5, n. 11, p. 1810, doi. 10.1002/cmdc.201090052
Publication type:: Article

A Turning Point in The Fight against HIV.

Published in:

ChemMedChem, 2010, v. 5, n. 11, p. 1799, doi. 10.1002/cmdc.201000338

By:

Williams, Scott D.

Publication type:

Article

Cover Picture: Probing Multidrug-Resistance and Protein-Ligand Interactions with Oxatricyclic Designed Ligands in HIV-1 Protease Inhibitors (ChemMedChem 11/2010).

Published in:

ChemMedChem, 2010, v. 5, n. 11, p. 1797, doi. 10.1002/cmdc.201090049

By:

Ghosh, Arun K.;
Xu, Chun-Xiao;
Rao, Kalapala Venkateswara;
Baldridge, Abigail;
Agniswamy, Johnson;
Wang, Yuan-Fang;
Weber, Irene T.;
Aoki, Manabu;
Miguel, Salcedo Gomez Pedro;
Amano, Masayuki;
Mitsuya, Hiroaki

Publication type:

Article

Development of Peptide and Small-Molecule HIV-1 Fusion Inhibitors that Target gp41.

Published in:

ChemMedChem, 2010, v. 5, n. 11, p. 1813, doi. 10.1002/cmdc.201000289

By:

Cai, Lifeng;
Jiang, Shibo

Publication type:

Article

Graphical Abstract: ChemMedChem 11/2010.

Published in:: ChemMedChem, 2010, v. 5, n. 11, p. 1804, doi. 10.1002/cmdc.201090051
Publication type:: Article

Enzyme Inhibition in Drug Discovery and Development: The Good and the Bad. Edited by Chuang Lu and Albert P. Li.

Published in:

ChemMedChem, 2010, v. 5, n. 11, p. 1949, doi. 10.1002/cmdc.201000315

By:

Costi, Maria Paola

Publication type:

Article

Inhibition of HIV-1 Entry: Multiple Keys to Close the Door.

Published in:

ChemMedChem, 2010, v. 5, n. 11, p. 1825, doi. 10.1002/cmdc.201000292

By:

Hertje, Maria;
Zhou, Mingkui;
Dietrich, Ursula

Publication type:

Article

Toward the First Nonpeptidic Molecular Tong Inhibitor of Wild-Type and Mutated HIV-1 Protease Dimerization.

Published in:

ChemMedChem, 2010, v. 5, n. 11, p. 1899, doi. 10.1002/cmdc.201000308

By:

Vidu, Anamaria;
Dufau, Laure;
Bannwarth, Ludovic;
Soulier, Jean-Louis;
Sicsic, Sames;
Piarulli, Umberto;
Reboud-Ravaux, Michèle;
Ongeri, Sandrine

Publication type:

Article

Studies of Anti-HIV Transcription Inhibitor Quinolones: Identification of Potent N1-Vinyl Derivatives.

Published in:

ChemMedChem, 2010, v. 5, n. 11, p. 1880, doi. 10.1002/cmdc.201000267

By:

Tabarrini, Oriana;
Massari, Serena;
Daelemans, Dirk;
Meschini, Francesco;
Manfroni, Giuseppe;
Bottega, Laura;
Gatto, Barbara;
Palumbo, Manlio;
Pannecouque, Christophe;
Cecchetti, Violetta

Publication type:

Article

Novel Huprine Derivatives with Inhibitory Activity toward β-Amyloid Aggregation and Formation as Disease-Modifying Anti-Alzheimer Drug Candidates.

Published in:

ChemMedChem, 2010, v. 5, n. 11, p. 1855, doi. 10.1002/cmdc.201000322

By:

Viayna, Elisabet;
Gómez, Tània;
Galdeano, Carles;
Ramírez, Lorena;
Ratia, Míriam;
Badia, Albert;
Clos, M. Victòria;
Verdaguer, Ester;
Junyent, Félix;
Camins, Antoni;
Pallàs, Mercè;
Bartolini, Manuela;
Mancini, Francesca;
Andrisano, Vincenza;
Arce, Mariana P.;
Rodríguez-Franco, María Isabel;
Bidon-Chanal, Axel;
Luque, F. Javier;
Camps, Pelayo;
Muñoz-Torrero, Diego

Publication type:

Article

Phosphoramidate Prodrugs Deliver with Potency Against Hepatitis C Virus.

Published in:

ChemMedChem, 2010, v. 5, n. 11, p. 1841, doi. 10.1002/cmdc.201000310

By:

Mehellou, Youcef

Publication type:

Article

Inside Cover: Studies of Anti-HIV Transcription Inhibitor Quinolones: Identification of Potent N1-Vinyl Derivatives (ChemMedChem 11/2010).

Published in:

ChemMedChem, 2010, v. 5, n. 11, p. 1798, doi. 10.1002/cmdc.201090050

By:

Tabarrini, Oriana;
Massari, Serena;
Daelemans, Dirk;
Meschini, Francesco;
Manfroni, Giuseppe;
Bottega, Laura;
Gatto, Barbara;
Palumbo, Manlio;
Pannecouque, Christophe;
Cecchetti, Violetta

Publication type:

Article

Target Profiling of a Small Library of Phosphodiesterase 5 (PDE5) Inhibitors using Chemical Proteomics.

Published in:

ChemMedChem, 2010, v. 5, n. 11, p. 1927, doi. 10.1002/cmdc.201000303

By:

Raijmakers, Reinout;
Dadvar, Poupak;
Pelletier, Sarah;
Gouw, Joost;
Rumpel, Klaus;
Heck, Albert J. R.

Publication type:

Article

Towards the Discovery of New Hypnotic Agents: Synthesis and Preliminary Pharmacological Evaluation of a Novel Class of Dibenzo[ a, d]cycloheptene Derivatives.

Published in:

ChemMedChem, 2010, v. 5, n. 11, p. 1843, doi. 10.1002/cmdc.201000280

By:

Castiglioni, Emiliano;
Di Fabio, Romano;
Togninelli, Andrea;
Brough, Stephen;
Brown, Fiona;
Cin, Michele Dal;
Gianotti, Massimo;
Marchioro, Carla;
Merlo, Giancarlo;
Spinosa, Raffaella;
Wigglesworth, Mark J.;
Botta, Maurizio

Publication type:

Article

The Active Core in a Triazole Peptide Dual-Site Antagonist of HIV-1 gp120.

Published in:

ChemMedChem, 2010, v. 5, n. 11, p. 1871, doi. 10.1002/cmdc.201000222

By:

Umashankara, Muddegowda;
McFadden, Karyn;
Zentner, Isaac;
Schön, Arne;
Rajagopal, Srivats;
Tuzer, Ferit;
Kuriakose, Syna A.;
Contarino, Mark;
LaLonde, Judith;
Freire, Ernesto;
Chaiken, Irwin

Publication type:

Article

Probing Multidrug-Resistance and Protein-Ligand Interactions with Oxatricyclic Designed Ligands in HIV-1 Protease Inhibitors.

Published in:

ChemMedChem, 2010, v. 5, n. 11, p. 1850, doi. 10.1002/cmdc.201000318

By:

Ghosh, Arun K.;
Xu, Chun-Xiao;
Rao, Kalapala Venkateswara;
Baldridge, Abigail;
Agniswamy, Johnson;
Wang, Yuan-Fang;
Weber, Irene T.;
Aoki, Manabu;
Miguel, Salcedo Gomez Pedro;
Amano, Masayuki;
Mitsuya, Hiroaki

Publication type:

Article

A Novel Synthetic Route for the Anti-HIV Drug MC-1220 and its Analogues.

Published in:

ChemMedChem, 2010, v. 5, n. 11, p. 1847, doi. 10.1002/cmdc.201000244

By:

Loksha, Yasser M.;
Globisch, Daniel;
Loddo, Roberta;
Collu, Gabriella;
La Colla, Paolo;
Pedersen, Erik B.

Publication type:

Article

Targeting Protein Kinases for Cancer Therapy. By David J. Matthews and Mary E. Gerritsen.

Published in:

ChemMedChem, 2010, v. 5, n. 11, p. 1948, doi. 10.1002/cmdc.201000398

By:

Kuhn, Daniel

Publication type:

Article