Works matching IS 18607179 AND DT 2009 AND VI 4 AND IP 1

Results: 21

Guest Editorial: From Chem. Eur. J. to ChemSusChem: All from ChemPubSoc Europe.

Published in:

ChemMedChem, 2009, v. 4, n. 1, p. 6, doi. 10.1002/cmdc.200800385

By:

Koch, Wolfram

Publication type:

Article

Synthesis and Evaluation of 1,1′-Hydrocarbylenebis(indazol-3-ols) as Potential Antimalarial Drugs.

Published in:

ChemMedChem, 2009, v. 4, n. 1, p. 78, doi. 10.1002/cmdc.200800176

By:

Martins Alho, Miriam;
García-Sánchez, Rory N.;
Nogal-Ruiz, Juan José;
Escario, José Antonio;
Gómez-Barrio, Alicia;
Martínez-Fernández, Antonio R.;
Arán, Vicente J.

Publication type:

Article

Preview: ChemMedChem 2/2009.

Published in:: ChemMedChem, 2009, v. 4, n. 1, p. 130, doi. 10.1002/cmdc.200990001
Publication type:: Article

Hit Expansion through Computational Selectivity Searching.

Published in:

ChemMedChem, 2009, v. 4, n. 1, p. 52, doi. 10.1002/cmdc.200800304

By:

Stumpfe, Dagmar;
Frizler, Maxim;
Sisay, Mihiret T.;
Batista, José;
Vogt, Ingo;
Gütschow, Michael;
Bajorath, Jürgen

Publication type:

Article

Evolution of Tertiary Carbinamine BACE-1 Inhibitors: Aβ Reduction in Rhesus CSF upon Oral Dosing.

Published in:

ChemMedChem, 2009, v. 4, n. 1, p. 37, doi. 10.1002/cmdc.200800308

By:

Nantermet, Philippe G.;
Rajapakse, Hemaka A.;
Stanton, Mathew G.;
Stauffer, Shaun R.;
Barrow, James C.;
Gregro, Allison R.;
Moore, Keith P.;
Steinbeiser, Melissa A.;
Swestock, John;
Selnick, Harold G.;
Graham, Samuel L.;
McGaughey, Georgia B.;
Colussi, Dennis;
Lai, Ming-Tain;
Sankaranarayanan, Sethu;
Simon, Adam J.;
Munshi, Sanjeev;
Cook, Jacquelynn J.;
Holahan, Marie A.;
Michener, Maria S.

Publication type:

Article

Mixed-Model QSAR at the Glucocorticoid Receptor: Predicting the Binding Mode and Affinity of Psychotropic Drugs.

Published in:

ChemMedChem, 2009, v. 4, n. 1, p. 100, doi. 10.1002/cmdc.200800274

By:

Spreafico, Morena;
Ernst, Beat;
Lill, Markus A.;
Smiesko, Martin;
Vedani, Angelo

Publication type:

Article

Cover Picture: Diphenyl Ether Non-Nucleoside Reverse Transcriptase Inhibitors with Excellent Potency Against Resistant Mutant Viruses and Promising Pharmacokinetic Properties (ChemMedChem 1/2009).

Published in:

ChemMedChem, 2009, v. 4, n. 1, p. 1, doi. 10.1002/cmdc.200990000

By:

Sweeney, Zachary K.;
Kennedy-Smith, Joshua J.;
Wu, Jeffrey;
Arora, Nidhi;
Billedeau, J. Roland;
Davidson, James P.;
Fretland, Jennifer;
Hang, Julie Q.;
Heilek, Gabrielle M.;
Harris, Seth F.;
Hirschfeld, Donald;
Inbar, Petra;
Javanbakht, Hassan;
Jernelius, Jesper A.;
Jin, Qingwu;
Li, Yu;
Liang, Weiling;
Roetz, Ralf;
Sarma, Keshab;
Smith, Mark

Publication type:

Article

Assessing the Bioisosterism of the Trifluoromethyl Group with a Protease Probe.

Published in:

ChemMedChem, 2009, v. 4, n. 1, p. 49, doi. 10.1002/cmdc.200800321

By:

Jagodzinska, Monika;
Huguenot, Florent;
Candiani, Gabriele;
Zanda, Matteo

Publication type:

Article

From Molecular Shape to Potent Bioactive Agents II: Fragment-Based de novo Design.

Published in:

ChemMedChem, 2009, v. 4, n. 1, p. 45, doi. 10.1002/cmdc.200800314

By:

Proschak, Ewgenij;
Sander, Kerstin;
Zettl, Heiko;
Tanrikulu, Yusuf;
Rau, Oliver;
Schneider, Petra;
Schubert-Zsilavecz, Manfred;
Stark, Holger;
Schneider, Gisbert

Publication type:

Article

Semi-Synthetic Ecdysteroids as Gene-Switch Actuators: Synthesis, Structure-Activity Relationships, and Prospective ADME Properties.

Published in:

ChemMedChem, 2009, v. 4, n. 1, p. 55, doi. 10.1002/cmdc.200800280

By:

Lapenna, Silvia;
Dinan, Laurence;
Friz, Jennifer;
Hopfinger, Anton J.;
Liu, Jianzhong;
Hormann, Robert E.

Publication type:

Article

Diphenyl Ether Non-Nucleoside Reverse Transcriptase Inhibitors with Excellent Potency Against Resistant Mutant Viruses and Promising Pharmacokinetic Properties.

Published in:

ChemMedChem, 2009, v. 4, n. 1, p. 88, doi. 10.1002/cmdc.200800262

By:

Sweeney, Zachary K.;
Kennedy-Smith, Joshua J.;
Wu, Jeffrey;
Arora, Nidhi;
Billedeau, J. Roland;
Davidson, James P.;
Fretland, Jennifer;
Hang, Julie Q.;
Heilek, Gabrielle M.;
Harris, Seth F.;
Hirschfeld, Donald;
Inbar, Petra;
Javanbakht, Hassan;
Jernelius, Jesper A.;
Jin, Qingwu;
Li, Yu;
Liang, Weiling;
Roetz, Ralf;
Sarma, Keshab;
Smith, Mark

Publication type:

Article

Editorial: A Journal with Impact.

Published in:: ChemMedChem, 2009, v. 4, n. 1, p. 3, doi. 10.1002/cmdc.200800369
Publication type:: Article

Stereocontrolled Synthesis and Pharmacological Evaluation of Azetidine-2,3-Dicarboxylic Acids at NMDA Receptors.

Published in:

ChemMedChem, 2009, v. 4, n. 1, p. 110, doi. 10.1002/cmdc.200800226

By:

Sivaprakasam, Mangaleswaran;
Hansen, Kasper B.;
David, Olivier;
Nielsen, Birgitte;
Traynelis, Stephen F.;
Clausen, Rasmus P.;
Couty, François;
Bunch, Lennart

Publication type:

Article

How to Extend the Use of Grid-Based Interaction Energy Maps from Chemistry to Biotopics.

Published in:

ChemMedChem, 2009, v. 4, n. 1, p. 29, doi. 10.1002/cmdc.200800259

By:

Caron, Giulia;
Nurisso, Alessandra;
Ermondi, Giuseppe

Publication type:

Article

ATP-Noncompetitive Inhibitors of CDK-Cyclin Complexes.

Published in:

ChemMedChem, 2009, v. 4, n. 1, p. 19, doi. 10.1002/cmdc.200800185

By:

Orzáez, Mar;
Gortat, Anna;
Mondragón, Laura;
Bachs, Oriol;
Pérez-Payá, Enrique

Publication type:

Article

C6-Unsubstituted Pyrazolo[3,4- d]pyrimidines Are Dual Src/Abl Inhibitors Effective against Imatinib Mesylate Resistant Chronic Myeloid Leukemia Cell Lines.

Published in:

ChemMedChem, 2009, v. 4, n. 1, p. 118, doi. 10.1002/cmdc.200800320

By:

Santucci, Maria Alessandra;
Corradi, Valentina;
Mancini, Manuela;
Manetti, Fabrizio;
Radi, Marco;
Schenone, Silvia;
Botta, Maurizio

Publication type:

Article

Graphical Abstract: ChemMedChem 1/2009.

Published in:: ChemMedChem, 2009, v. 4, n. 1, p. 7, doi. 10.1002/cmdc.200990003
Publication type:: Article

From Molecular Shape to Potent Bioactive Agents I: Bioisosteric Replacement of Molecular Fragments.

Published in:

ChemMedChem, 2009, v. 4, n. 1, p. 41, doi. 10.1002/cmdc.200800313

By:

Proschak, Ewgenij;
Zettl, Heiko;
Tanrikulu, Yusuf;
Weisel, Martin;
Kriegl, Jan M.;
Rau, Oliver;
Schubert-Zsilavecz, Manfred;
Schneider, Gisbert

Publication type:

Article

Solute-Binding Sites in ABC Transporters for Recognition, Occlusion and Trans-Inhibition.

Published in:

ChemMedChem, 2009, v. 4, n. 1, p. 25, doi. 10.1002/cmdc.200800328

By:

Parcej, David;
Tampé, Robert

Publication type:

Article

Virtual Screening and Biological Characterization of Novel Histone Arginine Methyltransferase PRMT1 Inhibitors.

Published in:

ChemMedChem, 2009, v. 4, n. 1, p. 69, doi. 10.1002/cmdc.200800301

By:

Heinke, Ralf;
Spannhoff, Astrid;
Meier, Rene;
Trojer, Patrick;
Bauer, Ingo;
Jung, Manfred;
Sippl, Wolfgang

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 1/2009.

Published in:: ChemMedChem, 2009, v. 4, n. 1, p. 14, doi. 10.1002/cmdc.200990002
Publication type:: Article