Works matching AU Spasov, Alexander


Results: 44
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    Guanidine Derivatives of Quinazoline-2,4(1 H ,3 H)-Dione as NHE-1 Inhibitors and Anti-Inflammatory Agents.

    Published in:
    Life (2075-1729), 2022, v. 12, n. 10, p. 1647, doi. 10.3390/life12101647
    By:
    • Spasov, Alexander;
    • Ozerov, Alexander;
    • Kosolapov, Vadim;
    • Gurova, Natalia;
    • Kucheryavenko, Aida;
    • Naumenko, Ludmila;
    • Babkov, Denis;
    • Sirotenko, Viktor;
    • Taran, Alena;
    • Borisov, Alexander;
    • Sokolova, Elena;
    • Klochkov, Vladlen;
    • Merezhkina, Darya;
    • Miroshnikov, Mikhail;
    • Ovsyankina, Nadezhda;
    • Smirnov, Alexey;
    • Velikorodnaya, Yulia
    Publication type:
    Article
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    Synthesis and multifaceted pharmacological activity of novel quinazoline NHE-1 inhibitors.

    Published in:
    Scientific Reports, 2021, v. 11, n. 1, p. 1, doi. 10.1038/s41598-021-03722-w
    By:
    • Spasov, Alexander;
    • Ozerov, Alexander;
    • Vassiliev, Pavel;
    • Kosolapov, Vadim;
    • Gurova, Natalia;
    • Kucheryavenko, Aida;
    • Naumenko, Ludmila;
    • Babkov, Denis;
    • Sirotenko, Viktor;
    • Taran, Alena;
    • Litvinov, Roman;
    • Borisov, Alexander;
    • Klochkov, Vladlen;
    • Merezhkina, Darya;
    • Miroshnikov, Mikhail;
    • Uskov, Georgy;
    • Ovsyankina, Nadezhda
    Publication type:
    Article
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    6-Nitroazolo[1,5- a]pyrimidin-7(4 H)-ones as Antidiabetic Agents.

    Published in:
    Archiv der Pharmazie, 2017, v. 350, n. 12, p. n/a, doi. 10.1002/ardp.201700226
    By:
    • Spasov, Alexander A.;
    • Babkov, Denis A.;
    • Sysoeva, Valentina A.;
    • Litvinov, Roman A.;
    • Shamshina, Darya D.;
    • Ulomsky, Evgeny N.;
    • Savateev, Konstantin V.;
    • Fedotov, Viktor V.;
    • Slepukhin, Pavel A.;
    • Chupakhin, Oleg N.;
    • Charushin, Valery N.;
    • Rusinov, Vladimir L.
    Publication type:
    Article
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    3-Arylidene-2-oxindoles as Potent NRH:Quinone Oxidoreductase 2 Inhibitors.

    Published in:
    Molecules, 2023, v. 28, n. 3, p. 1174, doi. 10.3390/molecules28031174
    By:
    • Lozinskaya, Natalia A.;
    • Bezsonova, Elena N.;
    • Dubar, Meriam;
    • Melekhina, Daria D.;
    • Bazanov, Daniil R.;
    • Bunev, Alexander S.;
    • Grigor'eva, Olga B.;
    • Klochkov, Vladlen G.;
    • Sokolova, Elena V.;
    • Babkov, Denis A.;
    • Spasov, Alexander A.;
    • Sosonyuk, Sergey E.
    Publication type:
    Article
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    CK2 Inhibition and Antitumor Activity of 4,7-Dihydro-6-nitroazolo[1,5-a]pyrimidines.

    Published in:
    Molecules, 2022, v. 27, n. 16, p. 5239, doi. 10.3390/molecules27165239
    By:
    • Lyapustin, Daniil N.;
    • Kotovskaya, Svetlana K.;
    • Butorin, Ilya I.;
    • Ulomsky, Evgeny N.;
    • Rusinov, Vladimir L.;
    • Babkov, Denis A.;
    • Pokhlebin, Alexander A.;
    • Spasov, Alexander A.;
    • Melekhin, Vsevolod V.;
    • Tokhtueva, Maria D.;
    • Shcheglova, Anna V.;
    • Makeev, Oleg G.
    Publication type:
    Article
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    Synthesis and Pharmacological Evaluation of Novel 2,3,4,5-tetrahydro[1,3]diazepino[1,2- a ]benzimidazole Derivatives as Promising Anxiolytic and Analgesic Agents.

    Published in:
    Molecules, 2021, v. 26, n. 19, p. 6049, doi. 10.3390/molecules26196049
    By:
    • Maltsev, Dmitriy V.;
    • Spasov, Alexander A.;
    • Vassiliev, Pavel M.;
    • Skripka, Maria O.;
    • Miroshnikov, Mikhail V.;
    • Kochetkov, Andrey N.;
    • Eliseeva, Nataliya V.;
    • Lifanova, Yuliya V.;
    • Kuzmenko, Tatyana A.;
    • Divaeva, Lyudmila N.;
    • Morkovnik, Anatolii S.
    Publication type:
    Article
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    Hypoglycemic potential of cyclic guanidine derivatives.

    Published in:
    Pure & Applied Chemistry, 2017, v. 89, n. 8, p. 1007, doi. 10.1515/pac-2016-1024
    By:
    • Spasov, Alexander A.;
    • Vassiliev, Pavel M.;
    • Lenskaya, Karina V.;
    • Anisimova, Vera A.;
    • Kuzmenko, Tatyana A.;
    • Morkovnik, Anatolii S.;
    • Kosolapov, Vadim A.;
    • Babkov, Denis A.
    Publication type:
    Article
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    Novel Substituted Azoloazines with Anticoagulant Activity.

    Published in:
    International Journal of Molecular Sciences, 2023, v. 24, n. 21, p. 15581, doi. 10.3390/ijms242115581
    By:
    • Spasov, Alexander A.;
    • Fedorova, Olga V.;
    • Rasputin, Nikolay A.;
    • Ovchinnikova, Irina G.;
    • Ishmetova, Rashida I.;
    • Ignatenko, Nina K.;
    • Gorbunov, Evgeny B.;
    • Sadykhov, Gusein A. o.;
    • Kucheryavenko, Aida F.;
    • Gaidukova, Kseniia A.;
    • Sirotenko, Victor S.;
    • Rusinov, Gennady L.;
    • Verbitskiy, Egor V.;
    • Charushin, Valery N.
    Publication type:
    Article
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    Design, Synthesis and Pharmacological Evaluation of Novel C 2 ,C 3 -Quinoxaline Derivatives as Promising Anxiolytic Agents.

    Published in:
    International Journal of Molecular Sciences, 2022, v. 23, n. 22, p. 14401, doi. 10.3390/ijms232214401
    By:
    • Maltsev, Dmitriy V.;
    • Skripka, Maria O.;
    • Spasov, Alexander A.;
    • Vassiliev, Pavel M.;
    • Perfiliev, Maxim A.;
    • Divaeva, Lyudmila N.;
    • Zubenko, Alexander A.;
    • Morkovnik, Anatolii S.;
    • Klimenko, Alexander I.;
    • Miroshnikov, Mikhail V.;
    • Klochkov, Vladlen G.;
    • Ianalieva, Laura R.
    Publication type:
    Article
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    Anti-Inflammatory Activity of Soluble Epoxide Hydrolase Inhibitors Based on Selenoureas Bearing an Adamantane Moiety.

    Published in:
    International Journal of Molecular Sciences, 2022, v. 23, n. 18, p. N.PAG, doi. 10.3390/ijms231810710
    By:
    • Burmistrov, Vladimir;
    • Morisseau, Christophe;
    • Babkov, Denis A.;
    • Golubeva, Tatiana;
    • Pitushkin, Dmitry;
    • Sokolova, Elena V.;
    • Vasipov, Vladimir;
    • Kuznetsov, Yaroslav;
    • Bazhenov, Sergey V.;
    • Novoyatlova, Uliana S.;
    • Bondarev, Nikolay A.;
    • Manukhov, Ilya V.;
    • Osipova, Victoria;
    • Berberova, Nadezhda;
    • Spasov, Alexander A.;
    • Butov, Gennady M.;
    • Hammock, Bruce D.
    Publication type:
    Article
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    Combined In Silico, Ex Vivo, and In Vivo Assessment of L-17, a Thiadiazine Derivative with Putative Neuro- and Cardioprotective and Antidepressant Effects.

    Published in:
    International Journal of Molecular Sciences, 2021, v. 22, n. 24, p. 13626, doi. 10.3390/ijms222413626
    By:
    • Sarapultsev, Alexey;
    • Vassiliev, Pavel;
    • Grinchii, Daniil;
    • Kiss, Alexander;
    • Mach, Mojmir;
    • Osacka, Jana;
    • Balloova, Alexandra;
    • Paliokha, Ruslan;
    • Kochetkov, Andrey;
    • Sidorova, Larisa;
    • Sarapultsev, Petr;
    • Chupakhin, Oleg;
    • Rantsev, Maxim;
    • Spasov, Alexander;
    • Dremencov, Eliyahu
    Publication type:
    Article
    40

    Ru(III) Complexes with Lonidamine-Modified Ligands.

    Published in:
    International Journal of Molecular Sciences, 2021, v. 22, n. 24, p. 13468, doi. 10.3390/ijms222413468
    By:
    • Shutkov, Ilya A.;
    • Okulova, Yulia N.;
    • Tyurin, Vladimir Yu.;
    • Sokolova, Elena V.;
    • Babkov, Denis A.;
    • Spasov, Alexander A.;
    • Gracheva, Yulia A.;
    • Schmidt, Claudia;
    • Kirsanov, Kirill I.;
    • Shtil, Alexander A.;
    • Redkozubova, Olga M.;
    • Shevtsova, Elena F.;
    • Milaeva, Elena R.;
    • Ott, Ingo;
    • Nazarov, Alexey A.
    Publication type:
    Article
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