Works matching AU Supuran, Claudiu T.

Results: 882

Repositioning FDA-Approved Sulfonamide-Based Drugs as Potential Carbonic Anhydrase Inhibitors in Trypanosoma cruzi : Virtual Screening and In Vitro Studies.

Published in:

Pharmaceuticals (14248247), 2025, v. 18, n. 5, p. 669, doi. 10.3390/ph18050669

By:

Ortiz-Pérez, Eyra;
Moreno-Rodríguez, Adriana;
Delgado-Maldonado, Timoteo;
Ortega-Balleza, Jessica L.;
González-González, Alonzo;
Paz-González, Alma D.;
Vázquez, Karina;
Avalos-Navarro, Guadalupe;
Giovannuzzi, Simone;
Supuran, Claudiu T.;
Rivera, Gildardo

Publication type:

Article

Acetazolamide-Loaded Nanoparticle Based on Modified Hyaluronic Acid as Delivery System to Target Carbonic Anhydrases in Escherichia coli.

Published in:

International Journal of Molecular Sciences, 2025, v. 26, n. 10, p. 4908, doi. 10.3390/ijms26104908

By:

Verdoliva, Valentina;
De Luca, Viviana;
Supuran, Claudiu T.;
De Luca, Stefania;
Capasso, Clemente

Publication type:

Article

Calixarenes Incorporating Sulfonamide Moieties: Versatile Ligands for Carbonic Anhydrases Inhibition.

Published in:

Chemistry - A European Journal, 2022, v. 28, n. 6, p. 1, doi. 10.1002/chem.202103527

By:

Sbravati, Davide;
Bonardi, Alessandro;
Bua, Silvia;
Angeli, Andrea;
Ferraroni, Marta;
Nocentini, Alessio;
Casnati, Alessandro;
Gratteri, Paola;
Sansone, Francesco;
Supuran, Claudiu T.

Publication type:

Article

Ein niedermolekulares Ligand-Wirkstoff-Konjugat zur Behandlung von Carboanhydrase IX exprimierenden Tumoren.

Published in:

Angewandte Chemie, 2014, v. 126, n. 16, p. 4315, doi. 10.1002/ange.201310709

By:

Krall, Nikolaus;
Pretto, Francesca;
Decurtins, Willy;
Bernardes, Gonçalo J. L.;
Supuran, Claudiu T.;
Neri, Dario

Publication type:

Article

[(Cp-R)M(CO)<sub>3</sub>] (M=Re or <sup>99m</sup>Tc) Arylsulfonamide, Arylsulfamide, and Arylsulfamate Conjugates for Selective Targeting of Human Carbonic Anhydrase IX.

Published in:

Angewandte Chemie, 2012, v. 124, n. 14, p. 3410, doi. 10.1002/ange.201107333

By:

Can, Daniel;
Spingler, Bernhard;
Schmutz, Paul;
Mendes, Filipa;
Raposinho, Paula;
Fernandes, Célia;
Carta, Fabrizio;
Innocenti, Alessio;
Santos, Isabel;
Supuran, Claudiu T.;
Alberto, Roger

Publication type:

Article

Organometallic compounds with biologically active molecules: in vitro antibacterial and antifungal activity of some 1,1′-(dicarbohydrazono) ferrocenes and their cobalt(II), copper(II), nickel(II) and zinc(II) complexes.

Published in:

Applied Organometallic Chemistry, 2005, v. 19, n. 12, p. 1207, doi. 10.1002/aoc.944

By:

Chohan, Zahid H.;
Supuran, Claudiu T.

Publication type:

Article

Synthesis of antibacterial and antifungal cobalt(II), copper(II), nickel(II) and zinc(II) complexes with bis-(1,1′-disubstituted ferrocenyl)thiocarbohydrazone and bis-(1,1′-disubstituted ferrocenyl)carbohydrazone.

Published in:

Applied Organometallic Chemistry, 2004, v. 18, n. 7, p. 305, doi. 10.1002/aoc.620

By:

Chohan, Zahid H.;
Khan, Khalid M.;
Supuran, Claudiu T.

Publication type:

Article

Progress in the development of human carbonic anhydrase inhibitors and their pharmacological applications: Where are we today?

Published in:

Medicinal Research Reviews, 2020, v. 40, n. 6, p. 2485, doi. 10.1002/med.21713

By:

Mishra, Chandra B.;
Tiwari, Manisha;
Supuran, Claudiu T.

Publication type:

Article

Inhibition of carbonic anhydrase IX targets primary tumors, metastases, and cancer stem cells: Three for the price of one.

Published in:

Medicinal Research Reviews, 2018, v. 38, n. 6, p. 1799, doi. 10.1002/med.21497

By:

Supuran, Claudiu T.;
Alterio, Vincenzo;
Di Fiore, Anna;
D’ Ambrosio, Katia;
Carta, Fabrizio;
Monti, Simona Maria;
De Simone, Giuseppina

Publication type:

Article

Therapeutic applications of glycosidic carbonic anhydrase inhibitors.

Published in:

Medicinal Research Reviews, 2009, v. 29, n. 3, p. 419, doi. 10.1002/med.20141

By:

Winum, Jean-Yves;
Poulsen,, Sally-Ann;
Supuran, Claudiu T.

Publication type:

Article

Therapeutic potential of sulfamides as enzyme inhibitors.

Published in:

Medicinal Research Reviews, 2006, v. 26, n. 6, p. 767, doi. 10.1002/med.20068

By:

Winum, Jean-Yves;
Scozzafava, Andrea;
Montero, Jean-Louis;
Supuran, Claudiu T.

Publication type:

Article

Sulfamates and their therapeutic potential.

Published in:

Medicinal Research Reviews, 2005, v. 25, n. 2, p. 186, doi. 10.1002/med.20021

By:

Winum, Jean-Yves;
Scozzafava, Andrea;
Montero, Jean-Louis;
Supuran, Claudiu T.

Publication type:

Article

Protease inhibitors of the sulfonamide type: Anticancer, antiinflammatory, and antiviral agents.

Published in:

Medicinal Research Reviews, 2003, v. 23, n. 5, p. 535, doi. 10.1002/med.10047

By:

Claudiu T. Supuran;
Angela Casini;
Andrea Scozzafava

Publication type:

Article

Carbonic anhydrase inhibitors.

Published in:

Medicinal Research Reviews, 2003, v. 23, n. 2, p. 146, doi. 10.1002/med.10025

By:

Supuran, Claudiu T.;
Scozzafava, Andrea;
Casini, Angela

Publication type:

Article

Bacterial protease inhibitors.

Published in:

Medicinal Research Reviews, 2002, v. 22, n. 4, p. 329, doi. 10.1002/med.10007

By:

Supuran, Claudiu T.;
Scozzafava, Andrea;
Clare, Brian W.

Publication type:

Article

The structural comparison between membrane-associated human carbonic anhydrases provides insights into drug design of selective inhibitors.

Published in:

Biopolymers, 2014, v. 101, n. 7, p. 769, doi. 10.1002/bip.22456

By:

Alterio, Vincenzo;
Pan, Peiwen;
Parkkila, Seppo;
Buonanno, Martina;
Supuran, Claudiu T.;
Monti, Simona M.;
Simone, Giuseppina

Publication type:

Article

Post-translational modifications in tumor-associated carbonic anhydrases.

Published in:

Amino Acids, 2022, v. 54, n. 4, p. 543, doi. 10.1007/s00726-021-03063-y

By:

Di Fiore, Anna;
Supuran, Claudiu T.;
Scaloni, Andrea;
De Simone, Giuseppina

Publication type:

Article

Development of a New LC-MS/MS Screening Method for Detection of 120 NPS and 43 Drugs in Blood.

Published in:

Separations (2297-8739), 2021, v. 8, n. 11, p. 1, doi. 10.3390/separations8110221

By:

Vaiano, Fabio;
Berto, Elisabetta;
Mineo, Maria;
Pietrosemoli, Laura;
Rubicondo, Jolanda;
Supuran, Claudiu T.;
Carta, Fabrizio

Publication type:

Article

Blocking HIF signaling via novel inhibitors of CA9 and APE1/Ref-1 dramatically affects pancreatic cancer cell survival.

Published in:

Scientific Reports, 2018, v. 8, n. 1, p. 1, doi. 10.1038/s41598-018-32034-9

By:

Logsdon, Derek P.;
Shah, Fenil;
Carta, Fabrizio;
Supuran, Claudiu T.;
Kamocka, Malgorzata;
Jacobsen, Max H.;
Sandusky, George E.;
Kelley, Mark R.;
Fishel, Melissa L.

Publication type:

Article

Synthesis and Biological Evaluation of Coumarin-Linked 4-Anilinomethyl-1,2,3-Triazoles as Potent Inhibitors of Carbonic Anhydrases IX and XIII Involved in Tumorigenesis.

Published in:

Metabolites (2218-1989), 2021, v. 11, n. 4, p. 225, doi. 10.3390/metabo11040225

By:

Thacker, Pavitra S.;
Tiwari, Prerna L.;
Angeli, Andrea;
Srikanth, Danaboina;
Swain, Baijayantimala;
Arifuddin, Mohammed;
Supuran, Claudiu T.

Publication type:

Article

Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment.

Published in:

Metabolites (2218-1989), 2020, v. 10, n. 10, p. 412, doi. 10.3390/metabo10100412

By:

Angeli, Andrea;
Carta, Fabrizio;
Nocentini, Alessio;
Winum, Jean-Yves;
Zalubovskis, Raivis;
Akdemir, Atilla;
Onnis, Valentina;
Eldehna, Wagdy M.;
Capasso, Clemente;
Simone, Giuseppina De;
Monti, Simona Maria;
Carradori, Simone;
Donald, William A.;
Dedhar, Shoukat;
Supuran, Claudiu T.

Publication type:

Article

Design, Synthesis, and Biological Evaluation of 1,2,3-Triazole-linked triazino[5,6-b]indole-benzene sulfonamide Conjugates as Potent Carbonic Anhydrase I, II, IX, and XIII Inhibitors.

Published in:

Metabolites (2218-1989), 2020, v. 10, n. 5, p. 200, doi. 10.3390/metabo10050200

By:

Chinchilli, Krishna Kartheek;
Angeli, Andrea;
Thacker, Pavitra S.;
Korra, Laxman Naik;
Biswas, Rashmita;
Arifuddin, Mohammed;
Supuran, Claudiu T.

Publication type:

Article

Synthesis and Biological Evaluation of Imidazo[2,1-b]Thiazole based Sulfonyl Piperazines as Novel Carbonic Anhydrase II Inhibitors.

Published in:

Metabolites (2218-1989), 2020, v. 10, n. 4, p. 136, doi. 10.3390/metabo10040136

By:

Manasa, Kesari Lakshmi;
Pujitha, Sravya;
Sethi, Aaftaab;
Arifuddin, Mohammed;
Alvala, Mallika;
Angeli, Andrea;
Supuran, Claudiu T.

Publication type:

Article

Anion Inhibition Studies of the β-Class Carbonic Anhydrase CAS3 from the Filamentous Ascomycete Sordaria macrospora.

Published in:

Metabolites (2218-1989), 2020, v. 10, n. 3, p. 93, doi. 10.3390/metabo10030093

By:

Vullo, Daniela;
Lehneck, Ronny;
Donald, William A.;
Pöggeler, Stefanie;
Supuran, Claudiu T.

Publication type:

Article

Sulfonamide Inhibition Profile of the β-Carbonic Anhydrase from Malassezia restricta, An Opportunistic Pathogen Triggering Scalp Conditions.

Published in:

Metabolites (2218-1989), 2020, v. 10, n. 1, p. 39, doi. 10.3390/metabo10010039

By:

Del Prete, Sonia;
Angeli, Andrea;
Ghobril, Cynthia;
Hitce, Julien;
Clavaud, Cécile;
Marat, Xavier;
Supuran, Claudiu T.;
Capasso, Clemente

Publication type:

Article

Anion Inhibition Profile of the β-Carbonic Anhydrase from the Opportunist Pathogenic Fungus Malassezia restricta Involved in Dandruff and Seborrheic Dermatitis.

Published in:

Metabolites (2218-1989), 2019, v. 9, n. 7, p. 147, doi. 10.3390/metabo9070147

By:

Prete, Sonia Del;
Angeli, Andrea;
Ghobril, Cynthia;
Hitce, Julien;
Clavaud, Cécile;
Marat, Xavier;
Supuran, Claudiu T.;
Capasso, Clemente

Publication type:

Article

Activation Studies of the β-Carbonic Anhydrase from the Pathogenic Protozoan Entamoeba histolytica with Amino Acids and Amines.

Published in:

Metabolites (2218-1989), 2019, v. 9, n. 2, p. 26, doi. 10.3390/metabo9020026

By:

Bua, Silvia;
Haapanen, Susanna;
Kuuslahti, Marianne;
Parkkila, Seppo;
Supuran, Claudiu T.

Publication type:

Article

Benzamide-4-Sulfonamides Are Effective Human Carbonic Anhydrase I, II, VII, and IX Inhibitors.

Published in:

Metabolites (2218-1989), 2018, v. 8, n. 2, p. 37, doi. 10.3390/metabo8020037

By:

Abdoli, Morteza;
Bozdag, Murat;
Angeli, Andrea;
Supuran, Claudiu T.

Publication type:

Article

Amino Acids as Building Blocks for Carbonic Anhydrase Inhibitors.

Published in:

Metabolites (2218-1989), 2018, v. 8, n. 2, p. 36, doi. 10.3390/metabo8020036

By:

Chiaramonte, Niccolò;
Romanelli, Maria Novella;
Teodori, Elisabetta;
Supuran, Claudiu T.

Publication type:

Article

Carbonic Anhydrases and Metabolism.

Published in:

2018

By:

Supuran, Claudiu T.

Publication type:

Editorial

Rethinking the Combination of Proton Exchanger Inhibitors in Cancer Therapy.

Published in:

Metabolites (2218-1989), 2018, v. 8, n. 1, p. 2, doi. 10.3390/metabo8010002

By:

Iessi, Elisabetta;
Logozzi, Mariantonia;
Mizzoni, Davide;
Di Raimo, Rossella;
Supuran, Claudiu T.;
Fais, Stefano

Publication type:

Article

An Overview of the Bacterial Carbonic Anhydrases.

Published in:

Metabolites (2218-1989), 2017, v. 7, n. 4, p. 56, doi. 10.3390/metabo7040056

By:

Supuran, Claudiu T.;
Capasso, Clemente

Publication type:

Article

Carbonic Anhydrase Inhibition and the Management of Hypoxic Tumors.

Published in:

Metabolites (2218-1989), 2017, v. 7, n. 3, p. 48, doi. 10.3390/metabo7030048

By:

Supuran, Claudiu T.

Publication type:

Article

Cloning, polymorphism, and inhibition of beta-carbonic anhydrase of Helicobacter pylori.

Published in:

2008

By:

Morishita S;
Nishimori I;
Minakuchi T;
Onishi S;
Takeuchi H;
Sugiura T;
Vullo D;
Scozzafava A;
Supuran CT;
Morishita, Saori;
Nishimori, Isao;
Minakuchi, Tomoko;
Onishi, Saburo;
Takeuchi, Hiroaki;
Sugiura, Tetsuro;
Vullo, Daniela;
Scozzafava, Andrea;
Supuran, Claudiu T

Publication type:

journal article

Selective inhibition of carbonic anhydrase IX over carbonic anhydrase XII in breast cancer cells using benzene sulfonamides: Disconnect between activity and growth inhibition.

Published in:

PLoS ONE, 2018, v. 13, n. 11, p. 1, doi. 10.1371/journal.pone.0207417

By:

Mboge, Mam Y.;
Chen, Zhijuan;
Wolff, Alyssa;
Mathias, John V.;
Tu, Chingkuang;
Brown, Kevin D.;
Bozdag, Murat;
Carta, Fabrizio;
Supuran, Claudiu T.;
McKenna, Robert;
Frost, Susan C.

Publication type:

Article

Antibacterial carbonic anhydrase inhibitors targeting Vibrio cholerae enzymes.

Published in:

Expert Opinion on Therapeutic Targets, 2024, v. 28, n. 7, p. 623, doi. 10.1080/14728222.2024.2369622

By:

Gheibzadeh, Mohammad Sadegh;
Capasso, Clemente;
Supuran, Claudiu T.;
Zolfaghari Emameh, Reza

Publication type:

Article

Are tumour-associated carbonic anhydrases genuine therapeutic targets for photodynamic therapy?

Published in:

Expert Opinion on Therapeutic Targets, 2023, v. 27, n. 9, p. 817, doi. 10.1080/14728222.2023.2255380

By:

Merabti, Amina;
Richeter, Sébastien;
Supuran, Claudiu T.;
Clement, Sébastien;
Winum, Jean-Yves

Publication type:

Article

An overview of novel antimicrobial carbonic anhydrase inhibitors.

Published in:

Expert Opinion on Therapeutic Targets, 2023, v. 27, n. 10, p. 897, doi. 10.1080/14728222.2023.2263914

By:

Supuran, Claudiu T

Publication type:

Article

Saccharin Inhibits Carbonic Anhydrases: Possible Explanation for its Unpleasant Metallic Aftertaste.

Published in:

Angewandte Chemie International Edition, 2007, v. 46, n. 40, p. 7697, doi. 10.1002/anie.200701189

By:

Köhler, Karen;
Hillebrecht, Alexander;
Schulze Wischeler, Johannes;
Innocenti, Alessio;
Heine, Andreas;
Supuran, Claudiu T.;
Klebe, Gerhard

Publication type:

Article

A Journey Around Boronic Acids: Sulfonyl Hydrazone‐Containing Derivatives as Carbonic Anhydrase Inhibitors.

Published in:

Chemical Biology & Drug Design, 2025, v. 105, n. 4, p. 1, doi. 10.1111/cbdd.70108

By:

Anakök, Deniz A.;
Angeli, Andrea;
D'Agostino, Ilaria;
Renzi, Gioele;
Massardi, Maria Luisa;
Tavani, Camilla;
Çete, Servet;
Carradori, Simone;
Ronca, Roberto;
Capasso, Clemente;
Carta, Fabrizio;
Supuran, Claudiu T.

Publication type:

Article

4-Substituted Pyridine-3-Sulfonamides as Carbonic Anhydrase Inhibitors Modified by Click Tailing: Synthesis, Activity, and Docking Studies.

Published in:

International Journal of Molecular Sciences, 2025, v. 26, n. 8, p. 3817, doi. 10.3390/ijms26083817

By:

Szafrański, Krzysztof;
Sławiński, Jarosław;
Kawiak, Anna;
Chojnacki, Jarosław;
Kosno, Michał;
Ammara, Andrea;
Supuran, Claudiu T.

Publication type:

Article

Multifaceted Sulfonamide-Derived Thiosemicarbazones: Combining Metal Chelation and Carbonic Anhydrases Inhibition in Anticancer Therapy.

Published in:

International Journal of Molecular Sciences, 2025, v. 26, n. 3, p. 1225, doi. 10.3390/ijms26031225

By:

Martínez-Montiel, Mónica;
Arrighi, Giulia;
Begines, Paloma;
González-Bakker, Aday;
Puerta, Adrián;
Fernandes, Miguel X.;
Merino-Montiel, Penélope;
Montiel-Smith, Sara;
Nocentini, Alessio;
Supuran, Claudiu T.;
Padrón, José M.;
Fernández-Bolaños, José G.;
López, Óscar

Publication type:

Article

Exploring the Inhibition of Toxoplasma gondii α-Carbonic Anhydrase by Sulfonamides: Insights into Potential Drug Targeting.

Published in:

International Journal of Molecular Sciences, 2025, v. 26, n. 1, p. 116, doi. 10.3390/ijms26010116

By:

Giovannuzzi, Simone;
De Luca, Viviana;
Capasso, Clemente;
Supuran, Claudiu T.

Publication type:

Article

Phosphorus versus Sulfur: Discovery of Benzenephosphonamidates as Versatile Sulfonamide‐Mimic Chemotypes Acting as Carbonic Anhydrase Inhibitors.

Published in:

Chemistry - A European Journal, 2019, v. 25, n. 5, p. 1188, doi. 10.1002/chem.201805039

By:

Nocentini, Alessio;
Gratteri, Paola;
Supuran, Claudiu T.

Publication type:

Article

Deciphering the Mechanism of Human Carbonic Anhydrases Inhibition with Sulfocoumarins: Computational and Experimental Studies.

Published in:

Chemistry - A European Journal, 2018, v. 24, n. 31, p. 7840, doi. 10.1002/chem.201800941

By:

Nocentini, Alessio;
Carta, Fabrizio;
Tanc, Muhammet;
Selleri, Silvia;
Supuran, Claudiu T.;
Bazzicalupi, Carla;
Gratteri, Paola

Publication type:

Article

Exponential Activation of Carbonic Anhydrase by Encapsulation in Dynameric Host Matrices with Chiral Discrimination.

Published in:

Chemistry - A European Journal, 2018, v. 24, n. 3, p. 715, doi. 10.1002/chem.201704605

By:

Barboiu, Mihail;
Zhang, Yan;
Supuran, Claudiu T.

Publication type:

Article

Inside Cover: Effective Access to Multivalent Inhibitors of Carbonic Anhydrases Promoted by Peptide Bioconjugation (Chem. Eur. J. 28/2017).

Published in:

Chemistry - A European Journal, 2017, v. 23, n. 28, p. 6704, doi. 10.1002/chem.201700987

By:

Kanfar, Nasreddine;
Tanc, Muhammet;
Dumy, Pascal;
Supuran, Claudiu T.;
Ulrich, Sébastien;
Winum, Jean‐Yves

Publication type:

Article

Effective Access to Multivalent Inhibitors of Carbonic Anhydrases Promoted by Peptide Bioconjugation.

Published in:

Chemistry - A European Journal, 2017, v. 23, n. 28, p. 6788, doi. 10.1002/chem.201700241

By:

Kanfar, Nasreddine;
Tanc, Muhammet;
Dumy, Pascal;
Supuran, Claudiu T.;
Ulrich, Sébastien;
Winum, Jean‐Yves

Publication type:

Article

A Combined Crystallographic and Theoretical Study Explains the Capability of Carboxylic Acids to Adopt Multiple Binding Modes in the Active Site of Carbonic Anhydrases.

Published in:

Chemistry - A European Journal, 2016, v. 22, n. 1, p. 97, doi. 10.1002/chem.201503748

By:

Langella, Emma;
D'Ambrosio, Katia;
D'Ascenzio, Melissa;
Carradori, Simone;
Monti, Simona M.;
Supuran, Claudiu T.;
De Simone, Giuseppina

Publication type:

Article

Crystal structure and chemical inhibition of essential schistosome host-interactive virulence factor carbonic anhydrase SmCA.

Published in:

Communications Biology, 2019, v. 2, n. 1, p. N.PAG, doi. 10.1038/s42003-019-0578-0

By:

Da'dara, Akram A.;
Angeli, Andrea;
Ferraroni, Marta;
Supuran, Claudiu T.;
Skelly, Patrick J.

Publication type:

Article