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Wohldefinierte polymere Paclitaxel-Prodrugs über eine Grafting-From-Methode ausgehend vom Arzneistoff.
Published in:
Angewandte Chemie, 2016, v. 128, n. 39, p. 11967, doi. 10.1002/ange.201605892
By:
- Louage, Benoit;
- Nuhn, Lutz;
- Risseeuw, Martijn D. P.;
- Vanparijs, Nane;
- De Coen, Ruben;
- Karalic, Izet;
- Van Calenbergh, Serge;
- De Geest, Bruno G.
Publication type:
Article
Hamamelitannin Analogues that Modulate Quorum Sensing as Potentiators of Antibiotics against Staphylococcus aureus.
Published in:
Angewandte Chemie, 2016, v. 128, n. 22, p. 6661, doi. 10.1002/ange.201601973
By:
- Vermote, Arno;
- Brackman, Gilles;
- Risseeuw, Martijn D. P.;
- Vanhoutte, Bieke;
- Cos, Paul;
- Van Hecke, Kristof;
- Breyne, Koen;
- Meyer, Evelyne;
- Coenye, Tom;
- Van Calenbergh, Serge
Publication type:
Article
Radiosynthesis, in vitro and preliminary biological evaluation of [18F]2‐amino‐4‐((2‐((3‐fluorobenzyl)oxy)benzyl)(2‐((3‐(fluoromethyl)benzyl)oxy)benzyl)amino)butanoic acid, a novel alanine serine cysteine transporter 2 inhibitor‐based positron emission tomography tracer
Published in:
Journal of Labelled Compounds & Radiopharmaceuticals, 2020, v. 63, n. 10, p. 442, doi. 10.1002/jlcr.3863
By:
- Baguet, Tristan;
- Bouton, Jakob;
- Janssens, Jonas;
- Pauwelyn, Glenn;
- Verhoeven, Jeroen;
- Descamps, Benedicte;
- Van Calenbergh, Serge;
- Vanhove, Christian;
- De Vos, Filip
Publication type:
Article
Cytotoxic Activity of Laserpitium latifolium L. Extract and Its Daucane and Phenylpropanoid Constituents.
Published in:
Records of Natural Products, 2013, v. 7, n. 3, p. 245
By:
- Popović, Višnja;
- Heyerick, Arne;
- Petrović, Silvana;
- Van Calenbergh, Serge;
- Karalić, Izet;
- Niketić, Marjan;
- Deforce, Dieter
Publication type:
Article
Practical and Divergent Synthesis of Carbocyclic Pyrazolo[3,4‐d]pyrimidine Nucleoside Analogues.
Published in:
European Journal of Organic Chemistry, 2024, v. 27, n. 19, p. 1, doi. 10.1002/ejoc.202400181
By:
- Van de Velde, Ewout;
- Van Hauwermeiren, Anouk;
- Van Pelt, Natascha;
- Matheeussen, An;
- Caljon, Guy;
- Van Calenbergh, Serge
Publication type:
Article
Well-Defined Polymer-Paclitaxel Prodrugs by a Grafting-from-Drug Approach.
Published in:
Angewandte Chemie International Edition, 2016, v. 55, n. 39, p. 11791, doi. 10.1002/anie.201605892
By:
- Louage, Benoit;
- Nuhn, Lutz;
- Risseeuw, Martijn D. P.;
- Vanparijs, Nane;
- De Coen, Ruben;
- Karalic, Izet;
- Van Calenbergh, Serge;
- De Geest, Bruno G.
Publication type:
Article
Hamamelitannin Analogues that Modulate Quorum Sensing as Potentiators of Antibiotics against Staphylococcus aureus.
Published in:
Angewandte Chemie International Edition, 2016, v. 55, n. 22, p. 6551, doi. 10.1002/anie.201601973
By:
- Vermote, Arno;
- Brackman, Gilles;
- Risseeuw, Martijn D. P.;
- Vanhoutte, Bieke;
- Cos, Paul;
- Van Hecke, Kristof;
- Breyne, Koen;
- Meyer, Evelyne;
- Coenye, Tom;
- Van Calenbergh, Serge
Publication type:
Article
Cloning and Characterization of Trypanosoma congolense and T. vivax Nucleoside Transporters Reveal the Potential of P1-Type Carriers for the Discovery of Broad-Spectrum Nucleoside-Based Therapeutics against Animal African Trypanosomiasis.
Published in:
International Journal of Molecular Sciences, 2023, v. 24, n. 4, p. 3144, doi. 10.3390/ijms24043144
By:
- Ungogo, Marzuq A.;
- Aldfer, Mustafa M.;
- Natto, Manal J.;
- Zhuang, Hainan;
- Chisholm, Robyn;
- Walsh, Katy;
- McGee, MarieClaire;
- Ilbeigi, Kayhan;
- Asseri, Jamal Ibrahim;
- Burchmore, Richard J. S.;
- Caljon, Guy;
- Van Calenbergh, Serge;
- De Koning, Harry P.
Publication type:
Article
Ex Vivo Feedback Control of Neurotransmission Using a Photocaged Adenosine A1 Receptor Agonist.
Published in:
International Journal of Molecular Sciences, 2022, v. 23, n. 16, p. 8887, doi. 10.3390/ijms23168887
By:
- Craey, Erine;
- Hulpia, Fabian;
- Spanoghe, Jeroen;
- Manzella, Simona;
- Larsen, Lars E.;
- Sprengers, Mathieu;
- De Bundel, Dimitri;
- Smolders, Ilse;
- Carrette, Evelien;
- Delbeke, Jean;
- Vonck, Kristl;
- Boon, Paul;
- Van Calenbergh, Serge;
- Wadman, Wytse J.;
- Raedt, Robrecht
Publication type:
Article
A Toxoplasma gondii Oxopurine Transporter Binds Nucleobases and Nucleosides Using Different Binding Modes.
Published in:
International Journal of Molecular Sciences, 2022, v. 23, n. 2, p. 710, doi. 10.3390/ijms23020710
By:
- Campagnaro, Gustavo D.;
- Elati, Hamza A. A.;
- Balaska, Sofia;
- Martin Abril, Maria Esther;
- Natto, Manal J.;
- Hulpia, Fabian;
- Lee, Kelly;
- Sheiner, Lilach;
- Van Calenbergh, Serge;
- de Koning, Harry P.
Publication type:
Article
The bovine CD1D gene has an unusual gene structure and is expressed but cannot present α-galactosylceramide with a C26 fatty acid.
Published in:
International Immunology, 2013, v. 25, n. 2, p. 91, doi. 10.1093/intimm/dxs092
By:
- Nguyen, Thi Kim Anh;
- Koets, Ad P.;
- Vordermeier, Martin;
- Jervis, Peter J.;
- Cox, Liam R.;
- Graham, Simon P.;
- Santema, Wiebren J.;
- Moody, D. Branch;
- van Calenbergh, Serge;
- Zajonc, Dirk M.;
- Besra, Gurdyal S.;
- Van Rhijn, Ildiko
Publication type:
Article
Towards New Antimalarial Drugs: Synthesis of Non-Hydrolyzable Phosphate Mimics as Feed for a Predictive QSAR Study on 1-Deoxy- D-xylulose-5-phosphate Reductoisomerase Inhibitors.
Published in:
Chemistry & Biodiversity, 2008, v. 5, n. 4, p. 643, doi. 10.1002/cbdv.200890060
By:
- Gießmann, Dirk;
- Heidler, Philipp;
- Haemers, Timothy;
- Van Calenbergh, Serge;
- Reichenberg, Armin;
- Jomaa, Hassan;
- Weidemeyer, Claus;
- Sanderbrand, Silke;
- Wiesner, Jochen;
- Link, Andreas
Publication type:
Article
6‐Methyl‐7‐Aryl‐7‐Deazapurine Nucleosides as Anti‐Trypanosoma cruzi Agents: Structure‐Activity Relationship and in vivo Efficacy.
Published in:
ChemMedChem, 2021, v. 16, n. 14, p. 2231, doi. 10.1002/cmdc.202100144
By:
- Lin, Cai;
- Ferreira de Almeida Fiuza, Ludmila;
- Cardoso Santos, Camila;
- Ferreira Nunes, Daniela;
- Cruz Moreira, Otacílio;
- Bouton, Jakob;
- Karalic, Izet;
- Maes, Louis;
- Caljon, Guy;
- Hulpia, Fabian;
- Nazaré C. Soeiro, Maria;
- Van Calenbergh, Serge
Publication type:
Article
4"‐O‐Alkylated α‐Galactosylceramide Analogues as iNKT‐Cell Antigens: Synthetic, Biological, and Structural Studies.
Published in:
ChemMedChem, 2019, v. 14, n. 1, p. 147, doi. 10.1002/cmdc.201800649
By:
- Janssens, Jonas;
- Bitra, Aruna;
- Wang, Jing;
- Decruy, Tine;
- Venken, Koen;
- van der Eycken, Johan;
- Elewaut, Dirk;
- Zajonc, Dirk M.;
- van Calenbergh, Serge
Publication type:
Article
Design, Synthesis, and Biological Evaluation of Bivalent Ligands Targeting Dopamine D2‐Like Receptors and the μ‐Opioid Receptor.
Published in:
ChemMedChem, 2018, v. 13, n. 9, p. 944, doi. 10.1002/cmdc.201700787
By:
- Qian, Mingcheng;
- Vasudevan, Lakshmi;
- Huysentruyt, Jelle;
- Risseeuw, Martijn D. P.;
- Stove, Christophe;
- Vanderheyden, Patrick M. L.;
- Van Craenenbroeck, Kathleen;
- Van Calenbergh, Serge
Publication type:
Article
The Quorum Sensing Inhibitor Hamamelitannin Increases Antibiotic Susceptibility of Staphylococcus aureus Biofilms by Affecting Peptidoglycan Biosynthesis and eDNA Release.
Published in:
Scientific Reports, 2016, p. 20321, doi. 10.1038/srep20321
By:
- Brackman, Gilles;
- Breyne, Koen;
- De Rycke, Riet;
- Vermote, Arno;
- Van Nieuwerburgh, Filip;
- Meyer, Evelyne;
- Van Calenbergh, Serge;
- Coenye, Tom
Publication type:
Article
An In Silico Approach for Modelling T-Helper Polarizing iNKT Cell Agonists.
Published in:
PLoS ONE, 2014, v. 9, n. 1, p. 1, doi. 10.1371/journal.pone.0087000
By:
- De Spiegeleer, Anton;
- Wynendaele, Evelien;
- Vandekerckhove, Matthias;
- Stalmans, Sofie;
- Boucart, Maxime;
- Van Den Noortgate, Nele;
- Venken, Koen;
- Van Calenbergh, Serge;
- Aspeslagh, Sandrine;
- Elewaut, Dirk
Publication type:
Article
Crystal Structures of Bovine CD1d Reveal Altered αGalCer Presentation and a Restricted A' Pocket Unable to Bind Long-Chain Glycolipids.
Published in:
PLoS ONE, 2012, v. 7, n. 10, p. 1, doi. 10.1371/journal.pone.0047989
By:
- Wang, Jing;
- Guillaume, Joren;
- Pauwels, Nora;
- Van Calenbergh, Serge;
- Van Rhijn, Ildiko;
- Zajonc, Dirk M.
Publication type:
Article
Structure-Activity Relationship of Cinnamaldehyde Analogs as Inhibitors of AI-2 Based Quorum Sensing and Their Effect on Virulence of Vibrio spp.
Published in:
PLoS ONE, 2011, v. 6, n. 1, p. 1, doi. 10.1371/journal.pone.0016084
By:
- Brackman, Gilles;
- Celen, Shari;
- Hillaert, Ulrik;
- Calenbergh, Serge Van;
- Cos, Paul;
- Maes, Louis;
- Nelis, Hans J.;
- Coenye, Tom
Publication type:
Article
Ceramide‐Templated Macrolactams: Total Synthesis and Biological Evaluation of Macrocyclic α‐Galactosylceramide Analogues and their Aglycons.
Published in:
European Journal of Organic Chemistry, 2019, v. 2019, n. 12, p. 2253, doi. 10.1002/ejoc.201801839
By:
- Janssens, Jonas;
- Van der Eycken, Johan;
- Van Calenbergh, Serge
Publication type:
Article
Regioselective Ring Opening of 1,3‐Dioxane‐Type Acetals in Carbohydrates.
Published in:
European Journal of Organic Chemistry, 2018, v. 2018, n. 46, p. 6405, doi. 10.1002/ejoc.201801245
By:
- Janssens, Jonas;
- Risseeuw, Martijn D. P.;
- Van der Eycken, Johan;
- Van Calenbergh, Serge
Publication type:
Article
Synthesis and Conformational Analysis of 2′-Deoxy-2′-(3-methoxybenzamido)adenosine, a rational-designed inhibitor of trypanosomal glyceraldehyde phosphate dehydrogenase (GAPDH).
Published in:
Helvetica Chimica Acta, 1994, v. 77, n. 3, p. 631, doi. 10.1002/hlca.19940770306
By:
- Van Calenbergh, Serge;
- Van Den Eeckhout, Elfride;
- Herdewijn, Piet;
- De Bruyn, André;
- Verlinde, Christophe;
- Hol, Wim;
- Callens, Mia;
- Van Aerschot, Arthur;
- Rozenski, Jef
Publication type:
Article
Phenethyl-4-ANPP: A Marginally Active Byproduct Suggesting a Switch in Illicit Fentanyl Synthesis Routes.
Published in:
Journal of Analytical Toxicology, 2022, v. 46, n. 4, p. 350, doi. 10.1093/jat/bkab032
By:
- Vandeputte, Marthe M;
- Krotulski, Alex J;
- Hulpia, Fabian;
- Calenbergh, Serge Van;
- Stove, Christophe P
Publication type:
Article
Report on a New Opioid NPS: Chemical and In Vitro Functional Characterization of a Structural Isomer of the MT-45 Derivative Diphenpipenol.
Published in:
Journal of Analytical Toxicology, 2021, v. 45, n. 2, p. 134, doi. 10.1093/jat/bkaa066
By:
- Cannaert, Annelies;
- Hulpia, Fabian;
- Risseeuw, Martijn;
- Uytfanghe, Katleen Van;
- Deconinck, Eric;
- Calenbergh, Serge Van;
- Blanckaert, Peter;
- Stove, Christophe
Publication type:
Article
First Report on Brorphine: The Next Opioid on the Deadly New Psychoactive Substance Horizon?
Published in:
Journal of Analytical Toxicology, 2020, v. 44, n. 9, p. 937, doi. 10.1093/jat/bkaa094
By:
- Verougstraete, Nick;
- Vandeputte, Marthe M;
- Lyphout, Cathelijne;
- Cannaert, Annelies;
- Hulpia, Fabian;
- Calenbergh, Serge Van;
- Verstraete, Alain G;
- Stove, Christophe
Publication type:
Article
Combining tubercidin and cordycepin scaffolds results in highly active candidates to treat late-stage sleeping sickness.
Published in:
Nature Communications, 2019, v. 10, n. 1, p. N.PAG, doi. 10.1038/s41467-019-13522-6
By:
- Hulpia, Fabian;
- Mabille, Dorien;
- Campagnaro, Gustavo D.;
- Schumann, Gabriela;
- Maes, Louis;
- Roditi, Isabel;
- Hofer, Anders;
- de Koning, Harry P.;
- Caljon, Guy;
- Van Calenbergh, Serge
Publication type:
Article
Mycobacterium tuberculosis Thymidine Monophosphate Kinase Inhibitors: Biological Evaluation and Conformational Analysis of 2'- and 3'-Modified Thymidine Analogues.
Published in:
European Journal of Organic Chemistry, 2003, v. 2003, n. 15, p. 2911, doi. 10.1002/ejoc.200300177
By:
- Philippe Van Rompaey;
- Koen Nauwelaerts;
- Veerle Vanheusden;
- Jef Rozenski;
- Hélène Munier-Lehmann;
- Piet Herdewijn;
- Serge Van Calenbergh
Publication type:
Article
Galactose-modified iNKT cell agonists stabilized by an induced fit of CD1d prevent tumour metastasis.
Published in:
EMBO Journal, 2011, v. 30, n. 11, p. 2294, doi. 10.1038/emboj.2011.145
By:
- Aspeslagh, Sandrine;
- Li, Yali;
- Yu, Esther Dawen;
- Pauwels, Nora;
- Trappeniers, Matthias;
- Girardi, Enrico;
- Decruy, Tine;
- Van Beneden, Katrien;
- Venken, Koen;
- Drennan, Michael;
- Leybaert, Luc;
- Wang, Jing;
- Franck, Richard W;
- Van Calenbergh, Serge;
- Zajonc, Dirk M;
- Elewaut, Dirk
Publication type:
Article
Host metabolites stimulate the bacterial proton motive force to enhance the activity of aminoglycoside antibiotics.
Published in:
PLoS Pathogens, 2019, v. 15, n. 4, p. 1, doi. 10.1371/journal.ppat.1007697
By:
- Crabbé, Aurélie;
- Ostyn, Lisa;
- Staelens, Sorien;
- Rigauts, Charlotte;
- Risseeuw, Martijn;
- Dhaenens, Maarten;
- Daled, Simon;
- Van Acker, Heleen;
- Deforce, Dieter;
- Van Calenbergh, Serge;
- Coenye, Tom
Publication type:
Article
Alternative Reagents for Methotrexate as Immobilizing Anchor Moieties in the Optimization of MASPIT: Synthesis and Biological Evaluation.
Published in:
ChemBioChem, 2015, v. 16, n. 5, p. 834, doi. 10.1002/cbic.201402702
By:
- De Clercq, Dries J. H.;
- Risseeuw, Martijn D. P.;
- Karalic, Izet;
- De Smet, Anne‐Sophie;
- Defever, Dieter;
- Tavernier, Jan;
- Lievens, Sam;
- Van Calenbergh, Serge
Publication type:
Article
Unbreakable Codes in Electrospun Fibers: Digitally Encoded Polymers to Stop Medicine Counterfeiting.
Published in:
Advanced Materials, 2010, v. 22, n. 24, p. 2657, doi. 10.1002/adma.201000130
By:
- Huang, Chaobo;
- Lucas, Bart;
- Vervaet, Chris;
- Braeckmans, Kevin;
- Van Calenbergh, Serge;
- Karalic, Izet;
- Vandewoestyne, Mado;
- Deforce, Dieter;
- Demeester, Jo;
- De Smedt, Stefaan C.
Publication type:
Article
Phenotypic Evaluation of Nucleoside Analogues against Trypanosoma cruzi Infection: In Vitro and In Vivo Approaches.
Published in:
Molecules, 2022, v. 27, n. 22, p. 8087, doi. 10.3390/molecules27228087
By:
- Fiuza, Ludmila F. de A.;
- Batista, Denise G. J.;
- Girão, Roberson D.;
- Hulpia, Fabian;
- Finamore-Araújo, Paula;
- Aldfer, Mustafa M.;
- Elmahallawy, Ehab Kotb;
- De Koning, Harry P.;
- Moreira, Otacílio;
- Van Calenbergh, Serge;
- Soeiro, Maria de Nazaré C.
Publication type:
Article
The Trypanosoma cruzi TcrNT2 Nucleoside Transporter Is a Conduit for the Uptake of 5-F-2′-Deoxyuridine and Tubercidin Analogues.
Published in:
Molecules, 2022, v. 27, n. 22, p. 0, doi. 10.3390/molecules27228045
By:
- Aldfer, Mustafa M.;
- Alfayez, Ibrahim A.;
- Elati, Hamza A. A.;
- Gayen, Nilanjana;
- Elmahallawy, Ehab Kotb;
- Milena Murillo, Ana;
- Marsiccobetre, Sabrina;
- Van Calenbergh, Serge;
- Silber, Ariel M.;
- de Koning, Harry P.
Publication type:
Article
4E Interacting Protein as a Potential Novel Drug Target for Nucleoside Analogues in Trypanosoma brucei.
Published in:
Microorganisms, 2021, v. 9, n. 4, p. 826, doi. 10.3390/microorganisms9040826
By:
- Mabille, Dorien;
- Cardoso Santos, Camila;
- Hendrickx, Rik;
- Claes, Mathieu;
- Takac, Peter;
- Clayton, Christine;
- Hendrickx, Sarah;
- Hulpia, Fabian;
- Maes, Louis;
- Van Calenbergh, Serge;
- Caljon, Guy
Publication type:
Article
Trapping mammalian protein complexes in viral particles.
Published in:
Nature Communications, 2016, v. 7, n. 4, p. 11416, doi. 10.1038/ncomms11416
By:
- Eyckerman, Sven;
- Titeca, Kevin;
- Van Quickelberghe, Emmy;
- Cloots, Eva;
- Verhee, Annick;
- Samyn, Noortje;
- De Ceuninck, Leentje;
- Timmerman, Evy;
- De Sutter, Delphine;
- Lievens, Sam;
- Van Calenbergh, Serge;
- Gevaert, Kris;
- Tavernier, Jan
Publication type:
Article
Determination of paramethoxyamphetamine and other amphetamine-related designer drugs by liquid chromatography/sonic spray ionization mass spectrometry.
Published in:
Rapid Communications in Mass Spectrometry: RCM, 2002, v. 16, n. 9, p. 865, doi. 10.1002/rcm.657
By:
- Mortier, Kjell A.;
- Dams, Riet;
- Lambert, Willy E.;
- Letter, Els A. De;
- Calenbergh, Serge Van;
- Leenheer, André P. De
Publication type:
Article
Synthesis of α-Aryl-Substituted and Conformationally Restricted Fosmidomycin Analogues as Promising Antimalarials.
Published in:
European Journal of Organic Chemistry, 2006, v. 2006, n. 17, p. 3856, doi. 10.1002/ejoc.200600202
By:
- Timothy Haemers;
- Jochen Wiesner;
- Roger Busson;
- Hassan Jomaa;
- Serge Van Calenbergh
Publication type:
Article
Analytical characterization of "etonitazepyne," a new pyrrolidinyl‐containing 2‐benzylbenzimidazole opioid sold online.
Published in:
Drug Testing & Analysis, 2021, v. 13, n. 9, p. 1627, doi. 10.1002/dta.3113
By:
- Blanckaert, Peter;
- Balcaen, Margot;
- Vanhee, Céline;
- Risseeuw, Martijn;
- Canfyn, Michaël;
- Desmedt, Bart;
- Van Calenbergh, Serge;
- Deconinck, Eric
Publication type:
Article
Report on a novel emerging class of highly potent benzimidazole NPS opioids: Chemical and in vitro functional characterization of isotonitazene.
Published in:
Drug Testing & Analysis, 2020, v. 12, n. 4, p. 422, doi. 10.1002/dta.2738
By:
- Blanckaert, Peter;
- Cannaert, Annelies;
- Van Uytfanghe, Katleen;
- Hulpia, Fabian;
- Deconinck, Eric;
- Van Calenbergh, Serge;
- Stove, Christophe
Publication type:
Article
1-(1-Arylethylpiperidin-4-yl)thymine Analogs as Antimycobacterial TMPK Inhibitors.
Published in:
Molecules, 2020, v. 25, n. 12, p. 2805, doi. 10.3390/molecules25122805
By:
- Jian, Yanlin;
- Hulpia, Fabian;
- D. P. Risseeuw, Martijn;
- Forbes, He Eun;
- Caljon, Guy;
- Munier-Lehmann, Hélène;
- I. M. Boshoff, Helena;
- Van Calenbergh, Serge;
- Geronikaki, Athina
Publication type:
Article
Design, Synthesis and Characterization of a New Series of Fluorescent Metabotropic Glutamate Receptor Type 5 Negative Allosteric Modulators.
Published in:
Molecules, 2020, v. 25, n. 7, p. 1532, doi. 10.3390/molecules25071532
By:
- Fernández-Dueñas, Víctor;
- Qian, Mingcheng;
- Argerich, Josep;
- Amaral, Carolina;
- Risseeuw, Martijn D.P.;
- Van Calenbergh, Serge;
- Ciruela, Francisco;
- Filipek, Sławomir
Publication type:
Article
Synthesis of Extended Uridine Phosphonates Derived from an Allosteric P2Y2 Receptor Ligand.
Published in:
Molecules, 2014, v. 19, n. 4, p. 4313, doi. 10.3390/molecules19044313
By:
- Lijun Song;
- Risseeuw, Martijn D. P.;
- Karalic, Izet;
- Barrett, Matthew O.;
- Brown, Kyle A.;
- Kendall Harden, T.;
- Van Calenbergh, Serge
Publication type:
Article
Synthetic Fosmidomycin Analogues with Altered Chelating Moieties Do Not Inhibit 1-Deoxy-D-xylulose 5-phosphate Reductoisomerase or Plasmodium falciparum Growth In Vitro.
Published in:
Molecules, 2014, v. 19, n. 2, p. 2571, doi. 10.3390/molecules19022571
By:
- Chofor, René;
- Risseeuw, Martijn D. P.;
- Pouyez, Jenny;
- Johny, Chinchu;
- Wouters, Johan;
- Dowd, Cynthia S.;
- Couch, Robin D.;
- Van Calenbergh, Serge
Publication type:
Article
New fluoroethyl phenylalanine analogues as potential LAT1-targeting PET tracers for glioblastoma.
Published in:
Scientific Reports, 2019, v. 9, n. 1, p. 1, doi. 10.1038/s41598-019-40013-x
By:
- Verhoeven, Jeroen;
- Hulpia, Fabian;
- Kersemans, Ken;
- Bolcaen, Julie;
- De Lombaerde, Stef;
- Goeman, Jan;
- Descamps, Benedicte;
- Hallaert, Giorgio;
- Van den Broecke, Caroline;
- Deblaere, Karel;
- Vanhove, Christian;
- Van der Eycken, Johan;
- Van Calenbergh, Serge;
- Goethals, Ingeborg;
- De Vos, Filip
Publication type:
Article
Nanobody-mediated SPECT/CT imaging reveals the spatiotemporal expression of programmed death-ligand 1 in response to a CD8+ T cell and iNKT cell activating mRNA vaccine.
Published in:
Theranostics, 2023, v. 13, n. 15, p. 5483, doi. 10.7150/thno.85106
By:
- Ertveldt, Thomas;
- Meulewaeter, Sofie;
- De Vlaeminck, Yannick;
- Olarte, Oscar;
- Broos, Katrijn;
- Van Calenbergh, Serge;
- Bourgeois, Stephanie;
- Deprez, Joke;
- Heremans, Yves;
- Goyvaerts, Cleo;
- Staels, Willem;
- De Smedt, Stefaan;
- Dewitte, Heleen;
- Devoogdt, Nick;
- Keyaerts, Marleen;
- Verbeke, Rein;
- Barbé, Kurt;
- Lentacker, Ine;
- Breckpot, Karine
Publication type:
Article
Targeting an Aromatic Hotspot in Plasmodium falciparum 1-Deoxy- d-xylulose-5-phosphate Reductoisomerase with β-Arylpropyl Analogues of Fosmidomycin.
Published in:
ChemMedChem, 2016, v. 11, n. 18, p. 2024, doi. 10.1002/cmdc.201600249
By:
- Sooriyaarachchi, Sanjeewani;
- Chofor, René;
- Risseeuw, Martijn D. P.;
- Bergfors, Terese;
- Pouyez, Jenny;
- Dowd, Cynthia S.;
- Maes, Louis;
- Wouters, Johan;
- Jones, T. Alwyn;
- Van Calenbergh, Serge;
- Mowbray, Sherry L.
Publication type:
Article
A 'Clickable' MTX Reagent as a Practical Tool for Profiling Small-Molecule-Intracellular Target Interactions via MASPIT.
Published in:
ChemMedChem, 2013, v. 8, n. 3, p. 521, doi. 10.1002/cmdc.201200493
By:
- Risseeuw, Martijn D. P.;
- De Clercq, Dries J. H.;
- Lievens, Sam;
- Hillaert, Ulrik;
- Sinnaeve, Davy;
- Van den Broeck, Freya;
- Martins, José C.;
- Tavernier, Jan;
- Van Calenbergh, Serge
Publication type:
Article
The Synthesis and in vivo Evaluation of 2′,2′-Difluoro KRN7000.
Published in:
ChemMedChem, 2009, v. 4, n. 3, p. 329, doi. 10.1002/cmdc.200800348
By:
- Leung, Leo;
- Tomassi, Cyrille;
- Van Beneden, Katrien;
- Decruy, Tine;
- Trappeniers, Matthias;
- Elewaut, Dirk;
- Gao, Yifang;
- Elliott, Tim;
- Al-Shamkhani, Aymen;
- Ottensmeier, Christian;
- Werner, Jörn M.;
- Williams, Anthony;
- Van Calenbergh, Serge;
- Linclau, Bruno
Publication type:
Article
Synthesis and in vitro Evaluation of α-GalCer Epimers.
Published in:
ChemMedChem, 2008, v. 3, n. 7, p. 1061, doi. 10.1002/cmdc.200800021
By:
- Trappeniers, Matthias;
- Goormans, Stijn;
- Van Beneden, Katrien;
- Decruy, Tine;
- Linclau, Bruno;
- Al-Shamkhani, Aymen;
- Elliott, Tim;
- Ottensmeier, Christian;
- Werner, Joern M.;
- Elewaut, Dirk;
- Van Calenbergh, Serge
Publication type:
Article
Synthesis and Biological Evaluation of Bicyclic Nucleosides as Inhibitors of M. tuberculosis Thymidylate Kinase.
Published in:
ChemMedChem, 2006, v. 1, n. 10, p. 1081, doi. 10.1002/cmdc.200600028
By:
- Van Daele, Ineke;
- Munier-Lehmann, Hélène;
- Hendrickx, Pieter M. S.;
- Marchal, Gilles;
- Chavarot, Pierre;
- Froeyen, Matheus;
- Qing, Li;
- Martins, José C.;
- Van Calenbergh, Serge
Publication type:
Article

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