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Discovery of Novel Amino Acids (Analogues)-Substituted Thiophene[3,2- d ]pyrimidine Derivatives as Potent HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors: Design, Synthesis, and Biological Evaluation.
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- International Journal of Molecular Sciences, 2024, v. 25, n. 16, p. 9028, doi. 10.3390/ijms25169028
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- Article
Design and synthesis of Fsp<sup>3</sup>‐enriched spirocyclic‐substituted diarylpyrimidine derivatives as novel HIV‐1 NNRTIs.
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- Chemical Biology & Drug Design, 2024, v. 103, n. 3, p. 1, doi. 10.1111/cbdd.14510
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- Article
Design, synthesis, and biological evaluation of piperidinyl‐substituted [1,2,4]triazolo[1,5‐a]pyrimidine derivatives as potential anti‐HIV‐1 agents with reduced cytotoxicity.
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- Chemical Biology & Drug Design, 2021, v. 97, n. 1, p. 67, doi. 10.1111/cbdd.13760
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Design, synthesis, and biologic evaluation of novel galloyl derivatives as HIV‐1 RNase H inhibitors.
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- Chemical Biology & Drug Design, 2019, v. 93, n. 4, p. 582, doi. 10.1111/cbdd.13455
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- Article
Discovery of potent HIV‐1 non‐nucleoside reverse transcriptase inhibitors by exploring the structure–activity relationship of solvent‐exposed regions I.
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- Chemical Biology & Drug Design, 2019, v. 93, n. 4, p. 430, doi. 10.1111/cbdd.13429
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- Article
Design, synthesis, and antiviral evaluation of novel hydrazone‐substituted thiophene[3,2‐d]pyrimidine derivatives as potent human immunodeficiency virus‐1 inhibitors.
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- Chemical Biology & Drug Design, 2018, v. 92, n. 6, p. 2009, doi. 10.1111/cbdd.13373
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- Article
Design, synthesis, and biological evaluation of novel 5-Alkyl-6-Adamantylmethylpyrimidin-4(3H)-ones as HIV-1 non-nucleoside reverse-transcriptase inhibitors.
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- Chemical Biology & Drug Design, 2016, v. 88, n. 3, p. 380, doi. 10.1111/cbdd.12765
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- Article
Arylazolyl(azinyl)thioacetanilides: Part 19.
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- Chemical Biology & Drug Design, 2016, v. 88, n. 2, p. 241, doi. 10.1111/cbdd.12751
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- Article
Design, Synthesis, and Biological Evaluation of Novel 2-(Pyridin-3-yloxy)acetamide Derivatives as Potential Anti- HIV-1 Agents.
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- Chemical Biology & Drug Design, 2016, v. 87, n. 2, p. 283, doi. 10.1111/cbdd.12657
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- Article
Synthesis and Preliminary Antiviral Activities of Piperidine-substituted Purines against HIV and Influenza A/H1N1 Infections.
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- Chemical Biology & Drug Design, 2015, v. 86, n. 4, p. 568, doi. 10.1111/cbdd.12520
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- Article
Synthesis and Biological Evaluation of a Series of 2-((1-substituted-1 H-1,2,3-triazol-4-yl)methylthio)-6-(naphthalen-1-ylmethyl)pyrimidin-4(3 H)-one As Potential HIV-1 Inhibitors.
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- Chemical Biology & Drug Design, 2015, v. 86, n. 4, p. 614, doi. 10.1111/cbdd.12524
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- Article
Design, Synthesis, and Biological Evaluation of Novel Benzoyl Diarylamine/ether Derivatives as Potential Anti-HIV-1 Agents.
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- Chemical Biology & Drug Design, 2015, v. 86, n. 3, p. 333, doi. 10.1111/cbdd.12497
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- Article
Design, Synthesis, and Biological Evaluation of Novel 4-Aminopiperidinyl-linked 3,5-Disubstituted-1,2,6-thiadiazine-1,1-dione Derivatives as HIV-1 NNRTIs.
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- Chemical Biology & Drug Design, 2015, v. 86, n. 1, p. 887, doi. 10.1111/cbdd.12468
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Design, Synthesis, and Anti- HIV Evaluation of Novel Triazine Derivatives Targeting the Entrance Channel of the NNRTI Binding Pocket.
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- Chemical Biology & Drug Design, 2015, v. 86, n. 1, p. 902, doi. 10.1111/cbdd.12471
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- Article
Synthesis and Anti- HIV Activity of 4-(Naphthalen-1-yl)-1,2,5-thiadiazol-3-hydroxyl Derivatives.
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- Chemical Biology & Drug Design, 2014, v. 84, n. 4, p. 420, doi. 10.1111/cbdd.12328
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Discovery of HIV-1 Integrase Inhibitors: Pharmacophore Mapping, Virtual Screening, Molecular Docking, Synthesis, and Biological Evaluation.
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- Chemical Biology & Drug Design, 2014, v. 83, n. 2, p. 154, doi. 10.1111/cbdd.12207
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- Article
Design, Synthesis, and Biological Evaluation of Novel 3,5-Disubstituted-1,2,6-Thiadiazine-1,1-Dione Derivatives as HIV-1 NNRTIs.
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- Chemical Biology & Drug Design, 2013, v. 82, n. 4, p. 384, doi. 10.1111/cbdd.12160
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Molecular design opportunities presented by solvent‐exposed regions of target proteins.
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- Medicinal Research Reviews, 2019, v. 39, n. 6, p. 2194, doi. 10.1002/med.21581
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Discovery and Mechanistic Investigation of Piperazinone Phenylalanine Derivatives with Terminal Indole or Benzene Ring as Novel HIV-1 Capsid Modulators.
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- Molecules, 2022, v. 27, n. 23, p. 8415, doi. 10.3390/molecules27238415
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Design, Synthesis, and Mechanistic Study of 2-Pyridone-Bearing Phenylalanine Derivatives as Novel HIV Capsid Modulators.
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- Molecules, 2022, v. 27, n. 21, p. 7640, doi. 10.3390/molecules27217640
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Identification of Boronate-Containing Diarylpyrimidine Derivatives as Novel HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors.
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- Molecules, 2022, v. 27, n. 21, p. 7538, doi. 10.3390/molecules27217538
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- Article
Design, Synthesis and Structure—Activity Relationships of Phenylalanine-Containing Peptidomimetics as Novel HIV-1 Capsid Binders Based on Ugi Four-Component Reaction.
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- Molecules, 2022, v. 27, n. 18, p. 5995, doi. 10.3390/molecules27185995
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- Article
Scaffold Hopping in Discovery of HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors: From CH(CN)-DABOs to CH(CN)-DAPYs.
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- Molecules, 2020, v. 25, n. 7, p. 1581, doi. 10.3390/molecules25071581
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- Article
1,2,4-Triazolo[1,5-a]pyrimidines as a Novel Class of Inhibitors of the HIV-1 Reverse Transcriptase-Associated Ribonuclease H Activity.
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- Molecules, 2020, v. 25, n. 5, p. 1183, doi. 10.3390/molecules25051183
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- Article
Design of Biphenyl-Substituted Diarylpyrimidines with a Cyanomethyl Linker as HIV-1 NNRTIs via a Molecular Hybridization Strategy.
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- Molecules, 2020, v. 25, n. 5, p. 1050, doi. 10.3390/molecules25051050
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- Article
Application of the Triazolization Reaction to Afford Dihydroartemisinin Derivatives with Anti-HIV Activity.
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- Molecules, 2017, v. 22, n. 2, p. 303, doi. 10.3390/molecules22020303
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- Article
Discovery of piperidine-substituted thiazolo[5,4-d]pyrimidine derivatives as potent and orally bioavailable HIV-1 non-nucleoside reverse transcriptase inhibitors.
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- Communications Chemistry, 2019, v. 2, n. 1, p. N.PAG, doi. 10.1038/s42004-019-0174-8
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In vitro anti-HIV activity of diverse substituted nitrosopyrimidine analogues.
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- Chemistry & Biology Interface, 2016, v. 6, n. 2, p. 69
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Exploration of the in vitro anti-HIV and cyclin-dependent kinase 2 (CDK2) inhibitory activities of new 6-aryl-pyrimidines and their nitroso analogues.
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- Chemistry & Biology Interface, 2016, v. 6, n. 1, p. 1
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- Article
In vitro anti-HIV and HCV activity of new thioureido and thiazole analogues of cholesterol conjugated α-amino acid residues and in silico molecular modeling study.
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- Chemistry & Biology Interface, 2015, v. 5, n. 6, p. 333
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- Article
Synthesis and biological evaluation of some new 1,3,4-thiadiazole and 1,2,4-triazole derivatives from L-methionine as antituberculosis and antiviral agents.
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- Marmara Pharmaceutical Journal, 2015, v. 19, n. 2, p. 88, doi. 10.12991/mpj.2015199639
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Synthesis and evaluation of antiviral, antitubercular and anticancer activities of some novel thioureas derived from 4-aminobenzohydrazide hydrazones.
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- Marmara Pharmaceutical Journal, 2010, v. 14, n. 1, p. 13
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Covalently Targeted Highly Conserved Tyr318 to Improve the Drug Resistance Profiles of HIV-1 NNRTIs: A Proof-of-Concept Study.
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- International Journal of Molecular Sciences, 2023, v. 24, n. 2, p. 1215, doi. 10.3390/ijms24021215
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- Article
Different Heterocycles Functionalized s-Triazine Analogues: Design, Synthesis and In Vitro Antimicrobial, Antituberculosis, and Anti-HIV Assessment.
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- Journal of Heterocyclic Chemistry, 2014, v. 51, n. 6, p. 1641, doi. 10.1002/jhet.1769
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Pyridazines 92. Synthesis of dialkyldipyridazinodiazepinones as potential HIV-1 reverse transcriptase inhibitors.
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- Journal of Heterocyclic Chemistry, 2001, v. 38, n. 1, p. 125, doi. 10.1002/jhet.5570380117
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- Article
Some Hydrazones of 2-Aroylamino-3-methylbutanohydrazide: Synthesis, Molecular Modeling Studies, and Identification as Stereoselective Inhibitors of HIV-1.
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- Archiv der Pharmazie, 2013, v. 346, n. 2, p. 140, doi. 10.1002/ardp.201200311
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- Article
Synthesis and Evaluation of Novel 4-Substituted Styryl Quinazolines as Potential Antimicrobial Agents.
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- Archiv der Pharmazie, 2012, v. 345, n. 12, p. 964, doi. 10.1002/ardp.201200291
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- Article
Non-nucleoside HIV Reverse Transcriptase Inhibitors, Part 6[1]: Synthesis and Anti-HIV Activity of Novel 2-[(Arylcarbonylmethyl)thio]-6-arylthio DABO Analogues.
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- Archiv der Pharmazie, 2005, v. 338, n. 10, p. 457, doi. 10.1002/ardp.200400961
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- Article
Anti-HIV Activity of Thiosemicarbazone and Semicarbazone Derivatives of (±)-3-Menthone.
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- Archiv der Pharmazie, 2002, v. 335, n. 5, p. 183, doi. 10.1002/1521-4184(200205)335:5<183::AID-ARDP183>3.0.CO;2-U
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- Article
Synthesis of 3-Nitrosoimidazo[1,2- a]pyridine Derivatives as Potential Antiretroviral Agents.
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- Archiv der Pharmazie, 2001, v. 334, n. 7, p. 224, doi. 10.1002/1521-4184(200107)334:7<224::AID-ARDP224>3.0.CO;2-7
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- Article
Inhibition of Human Immunodeficiency Virus Type (HIV-1) Replication by some Diversely Functionalized Spirocyclopropyl Derivatives.
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- Archiv der Pharmazie, 1999, v. 332, n. 5, p. 163, doi. 10.1002/(SICI)1521-4184(19995)332:5<163::AID-ARDP163>3.0.CO;2-2
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- Article
Pridine Oxide Derivatives: Structure-Activity Relationship for Inhibition of Human Immunodeficiency Virus and Cytomegalovirus Replication in Cell Culture.
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- Helvetica Chimica Acta, 2002, v. 85, n. 9, p. 2961, doi. 10.1002/1522-2675(200209)85:9<2961::AID-HLCA2961>3.0.CO;2-R
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- Article
1,2,4-Triazole Derivatives Inhibiting the Human Immunodeficiency Virus Type 1 (HIV-1) in vitro.
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- Helvetica Chimica Acta, 2002, v. 85, n. 7, p. 1883, doi. 10.1002/1522-2675(200207)85:7<1883::AID-HLCA1883>3.0.CO;2-R
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- Article
A phenyl-thiadiazolylidene-amine derivative ejects zinc from retroviral nucleocapsid zinc fingers and inactivates HIV virions.
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- Retrovirology, 2012, v. 9, n. 1, p. 95, doi. 10.1186/1742-4690-9-95
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- Article
Derivatives of 3′‐Azidothymidine with 6‐Cyanopyridone as Base or as Phosphoramidate Ester and their Antiretroviral Activity.
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- Helvetica Chimica Acta, 2023, v. 106, n. 1, p. 1, doi. 10.1002/hlca.202200157
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- Article
Synthesis, characterization and biological evaluation of 1,3-thiazolidine-4-ones derived from (2S)-2-benzoylamino-3-methylbutanohydrazide hydrazones.
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- Journal of Research in Pharmacy, 2021, v. 25, n. 4, p. 507, doi. 10.29228/jrp.41
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Synthesis, and prediction of molecular properties and antimicrobial activity of some acylhydrazones derived from N-(arylsulfonyl)methionine.
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- Turkish Journal of Chemistry, 2016, v. 40, n. 3, p. 510, doi. 10.3906/kim-1509-21
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- Article
Chelation Motifs Affecting Metal-dependent Viral Enzymes: N'-acylhydrazone Ligands as Dual Target Inhibitors of HIV-1 Integrase and Reverse Transcriptase Ribonuclease H Domain.
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- Frontiers in Microbiology, 2017, v. 8, p. 1, doi. 10.3389/fmicb.2017.00440
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- Article
Synthesis and anti-HIV activity of novel 2,4-disubstituted-7-methyl-1,1,3-trioxo-2H,4H-pyrazolo[4,5-e][1,2,4]thiadiazine derivatives.
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- Drug Discoveries & Therapeutics, 2011, v. 5, n. 6, p. 279, doi. 10.5582/ddt.2011.v5.6.279
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- Article
Cell-dependent interference of a series of new 6-aminoquinolone derivatives with viral (HIV/CMV) transactivation.
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- Journal of Antimicrobial Chemotherapy (JAC), 2005, v. 56, n. 5, p. 847, doi. 10.1093/jac/dki328
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- Article