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Crystallographic studies of piperazine derivatives of 3‐methyl‐5‐spirofluorenehydantoin in search of structural features of P‐gp inhibitors.
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- Acta Crystallographica Section C: Structural Chemistry, 2021, v. 77, n. 8, p. 467, doi. 10.1107/S2053229621006756
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- Article
Influence of 3-{5-[4-(diethylamino)benzylidene]-rhodanine}propionic acid on the conformation of 5-(4-chlorobenzylidene)-2-(4-methylpiperazin-1-yl)-3H-imidazol-4(5H)-one.
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- Acta Crystallographica Section C: Structural Chemistry, 2018, v. 74, n. 11, p. 1, doi. 10.1107/S2053229618013980
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- Article
Conformational study of ( Z)-5-(4-chlorobenzylidene)-2-[4-(2-hydroxyethyl)piperazin-1-yl]-3 H-imidazol-4(5 H)-one in different environments: insight into the structural properties of bacterial efflux pump inhibitors.
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- Acta Crystallographica Section C: Structural Chemistry, 2017, v. 73, n. 12, p. 1151, doi. 10.1107/S2053229617016461
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- Article
Efflux Pump Blockers in Gram-Negative Bacteria: The New Generation of Hydantoin Based-Modulators to Improve Antibiotic Activity.
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- Frontiers in Microbiology, 2016, p. 1, doi. 10.3389/fmicb.2016.00622
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- Article
Pharmaceutical and Safety Profile Evaluation of Novel Selenocompounds with Noteworthy Anticancer Activity.
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- Pharmaceutics, 2022, v. 14, n. 2, p. 367, doi. 10.3390/pharmaceutics14020367
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- Article
Turning Waste into Value: Nanosized Natural Plant Materials of Solanum incanum L. and Pterocarpus erinaceus Poir with Promising Antimicrobial Activities.
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- Pharmaceutics, 2016, v. 8, n. 2, p. 11, doi. 10.3390/pharmaceutics8020011
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- Article
Histamine H 3 Receptor Ligands—KSK-59 and KSK-73—Reduce Body Weight Gain in a Rat Model of Excessive Eating.
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- Pharmaceuticals (14248247), 2021, v. 14, n. 11, p. 1080, doi. 10.3390/ph14111080
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- Article
Pharmacophoric features for a very potent 5‐spirofluorenehydantoin inhibitor of cancer efflux pump ABCB1, based on X‐ray analysis.
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- Chemical Biology & Drug Design, 2019, v. 93, n. 5, p. 844, doi. 10.1111/cbdd.13473
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- Article
In the search for a lead structure among series of potent and selective hydantoin 5- HT<sub>7</sub>R agents: The drug-likeness in vitro study.
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- Chemical Biology & Drug Design, 2017, v. 90, n. 6, p. 1295, doi. 10.1111/cbdd.13106
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- Article
Multitargeting the Action of 5-HT 6 Serotonin Receptor Ligands by Additional Modulation of Kinases in the Search for a New Therapy for Alzheimer's Disease: Can It Work from a Molecular Point of View?
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- International Journal of Molecular Sciences, 2022, v. 23, n. 15, p. 8768, doi. 10.3390/ijms23158768
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- Article
Structure Prediction, Evaluation, and Validation of GPR18 Lipid Receptor Using Free Programs.
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- International Journal of Molecular Sciences, 2022, v. 23, n. 14, p. 7917, doi. 10.3390/ijms23147917
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- Article
2-{5-[(Z ,2 Z)-2-Chloro-3-(4-nitrophenyl)-2-propenylidene]-4-oxo-2-thioxothiazolidin-3-yl}-3-methylbutanoic Acid as a Potential Anti-Breast Cancer Molecule.
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- International Journal of Molecular Sciences, 2022, v. 23, n. 8, p. 4091, doi. 10.3390/ijms23084091
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- Article
The Phenoxyalkyltriazine Antagonists for 5-HT 6 Receptor with Promising Procognitive and Pharmacokinetic Properties In Vivo in Search for a Novel Therapeutic Approach to Dementia Diseases.
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- International Journal of Molecular Sciences, 2021, v. 22, n. 19, p. 10773, doi. 10.3390/ijms221910773
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- Article
Novel N-Substituted 3-Aryl-4-(diethoxyphosphoryl)azetidin-2-ones as Antibiotic Enhancers and Antiviral Agents in Search for a Successful Treatment of Complex Infections.
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- International Journal of Molecular Sciences, 2021, v. 22, n. 15, p. 8032, doi. 10.3390/ijms22158032
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- Article
Molecular Insights into an Antibiotic Enhancer Action of New Morpholine-Containing 5-Arylideneimidazolones in the Fight against MDR Bacteria.
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- International Journal of Molecular Sciences, 2021, v. 22, n. 4, p. 2062, doi. 10.3390/ijms22042062
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- Article
Low Basicity as a Characteristic for Atypical Ligands of Serotonin Receptor 5-HT2.
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- International Journal of Molecular Sciences, 2021, v. 22, n. 3, p. 1035, doi. 10.3390/ijms22031035
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- Article
The 1,3,5-Triazine Derivatives as Innovative Chemical Family of 5-HT6 Serotonin Receptor Agents with Therapeutic Perspectives for Cognitive Impairment.
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- International Journal of Molecular Sciences, 2019, v. 20, n. 14, p. 3420, doi. 10.3390/ijms20143420
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- Article
Studies on Anticonvulsant Effects of Novel Histamine H3R Antagonists in Electrically and Chemically Induced Seizures in Rats.
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- International Journal of Molecular Sciences, 2018, v. 19, n. 11, p. 3386, doi. 10.3390/ijms19113386
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- Article
The Search for Histamine H<sub>4</sub> Receptor Ligands with Anticancer Activity among Novel (Thio)urea Derivatives.
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- ChemistrySelect, 2019, v. 4, n. 36, p. 10943, doi. 10.1002/slct.201902747
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- Article
Chalcogen-Varied Imidazolone Derivatives as Antibiotic Resistance Breakers in Staphylococcus aureus Strains.
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- Antibiotics (2079-6382), 2023, v. 12, n. 11, p. 1618, doi. 10.3390/antibiotics12111618
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- Article
To Cut the Mustard: Antimicrobial Activity of Selenocyanates on the Plate and in the Gas Phase.
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- Antibiotics (2079-6382), 2023, v. 12, n. 2, p. 290, doi. 10.3390/antibiotics12020290
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- Article
Funnel metadynamics and behavioral studies reveal complex effect of D2AAK1 ligand on anxiety-like processes.
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- Scientific Reports, 2022, v. 12, n. 1, p. 1, doi. 10.1038/s41598-022-25478-7
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- Article
Computer‐Aided Search for 5‐Arylideneimidazolone Anticancer Agents Able To Overcome ABCB1‐Based Multidrug Resistance.
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- ChemMedChem, 2021, v. 16, n. 15, p. 2386, doi. 10.1002/cmdc.202100252
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- Article
New 3-(Dibenzyloxyphosphoryl)isoxazolidine Conjugates of N1-Benzylated Quinazoline-2,4-diones as Potential Cytotoxic Agents against Cancer Cell Lines.
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- Molecules, 2024, v. 29, n. 13, p. 1, doi. 10.3390/molecules29133050
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- Article
Relationships between Molecular Characteristics of Novel Organic Selenium Compounds and the Formation of Sulfur Compounds in Selenium Biofortified Kale Sprouts.
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- Molecules, 2023, v. 28, n. 5, p. 2062, doi. 10.3390/molecules28052062
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- Article
New Triazine Derivatives as Serotonin 5-HT 6 Receptor Ligands.
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- Molecules, 2023, v. 28, n. 3, p. 1108, doi. 10.3390/molecules28031108
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- Article
Benzophenone Derivatives with Histamine H 3 Receptor Affinity and Cholinesterase Inhibitory Potency as Multitarget-Directed Ligands for Possible Therapy of Alzheimer's Disease.
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- Molecules, 2023, v. 28, n. 1, p. 238, doi. 10.3390/molecules28010238
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- Article
The Structural Determinants for α 1 -Adrenergic/Serotonin Receptors Activity among Phenylpiperazine-Hydantoin Derivatives.
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- Molecules, 2021, v. 26, n. 22, p. 7025, doi. 10.3390/molecules26227025
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- Article
Antioxidant or/and prooxidant activity of new phenyl-piperazine derivatives.
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- Cell Membranes & Free Radical Research, 2008, v. 1, n. 1, p. 43
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- Article
Strategies for bypassing the membrane barrier in multidrug resistant Gram-negative bacteria
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- FEBS Letters, 2011, v. 585, n. 11, p. 1682, doi. 10.1016/j.febslet.2011.04.054
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- Article
N -Skatyltryptamines—Dual 5-HT 6 R/D 2 R Ligands with Antipsychotic and Procognitive Potential.
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- Molecules, 2021, v. 26, n. 15, p. 4605, doi. 10.3390/molecules26154605
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- Article
Phenylpiperazine 5,5-Dimethylhydantoin Derivatives as First Synthetic Inhibitors of Msr(A) Efflux Pump in Staphylococcus epidermidis.
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- Molecules, 2020, v. 25, n. 17, p. 3788, doi. 10.3390/molecules25173788
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- Article
Search for ABCB1 Modulators Among 2-Amine-5-Arylideneimidazolones as a New Perspective to Overcome Cancer Multidrug Resistance.
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- Molecules, 2020, v. 25, n. 9, p. 2258, doi. 10.3390/molecules25092258
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- Article
Are the Hydantoin-1,3,5-triazine 5-HT6R Ligands a Hope to a Find New Procognitive and Anti-Obesity Drug? Considerations Based on Primary In Vivo Assays and ADME-Tox Profile In Vitro.
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- Molecules, 2019, v. 24, n. 24, p. 4472, doi. 10.3390/molecules24244472
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- Article
Selenocompounds as Novel Antibacterial Agents and Bacterial Efflux Pump Inhibitors.
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- Molecules, 2019, v. 24, n. 8, p. 1487, doi. 10.3390/molecules24081487
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- Article
5-Arylideneimidazolones with Amine at Position 3 as Potential Antibiotic Adjuvants against Multidrug Resistant Bacteria.
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- Molecules, 2019, v. 24, n. 3, p. 438, doi. 10.3390/molecules24030438
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- Article
Computer-Aided Studies for Novel Arylhydantoin 1,3,5-Triazine Derivatives as 5-HT6 Serotonin Receptor Ligands with Antidepressive-Like, Anxiolytic and Antiobesity Action In Vivo.
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- Molecules, 2018, v. 23, n. 10, p. 2529, doi. 10.3390/molecules23102529
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- Article
Selenides and Diselenides: A Review of Their Anticancer and Chemopreventive Activity.
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- Molecules, 2018, v. 23, n. 3, p. 628, doi. 10.3390/molecules23030628
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- Article
Selenazolinium Salts as "Small Molecule Catalysts" with High Potency against ESKAPE Bacterial Pathogens.
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- Molecules, 2017, v. 22, n. 12, p. 2174, doi. 10.3390/molecules22122174
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- Article
Aspects of a Distinct Cytotoxicity of Selenium Salts and Organic Selenides in Living Cells with Possible Implications for Drug Design.
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- Molecules, 2015, v. 20, n. 8, p. 13894, doi. 10.3390/molecules200813894
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- Article
Perry Disease: Current Outlook and Advances in Drug Discovery Approach to Symptomatic Treatment.
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- International Journal of Molecular Sciences, 2024, v. 25, n. 19, p. 10652, doi. 10.3390/ijms251910652
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- Article
Studies on Autophagy and Apoptosis of Fibrosarcoma HT-1080 Cells Mediated by Chalcone with Indole Moiety.
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- International Journal of Molecular Sciences, 2024, v. 25, n. 11, p. 6100, doi. 10.3390/ijms25116100
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- Article
The Subtype Selectivity in Search of Potent Hypotensive Agents among 5,5-Dimethylhydantoin Derived α 1 -Adrenoceptors Antagonists.
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- International Journal of Molecular Sciences, 2023, v. 24, n. 23, p. 16609, doi. 10.3390/ijms242316609
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- Article