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A Photoswitchable Agonist for the Histamine H<sub>3</sub> Receptor, a Prototypic Family A G‐Protein‐Coupled Receptor.
- Published in:
- Angewandte Chemie, 2019, v. 131, n. 14, p. 4579, doi. 10.1002/ange.201813110
- By:
- Publication type:
- Article
Photoswitching the Efficacy of a Small‐Molecule Ligand for a Peptidergic GPCR: from Antagonism to Agonism.
- Published in:
- Angewandte Chemie, 2018, v. 130, n. 36, p. 11782, doi. 10.1002/ange.201804875
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- Publication type:
- Article
The histamine H<sub>3</sub> receptor: from gene cloning to H<sub>3</sub> receptor drugs.
- Published in:
- Nature Reviews Drug Discovery, 2005, v. 4, n. 2, p. 107, doi. 10.1038/nrd1631
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- Publication type:
- Article
Bromo-Cyclobutenaminones as New Covalent UDP- N -Acetylglucosamine Enolpyruvyl Transferase (MurA) Inhibitors.
- Published in:
- Pharmaceuticals (14248247), 2020, v. 13, n. 11, p. 362, doi. 10.3390/ph13110362
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- Publication type:
- Article
In Silico Veritas: The Pitfalls and Challenges of Predicting GPCR-Ligand Interactions.
- Published in:
- Pharmaceuticals (14248247), 2011, v. 4, n. 9, p. 1196, doi. 10.3390/ph4091196
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- Publication type:
- Article
Photoswitching the Efficacy of a Small‐Molecule Ligand for a Peptidergic GPCR: from Antagonism to Agonism.
- Published in:
- Angewandte Chemie International Edition, 2018, v. 57, n. 36, p. 11608, doi. 10.1002/anie.201804875
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- Publication type:
- Article
To Target or Not to Target Schistosoma mansoni Cyclic Nucleotide Phosphodiesterase 4A?
- Published in:
- International Journal of Molecular Sciences, 2023, v. 24, n. 7, p. 6817, doi. 10.3390/ijms24076817
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- Publication type:
- Article
Interrogating the Essential Bacterial Cell Division Protein FtsQ with Fragments Using Target Immobilized NMR Screening (TINS).
- Published in:
- International Journal of Molecular Sciences, 2019, v. 20, n. 15, p. 3684, doi. 10.3390/ijms20153684
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- Publication type:
- Article
KLIFS: a structural kinase-ligand interaction database.
- Published in:
- Nucleic Acids Research, 2016, v. 44, n. 1, p. D365, doi. 10.1093/nar/gkv1082
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- Publication type:
- Article
Puckering the Planar Landscape of Fragments: Design and Synthesis of a 3D Cyclobutane Fragment Library.
- Published in:
- ChemMedChem, 2022, v. 17, n. 9, p. 1, doi. 10.1002/cmdc.202200113
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- Publication type:
- Article
3D‐e‐Chem: Structural Cheminformatics Workflows for Computer‐Aided Drug Discovery.
- Published in:
- ChemMedChem, 2018, v. 13, n. 6, p. 614, doi. 10.1002/cmdc.201700754
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- Publication type:
- Article
Development of a microfluidic confocal fluorescence detection system for the hyphenation of nano-LC to on-line biochemical assays.
- Published in:
- Analytical & Bioanalytical Chemistry, 2010, v. 398, n. 7/8, p. 3023, doi. 10.1007/s00216-010-4210-x
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- Publication type:
- Article
Strain-dependent effects of the histamine H<sub>4</sub> receptor antagonist JNJ7777120 in a murine model of acute skin inflammation.
- Published in:
- Experimental Dermatology, 2012, v. 21, n. 1, p. 32, doi. 10.1111/j.1600-0625.2011.01396.x
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- Publication type:
- Article
Function-specific virtual screening for GPCR ligands using a combined scoring method.
- Published in:
- Scientific Reports, 2016, p. 28288, doi. 10.1038/srep28288
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- Publication type:
- Article
A Qualitative Model for the Histamine H<sub>3</sub> Receptor Explaining Agonistic and Antagonistic Activity Simultaneously.
- Published in:
- Archiv der Pharmazie, 2000, v. 333, n. 8, p. 254, doi. 10.1002/1521-4184(20008)333:8<254::AID-ARDP254>3.0.CO;2-G
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- Publication type:
- Article
Effects of Histamine H<sub>4</sub> Receptor Ligands in a Mouse Model of Gastric Ulceration.
- Published in:
- Pharmacology, 2012, v. 89, n. 5/6, p. 287, doi. 10.1159/000337736
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- Publication type:
- Article
Fragment Screening Yields a Small‐Molecule Stabilizer of 14‐3‐3 Dimers That Modulates Client Protein Interactions.
- Published in:
- ChemBioChem, 2022, v. 23, n. 17, p. 1, doi. 10.1002/cbic.202200178
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- Publication type:
- Article
SAR exploration of the non‐imidazole histamine H<sub>3</sub> receptor ligand ZEL‐H16 reveals potent inverse agonism.
- Published in:
- Archiv der Pharmazie, 2023, v. 356, n. 1, p. 1, doi. 10.1002/ardp.202200451
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- Publication type:
- Article
Green Drug Discovery: Novel Fragment Space from the Biomass-Derived Molecule Dihydrolevoglucosenone (Cyrene TM).
- Published in:
- Molecules, 2023, v. 28, n. 4, p. 1777, doi. 10.3390/molecules28041777
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- Publication type:
- Article
Sex- and Histamine-Dependent Long-Term Cognitive Effects of Methamphetamine Exposure.
- Published in:
- Neuropsychopharmacology, 2007, v. 32, n. 3, p. 665, doi. 10.1038/sj.npp.1301091
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- Publication type:
- Article
Assembly of a ?-? stack of ligands in the binding site of an acetylcholine-binding protein.
- Published in:
- Nature Communications, 2013, v. 4, n. 5, p. 1875, doi. 10.1038/ncomms2900
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- Publication type:
- Article
A Photoswitchable Agonist for the Histamine H<sub>3</sub> Receptor, a Prototypic Family A G‐Protein‐Coupled Receptor.
- Published in:
- Angewandte Chemie International Edition, 2019, v. 58, n. 14, p. 4531, doi. 10.1002/anie.201813110
- By:
- Publication type:
- Article
Predicting the target landscape of kinase inhibitors using 3D convolutional neural networks.
- Published in:
- PLoS Computational Biology, 2023, v. 19, n. 9, p. 1, doi. 10.1371/journal.pcbi.1011301
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- Publication type:
- Article
Pharmacological characterization of the new histamine H4 receptor agonist VUF 8430.
- Published in:
- 2009
- By:
- Publication type:
- journal article
Molecular and biochemical pharmacology of the histamine H4 receptor.
- Published in:
- 2009
- By:
- Publication type:
- journal article
KLIFS: an overhaul after the first 5 years of supporting kinase research.
- Published in:
- Nucleic Acids Research, 2021, v. 49, n. D1, p. D562, doi. 10.1093/nar/gkaa895
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- Publication type:
- Article
Crystal structure of the EphA4 protein tyrosine kinase domain in the apo- and dasatinib-bound state
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- FEBS Letters, 2011, v. 585, n. 22, p. 3593, doi. 10.1016/j.febslet.2011.10.028
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- Publication type:
- Article
Covalent Inhibition of the Histamine H3 Receptor.
- Published in:
- Molecules, 2019, v. 24, n. 24, p. 4541, doi. 10.3390/molecules24244541
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- Publication type:
- Article
Public-private partnerships influencing the initiation and duration of clinical trials for neglected tropical diseases.
- Published in:
- PLoS Neglected Tropical Diseases, 2023, v. 17, n. 11, p. 1, doi. 10.1371/journal.pntd.0011760
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- Publication type:
- Article
Structure-Activity Relationships of Quinoxaline-Based 5-HT<sub>3</sub>A and 5-HT<sub>3</sub>AB Receptor-Selective Ligands.
- Published in:
- ChemMedChem, 2013, v. 8, n. 6, p. 946, doi. 10.1002/cmdc.201300032
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- Publication type:
- Article
Back Cover: Structure-Activity Relationships of Quinoxaline-Based 5-HT<sub>3</sub>A and 5-HT<sub>3</sub>AB Receptor-Selective Ligands (ChemMedChem 6/2013).
- Published in:
- ChemMedChem, 2013, v. 8, n. 6, p. 1020, doi. 10.1002/cmdc.201390024
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- Publication type:
- Article
Combining Quantum Mechanical Ligand Conformation Analysis and Protein Modeling to Elucidate GPCR-Ligand Binding Modes.
- Published in:
- ChemMedChem, 2013, v. 8, n. 1, p. 49, doi. 10.1002/cmdc.201200412
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- Publication type:
- Article
Discovery of a New Class of Non-imidazole Oxazoline-Based Histamine H<sub>3</sub> Receptor (H<sub>3</sub>R) Inverse Agonists.
- Published in:
- ChemMedChem, 2009, v. 4, n. 7, p. 1063, doi. 10.1002/cmdc.200900055
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- Publication type:
- Article
Towards Small-Molecule CXCR3 Ligands with Clinical Potential.
- Published in:
- ChemMedChem, 2008, v. 3, n. 6, p. 861, doi. 10.1002/cmdc.200700365
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- Publication type:
- Article
RIDING THE WAVE OF A NEW SCIENTIFIC FIELD: HOW PIONEERS CREATE OPPORTUNITIES AMIDST HYPE AND HOPE.
- Published in:
- Frontiers of Entrepreneurship Research, 2019, v. 39, p. 80
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- Publication type:
- Article
Diazepam-bound GABA<sub>A</sub> receptor models identify new benzodiazepine binding-site ligands.
- Published in:
- Nature Chemical Biology, 2012, v. 8, n. 5, p. 455, doi. 10.1038/nchembio.917
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- Publication type:
- Article
Evaluation of phthalazinone phosphodiesterase inhibitors with improved activity and selectivity against Trypanosoma cruzi.
- Published in:
- 2020
- By:
- Publication type:
- journal article