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Multipotente Liganden mit kombinierter Cholinesterase- und Monoaminooxidase-Inhibition sowie Histamin-H3R-Antagonismus bei neurodegenerativen Erkrankungen.
Published in:
Angewandte Chemie, 2017, v. 129, n. 41, p. 12939, doi. 10.1002/ange.201706072
By:
- Bautista ‐ Aguilera, Óscar M.;
- Hagenow, Stefanie;
- Palomino ‐ Antolin, Alejandra;
- Farré ‐ Alins, Víctor;
- Ismaili, Lhassane;
- Joffrin, Pierre ‐ Louis;
- Jimeno, María L.;
- Soukup, Ondřej;
- Janočková, Jana;
- Kalinowsky, Lena;
- Proschak, Ewgenij;
- Iriepa, Isabel;
- Moraleda, Ignacio;
- Schwed, Johannes S.;
- Romero Martínez, Alejandro;
- López ‐ Muñoz, Francisco;
- Chioua, Mourad;
- Egea, Javier;
- Ramsay, Rona R.;
- Marco ‐ Contelles, José
Publication type:
Article
Multitarget-Directed Ligands Combining Cholinesterase and Monoamine Oxidase Inhibition with Histamine H3R Antagonism for Neurodegenerative Diseases.
Published in:
Angewandte Chemie International Edition, 2017, v. 56, n. 41, p. 12765, doi. 10.1002/anie.201706072
By:
- Bautista‐Aguilera, Óscar M.;
- Hagenow, Stefanie;
- Palomino‐Antolin, Alejandra;
- Farré‐Alins, Víctor;
- Ismaili, Lhassane;
- Joffrin, Pierre‐Louis;
- Jimeno, María L.;
- Soukup, Ondřej;
- Janočková, Jana;
- Kalinowsky, Lena;
- Proschak, Ewgenij;
- Iriepa, Isabel;
- Moraleda, Ignacio;
- Schwed, Johannes S.;
- Romero Martínez, Alejandro;
- López‐Muñoz, Francisco;
- Chioua, Mourad;
- Egea, Javier;
- Ramsay, Rona R.;
- Marco‐Contelles, José
Publication type:
Article
Acetylcholinesterase Inhibition of Diversely Functionalized Quinolinones for Alzheimer's Disease Therapy.
Published in:
International Journal of Molecular Sciences, 2020, v. 21, n. 11, p. 3913, doi. 10.3390/ijms21113913
By:
- Bautista-Aguilera, Óscar M.;
- Ismaili, Lhassane;
- Chioua, Mourad;
- Andrys, Rudolf;
- Schmidt, Monika;
- Bzonek, Petr;
- Martínez-Grau, María Ángeles;
- Beadle, Christopher D.;
- Vetman, Tatiana;
- López-Muñoz, Francisco;
- Iriepa, Isabel;
- Refouvelet, Bernard;
- Musilek, Kamil;
- Marco-Contelles, José
Publication type:
Article
Automated Synthesis of New Quinoxalinetacrines.
Published in:
ChemistrySelect, 2020, v. 5, n. 21, p. 6491, doi. 10.1002/slct.202001593
By:
- Bautista‐Aguilera, Óscar M.;
- Ismaili, Lhassane;
- Chioua, Mourad;
- Iriepa, Isabel;
- Ángeles Martinez‐Grau, Marìa;
- Beadle, Christopher D.;
- Vetman, Tatiana;
- López‐Muñoz, Francisco;
- Marco‐Contelles, José
Publication type:
Article
N -Hydroxy- N -Propargylamide Derivatives of Ferulic Acid: Inhibitors of Cholinesterases and Monoamine Oxidases.
Published in:
Molecules, 2022, v. 27, n. 21, p. 7437, doi. 10.3390/molecules27217437
By:
- Bautista-Aguilera, Óscar M.;
- Alonso, José M.;
- Catto, Marco;
- Iriepa, Isabel;
- Knez, Damijan;
- Gobec, Stanislav;
- Marco-Contelles, José
Publication type:
Article
Predicting targets of compounds against neurological diseases using cheminformatic methodology.
Published in:
Journal of Computer-Aided Molecular Design, 2015, v. 29, n. 2, p. 183, doi. 10.1007/s10822-014-9816-1
By:
- Nikolic, Katarina;
- Mavridis, Lazaros;
- Bautista-Aguilera, Oscar;
- Marco-Contelles, José;
- Stark, Holger;
- Carmo Carreiras, Maria;
- Rossi, Ilaria;
- Massarelli, Paola;
- Agbaba, Danica;
- Ramsay, Rona;
- Mitchell, John
Publication type:
Article
Multipotent cholinesterase/monoamine oxidase inhibitors for the treatment of Alzheimer's disease: design, synthesis, biochemical evaluation, ADMET, molecular modeling, and QSAR analysis of novel donepezil-pyridyl hybrids.
Published in:
Drug Design, Development & Therapy, 2014, v. 8, p. 1893, doi. 10.2147/DDDT.S69258
By:
- Bautista-Aguilera, Oscar M.;
- Esteban, Gerard;
- Chioua, Mourad;
- Nikolic, Katarina;
- Agbaba, Danica;
- Moraleda, Ignacio;
- Iriepa, Isabel;
- Soriano, Elena;
- Samadi, Abdelouahid;
- Unzeta, Mercedes;
- Marco-Contelles, José
Publication type:
Article
Synthesis of N -Substituted Pyrroles Catalyzed by Low-Cost and Commercially Available Aluminas.
Published in:
Catalysts (2073-4344), 2023, v. 13, n. 3, p. 603, doi. 10.3390/catal13030603
By:
- Portilla-Zúñiga, Omar;
- Bautista-Aguilera, Óscar M.;
- Martínez, José J.;
- Rojas, Hugo;
- Macías, Mario A.;
- Iriepa, Isabel;
- Pérez-Redondo, Adrián;
- Sathicq, Ángel;
- Castillo, Juan-Carlos;
- Romanelli, Gustavo P.
Publication type:
Article
Tacrines as Therapeutic Agents for Alzheimer's Disease. V. Recent Developments.
Published in:
Chemical Record, 2021, v. 21, n. 1, p. 162, doi. 10.1002/tcr.202000107
By:
- Bautista‐Aguilera, Óscar M.;
- Ismaili, Lhassane;
- Iriepa, Isabel;
- Diez‐Iriepa, Daniel;
- Chabchoub, Fakher;
- Marco‐Contelles, José;
- Pérez, Marta
Publication type:
Article
Triazolopyridopyrimidine: A New Scaffold for Dual-Target Small Molecules for Alzheimer's Disease Therapy.
Published in:
Molecules, 2020, v. 25, n. 14, p. 3190, doi. 10.3390/molecules25143190
By:
- Zribi, Lazhar;
- Pachòn-Angona, Irene;
- Bautista-Aguilera, Òscar M.;
- Diez-Iriepa, Daniel;
- Marco-Contelles, José;
- Ismaili, Lhassane;
- Iriepa, Isabel;
- Chabchoub, Fakher;
- Branco, Paula Sério
Publication type:
Article
Synthesis and Biological Evaluation of Benzochromenopyrimidinones as Cholinesterase Inhibitors and Potent Antioxidant, Non-Hepatotoxic Agents for Alzheimer’s Disease.
Published in:
Molecules, 2016, v. 21, n. 5, p. 634, doi. 10.3390/molecules21050634
By:
- Dgachi, Youssef;
- Bautista-Aguilera, Oscar M.;
- Benchekroun, Mohamed;
- Martin, Hélène;
- Bonet, Alexandre;
- Knez, Damijan;
- Godyń, Justyna;
- Malawska, Barbara;
- Gobec, Stanislav;
- Chioua, Mourad;
- Janockova, Jana;
- Soukup, Ondrej;
- Chabchoub, Fakher;
- Marco-Contelles, José;
- Ismaili, Lhassane
Publication type:
Article
Synthesis and Biological Assessment of Racemic Benzochromenopyrimidinimines as Antioxidant, Cholinesterase, and Aβ1−42 Aggregation Inhibitors for Alzheimer's Disease Therapy.
Published in:
ChemMedChem, 2016, v. 11, n. 12, p. 1318, doi. 10.1002/cmdc.201500539
By:
- Dgachi, Youssef;
- Ismaili, Lhassane;
- Knez, Damijan;
- Benchekroun, Mohamed;
- Martin, Hélène;
- Szałaj, Natalia;
- Wehle, Sarah;
- Bautista‐Aguilera, Oscar M.;
- Luzet, Vincent;
- Bonnet, Alexandre;
- Malawska, Barbara;
- Gobec, Stanislav;
- Chioua, Mourad;
- Decker, Michael;
- Chabchoub, Fakher;
- Marco‐Contelles, José
Publication type:
Article

Found: 12

Multipotente Liganden mit kombinierter Cholinesterase- und Monoaminooxidase-Inhibition sowie Histamin-H<sub>3</sub>R-Antagonismus bei neurodegenerativen Erkrankungen.

Multitarget-Directed Ligands Combining Cholinesterase and Monoamine Oxidase Inhibition with Histamine H<sub>3</sub>R Antagonism for Neurodegenerative Diseases.

Acetylcholinesterase Inhibition of Diversely Functionalized Quinolinones for Alzheimer's Disease Therapy.

Automated Synthesis of New Quinoxalinetacrines.

N -Hydroxy- N -Propargylamide Derivatives of Ferulic Acid: Inhibitors of Cholinesterases and Monoamine Oxidases.

Predicting targets of compounds against neurological diseases using cheminformatic methodology.

Multipotent cholinesterase/monoamine oxidase inhibitors for the treatment of Alzheimer's disease: design, synthesis, biochemical evaluation, ADMET, molecular modeling, and QSAR analysis of novel donepezil-pyridyl hybrids.

Synthesis of N -Substituted Pyrroles Catalyzed by Low-Cost and Commercially Available Aluminas.

Tacrines as Therapeutic Agents for Alzheimer's Disease. V. Recent Developments.

Triazolopyridopyrimidine: A New Scaffold for Dual-Target Small Molecules for Alzheimer's Disease Therapy.

Synthesis and Biological Evaluation of Benzochromenopyrimidinones as Cholinesterase Inhibitors and Potent Antioxidant, Non-Hepatotoxic Agents for Alzheimer’s Disease.

Synthesis and Biological Assessment of Racemic Benzochromenopyrimidinimines as Antioxidant, Cholinesterase, and Aβ<sub>1−42</sub> Aggregation Inhibitors for Alzheimer's Disease Therapy.