Works matching IS 18607179 AND DT 2020 AND VI 15 AND IP 7

Results: 12

Elucidation of an Allosteric Mode of Action for a Thienopyrazole RORγt Inverse Agonist.

Published in:

ChemMedChem, 2020, v. 15, n. 7, p. 561, doi. 10.1002/cmdc.202000044

By:

Vries, Rens M. J. M.;
Doveston, Richard G.;
Meijer, Femke A.;
Brunsveld, Luc

Publication type:

Article

Shape Similarity by Fractal Dimensionality: An Application in the de novo Design of (−)‐Englerin A Mimetics.

Published in:

ChemMedChem, 2020, v. 15, n. 7, p. 566, doi. 10.1002/cmdc.202000017

By:

Friedrich, Lukas;
Byrne, Ryan;
Treder, Aaron;
Singh, Inderjeet;
Bauer, Christoph;
Gudermann, Thomas;
Mederos y Schnitzler, Michael;
Storch, Ursula;
Schneider, Gisbert

Publication type:

Article

Design, Synthesis, and Dual Evaluation of Quinoline and Quinolinium Iodide Salt Derivatives as Potential Anticancer and Antibacterial Agents.

Published in:

ChemMedChem, 2020, v. 15, n. 7, p. 600, doi. 10.1002/cmdc.202000002

By:

Jin, Guofan;
Xiao, Fuyan;
Li, Zhenwang;
Qi, Xueyong;
Zhao, Lei;
Sun, Xianyu

Publication type:

Article

Tranylcypromine‐Based LSD1 Inhibitors: Structure‐Activity Relationships, Antiproliferative Effects in Leukemia, and Gene Target Modulation.

Published in:

ChemMedChem, 2020, v. 15, n. 7, p. 643, doi. 10.1002/cmdc.201900730

By:

Fioravanti, Rossella;
Romanelli, Annalisa;
Mautone, Nicola;
Di Bello, Elisabetta;
Rovere, Annarita;
Corinti, Davide;
Zwergel, Clemens;
Valente, Sergio;
Rotili, Dante;
Botrugno, Oronza A.;
Dessanti, Paola;
Vultaggio, Stefania;
Vianello, Paola;
Cappa, Anna;
Binda, Claudia;
Mattevi, Andrea;
Minucci, Saverio;
Mercurio, Ciro;
Varasi, Mario;
Mai, Antonello

Publication type:

Article

Covalent Complex of DNA and Bacterial Topoisomerase: Implications in Antibacterial Drug Development.

Published in:

ChemMedChem, 2020, v. 15, n. 7, p. 623, doi. 10.1002/cmdc.201900721

By:

Tiwari, Purushottam B.;
Chapagain, Prem P.;
Seddek, Ahmed;
Annamalai, Thirunavukkarasu;
Üren, Aykut;
Tse‐Dinh, Yuk‐Ching

Publication type:

Article

Comparative in vitro Studies of the Topoisomerase I Inhibition and Anticancer Activities of Metallated N‐Confused Porphyrins and Metallated Porphyrins.

Published in:

ChemMedChem, 2020, v. 15, n. 7, p. 632, doi. 10.1002/cmdc.201900633

By:

Halder, Nyancy;
Dzhemileva, Lilya U.;
Ramazanov, Ilfir R.;
D'yakonov, Vladimir A.;
Dzhemilev, Usein M.;
Rath, Harapriya

Publication type:

Article

Front Cover: Structure‐Based Design, Synthesis, and Biological Evaluation of Triazole‐Based smHDAC8 Inhibitors (ChemMedChem 7/2020).

Published in:

ChemMedChem, 2020, v. 15, n. 7, p. 559, doi. 10.1002/cmdc.201000139

By:

Kalinin, Dmitrii V.;
Jana, Sunit K.;
Pfafenrot, Maxim;
Chakrabarti, Alokta;
Melesina, Jelena;
Shaik, Tajith B.;
Lancelot, Julien;
Pierce, Raymond J.;
Sippl, Wolfgang;
Romier, Christophe;
Jung, Manfred;
Holl, Ralph

Publication type:

Article

A Comparative Study of in vitro Assays for Predicting the Nonspecific Binding of PET Imaging Agents in vivo.

Published in:

ChemMedChem, 2020, v. 15, n. 7, p. 585, doi. 10.1002/cmdc.201900608

By:

Gobbi, Luca;
Mercier, Joël;
Bang‐Andersen, Benny;
Nicolas, Jean‐Marie;
Reilly, John;
Wagner, Björn;
Whitehead, David;
Briard, Emmanuelle;
Maguire, R. Paul;
Borroni, Edilio;
Auberson, Yves P.

Publication type:

Article

Structure‐Based Design, Synthesis, and Biological Evaluation of Triazole‐Based smHDAC8 Inhibitors.

Published in:

ChemMedChem, 2020, v. 15, n. 7, p. 571, doi. 10.1002/cmdc.201900583

By:

Kalinin, Dmitrii V.;
Jana, Sunit K.;
Pfafenrot, Maxim;
Chakrabarti, Alokta;
Melesina, Jelena;
Shaik, Tajith B.;
Lancelot, Julien;
Pierce, Raymond J.;
Sippl, Wolfgang;
Romier, Christophe;
Jung, Manfred;
Holl, Ralph

Publication type:

Article

Cover Feature: A Comparative Study of in vitro Assays for Predicting the Nonspecific Binding of PET Imaging Agents in vivo (ChemMedChem 7/2020).

Published in:

ChemMedChem, 2020, v. 15, n. 7, p. 560, doi. 10.1002/cmdc.201000140

By:

Gobbi, Luca;
Mercier, Joël;
Bang‐Andersen, Benny;
Nicolas, Jean‐Marie;
Reilly, John;
Wagner, Björn;
Whitehead, David;
Briard, Emmanuelle;
Maguire, R. Paul;
Borroni, Edilio;
Auberson, Yves P.

Publication type:

Article

Synthesis, Molecular Docking, and Preliminary Evaluation of 2‐(1,2,3‐Triazoyl)benzaldehydes As Multifunctional Agents for the Treatment of Alzheimer's Disease.

Published in:

ChemMedChem, 2020, v. 15, n. 7, p. 610, doi. 10.1002/cmdc.201900622

By:

Costa, Gabriel P.;
Baldinotti, Rodolfo S. M.;
Fronza, Mariana G.;
Nascimento, José Edmilson R.;
Dias, Ítalo F. C.;
Sonego, Mariana Souza;
Seixas, Fabiana Kömmling;
Collares, Tiago;
Perin, Gelson;
Jacob, Raquel G.;
Savegnago, Lucielli;
Alves, Diego

Publication type:

Article

Biodegradable Periodic Mesoporous Organosilica (BPMO) Loaded with Daunorubicin: A Promising Nanoparticle‐Based Anticancer Drug.

Published in:

ChemMedChem, 2020, v. 15, n. 7, p. 593, doi. 10.1002/cmdc.201900595

By:

Mai, Ngoc Xuan Dat;
Birault, Albane;
Matsumoto, Kotaro;
Ta, Hanh Kieu Thi;
Intasa‐ard, Soontaree Grace;
Morrison, Kendall;
Thang, Phan Bach;
Doan, Tan Le Hoang;
Tamanoi, Fuyuhiko

Publication type:

Article