Found: 5

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  • Rational evolution for altering the ligand preference of estrogen receptor alpha.

    Published in:
    Protein Science: A Publication of the Protein Society, 2024, v. 33, n. 4, p. 1, doi. 10.1002/pro.4940
    By:
    • Eerlings, Roy;
    • Gupta, Purvi;
    • Lee, Xiao Yin;
    • Nguyen, Tien;
    • El Kharraz, Sarah;
    • Handle, Florian;
    • Smeets, Elien;
    • Moris, Lisa;
    • Devlies, Wout;
    • Vandewinkel, Bram;
    • Thiry, Irina;
    • Ta, Duy Tien;
    • Gorkovskiy, Anton;
    • Voordeckers, Karin;
    • Henckaerts, Els;
    • Pinheiro, Vitor B.;
    • Claessens, Frank;
    • Verstrepen, Kevin J.;
    • Voet, Arnout;
    • Helsen, Christine
    Publication type:
    Article
  • N/C Interactions Are Dispensable for Normal In Vivo Functioning of the Androgen Receptor in Male Mice.

    Published in:
    Endocrinology, 2022, v. 163, n. 9, p. 1, doi. 10.1210/endocr/bqac104
    By:
    • Kharraz, Sarah El;
    • Dubois, Vanessa;
    • Launonen, Kaisa-Mari;
    • Helminen, Laura;
    • Palvimo, Jorma J;
    • Libert, Claude;
    • Smeets, Elien;
    • Moris, Lisa;
    • Eerlings, Roy;
    • Vanderschueren, Dirk;
    • Helsen, Christine;
    • Claessens, Frank
    Publication type:
    Article
  • A disease‐associated missense mutation in CYP4F3 affects the metabolism of leukotriene B4 via disruption of electron transfer.

    Published in:
    Journal of Cachexia, Sarcopenia & Muscle, 2022, v. 13, n. 4, p. 2242, doi. 10.1002/jcsm.13022
    By:
    • Smeets, Elien;
    • Huang, Shengyun;
    • Lee, Xiao Yin;
    • Van Nieuwenhove, Erika;
    • Helsen, Christine;
    • Handle, Florian;
    • Moris, Lisa;
    • El Kharraz, Sarah;
    • Eerlings, Roy;
    • Devlies, Wout;
    • Willemsen, Mathijs;
    • Bücken, Leoni;
    • Prezzemolo, Teresa;
    • Humblet‐Baron, Stephanie;
    • Voet, Arnout;
    • Rochtus, Anne;
    • Van Schepdael, Ann;
    • de Zegher, Francis;
    • Claessens, Frank
    Publication type:
    Article
  • Drivers of AR indifferent anti-androgen resistance in prostate cancer cells.

    Published in:
    Scientific Reports, 2019, v. 9, n. 1, p. N.PAG, doi. 10.1038/s41598-019-50220-1
    By:
    • Handle, Florian;
    • Prekovic, Stefan;
    • Helsen, Christine;
    • Van den Broeck, Thomas;
    • Smeets, Elien;
    • Moris, Lisa;
    • Eerlings, Roy;
    • Kharraz, Sarah El;
    • Urbanucci, Alfonso;
    • Mills, Ian G.;
    • Joniau, Steven;
    • Attard, Gerhardt;
    • Claessens, Frank
    Publication type:
    Article
  • The androgen receptor depends on ligand‐binding domain dimerization for transcriptional activation.

    Published in:
    EMBO Reports, 2021, v. 22, n. 12, p. 1, doi. 10.15252/embr.202152764
    By:
    • El Kharraz, Sarah;
    • Dubois, Vanessa;
    • van Royen, Martin E;
    • Houtsmuller, Adriaan B;
    • Pavlova, Ekatarina;
    • Atanassova, Nina;
    • Nguyen, Tien;
    • Voet, Arnout;
    • Eerlings, Roy;
    • Handle, Florian;
    • Prekovic, Stefan;
    • Smeets, Elien;
    • Moris, Lisa;
    • Devlies, Wout;
    • Ohlsson, Claes;
    • Poutanen, Matti;
    • Verstrepen, Kevin J;
    • Carmeliet, Geert;
    • Launonen, Kaisa‐Mari;
    • Helminen, Laura
    Publication type:
    Article