Works matching AU Musa, Arafa


Results: 42
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    New Sulfamethoxazole Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors: Design, Synthesis, Cytotoxic Activity and Molecular Modeling.

    Published in:
    Pharmaceuticals (14248247), 2022, v. 15, n. 9, p. N.PAG, doi. 10.3390/ph15091134
    By:
    • Abdelgawad, Mohamed A.;
    • Bukhari, Syed N. A.;
    • Musa, Arafa;
    • Elmowafy, Mohammed;
    • Elkomy, Mohammed H.;
    • Nayl, AbdElAziz. A.;
    • El-Ghorab, Ahmed H.;
    • Alsohaimi, Ibrahim Hotan;
    • Abdel-Bakky, Mohamed Sadek;
    • Althobaiti, Ibrahim O.;
    • Altaleb, Hamud A.;
    • Omar, Hany A.;
    • Abdelazeem, Ahmed H.;
    • Zaki, Mohamed A.;
    • Shaker, Mohamed E.;
    • Elshemy, Heba A. H.
    Publication type:
    Article
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    Strawberry and Ginger Silver Nanoparticles as Potential Inhibitors for SARS-CoV-2 Assisted by In Silico Modeling and Metabolic Profiling.

    Published in:
    Antibiotics (2079-6382), 2021, v. 10, n. 7, p. 824, doi. 10.3390/antibiotics10070824
    By:
    • Al-Sanea, Mohammad M.;
    • Abelyan, Narek;
    • Abdelgawad, Mohamed A.;
    • Musa, Arafa;
    • Ghoneim, Mohammed M.;
    • Al-Warhi, Tarfah;
    • Aljaeed, Nada;
    • Alotaibi, Ohoud J.;
    • Alnusaire, Taghreed S.;
    • Abdelwahab, Sayed F.;
    • Helmy, Aya;
    • Abdelmohsen, Usama Ramadan;
    • Youssif, Khayrya A.
    Publication type:
    Article
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    Novel Phenolic Compounds as Potential Dual EGFR and COX-2 Inhibitors: Design, Semisynthesis, in vitro Biological Evaluation and in silico Insights.

    Published in:
    Drug Design, Development & Therapy, 2021, v. 15, p. 2325, doi. 10.2147/DDDT.S310820
    By:
    • Abdelgawad, Mohamed A;
    • Musa, Arafa;
    • Almalki, Atiah H;
    • Alzarea, Sami I;
    • Mostafa, Ehab M;
    • Hegazy, Mostafa M;
    • Mostafa-Hedeab, Gomaa;
    • Ghoneim, Mohammed M;
    • Parambi, Della GT;
    • Bakr, Rania B;
    • Al-Muaikel, Nayef S;
    • Alanazi, Abdullah S;
    • Alharbi, Metab;
    • Ahmad, Waqas;
    • Bukhari, Syed NA;
    • Al-Sanea, Mohammad M
    Publication type:
    Article
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    Design, synthesis, and biological investigation of new thiazole-based derivatives as multi-targeted inhibitors endowed with antiproliferative, antioxidant, and antibacterial properties.

    Published in:
    Frontiers in Chemistry, 2025, p. 1, doi. 10.3389/fchem.2025.1595997
    By:
    • Gomaa, Hesham A. M.;
    • Atta, Asmaa M.;
    • Shaker, Mohamed E.;
    • Alzarea, Sami I.;
    • Alsahli, Tariq G.;
    • Alatwi, Eid;
    • Musa, Arafa;
    • Mohamed, Fatma A. M.;
    • Alzahrani, Hayat Ali;
    • Mohassab, Aliaa M.;
    • Abdelmoez, Alshaimaa;
    • Bräse, Stefan;
    • Youssif, Bahaa G. M.
    Publication type:
    Article
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    Optimization of pyrazolo[1,5-a]pyrimidine based compounds with pyridine scaffold: Synthesis, biological evaluation and molecular modeling study.

    Published in:
    Arabian Journal of Chemistry, 2022, v. 15, n. 8, p. N.PAG, doi. 10.1016/j.arabjc.2022.104015
    By:
    • Abdelgawad, Mohamed A.;
    • Elkanzi, Nadia A.A.;
    • Musa, Arafa;
    • Ghoneim, Mohammed M.;
    • Ahmad, Waqas;
    • Elmowafy, Mohammed;
    • Abdelhaleem Ali, Ahmed M.;
    • Abdelazeem, Ahmed H.;
    • Bukhari, Syed N.A.;
    • El-Sherbiny, Mohamed;
    • Abourehab, Mohammed A.S.;
    • Bakr, Rania B.
    Publication type:
    Article
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    Curcumin: a bioactive compound with molecular targets for human malignancies.

    Published in:
    Food & Agricultural Immunology, 2023, v. 34, n. 1, p. 1, doi. 10.1080/09540105.2023.2280524
    By:
    • Shahbaz, Muhammad;
    • Imran, Muhammad;
    • Hussain, Muzzamal;
    • Alsagaby, Suliman A.;
    • Momal, Ushna;
    • Naeem, Hammad;
    • Abdelgawad, Mohamed A.;
    • El-Ghorab, Ahmed H.;
    • Al Abdulmonem, Waleed;
    • Waqar, Ahmed Bilal;
    • Ghoneim, Mohammed M.;
    • Musa, Arafa;
    • Al Jbawi, Entessar
    Publication type:
    Article
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    LC/MS Profiling and Gold Nanoparticle Formulation of Major Metabolites from Origanum majorana as Antibacterial and Antioxidant Potentialities.

    Published in:
    Plants (2223-7747), 2022, v. 11, n. 14, p. N.PAG, doi. 10.3390/plants11141871
    By:
    • El-Ghorab, Ahmed H.;
    • Behery, Fathy A.;
    • Abdelgawad, Mohamed A.;
    • Alsohaimi, Ibrahim Hotan;
    • Musa, Arafa;
    • Mostafa, Ehab M.;
    • Altaleb, Hamud A.;
    • Althobaiti, Ibrahim O.;
    • Hamza, Mohamed;
    • Elkomy, Mohammed H.;
    • Hamed, Ahmed A.;
    • Sayed, Ahmed M.;
    • Hassan, Hossam M.;
    • Aboseada, Mahmoud A.
    Publication type:
    Article
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    An In Vitro and In Silico Study of the Enhanced Antiproliferative and Pro-Oxidant Potential of Olea europaea L. cv. Arbosana Leaf Extract via Elastic Nanovesicles (Spanlastics).

    Published in:
    Antioxidants, 2021, v. 10, n. 12, p. 1860, doi. 10.3390/antiox10121860
    By:
    • Alnusaire, Taghreed S.;
    • Sayed, Ahmed M.;
    • Elmaidomy, Abeer H.;
    • Al-Sanea, Mohammad M.;
    • Albogami, Sarah;
    • Albqmi, Mha;
    • Alowaiesh, Bassam F.;
    • Mostafa, Ehab M.;
    • Musa, Arafa;
    • Youssif, Khayrya A.;
    • Refaat, Hesham;
    • Othman, Eman M.;
    • Dandekar, Thomas;
    • Alaaeldin, Eman;
    • Ghoneim, Mohammed M.;
    • Abdelmohsen, Usama Ramadan
    Publication type:
    Article
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    Antiulcer Potential of Olea europea L. cv. Arbequina Leaf Extract Supported by Metabolic Profiling and Molecular Docking.

    Published in:
    Antioxidants, 2021, v. 10, n. 5, p. 644, doi. 10.3390/antiox10050644
    By:
    • Musa, Arafa;
    • Shady, Nourhan Hisham;
    • Ahmed, Shaimaa R.;
    • Alnusaire, Taghreed S.;
    • Sayed, Ahmed M.;
    • Alowaiesh, Bassam F.;
    • Sabouni, Ibrahim;
    • Al-Sanea, Mohammad M.;
    • Mostafa, Ehab M.;
    • Youssif, Khayrya A.;
    • Abu-Baih, Dalia H.;
    • Elrehany, Mahmoud A.;
    • Abdelmohsen, Usama Ramadan;
    • Fernández-Bolaños, Juan;
    • Bermudez-Oria, Alejandra
    Publication type:
    Article
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    Design and construction of novel pyridine-pyrimidine hybrids as selective COX-2 suppressors: anti-inflammatory potential, ulcerogenic profile, molecular modeling and ADME/Tox studies.

    Published in:
    Journal of Biomolecular Structure & Dynamics, 2025, v. 43, n. 4, p. 1804, doi. 10.1080/07391102.2023.2293257
    By:
    • Shaker, Mohamed E.;
    • Goma, Hesham A. M.;
    • Alsalahat, Izzeddin;
    • Elkanzi, Nadia A. A.;
    • Azouz, Amany A.;
    • Abdel-Bakky, Mohamed Sadek;
    • Ghoneim, Mohammed M.;
    • Hazem, Sara H.;
    • El-Mesery, Mohamed E.;
    • Farouk, Amr;
    • Alzarea, Sami I.;
    • Alsahli, Tariq G.;
    • Alotaibi, Nasser Hadal;
    • Musa, Arafa;
    • Abdelgawad, Mohamed A.;
    • Bakr, Rania B.
    Publication type:
    Article
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    Introducing of novel class of pyrano[2,3-c]pyrazole-5-carbonitrile analogs with potent antimicrobial activity, DNA gyrase inhibition, and prominent pharmacokinetic and CNS toxicity profiles supported by molecular dynamic simulation.

    Published in:
    Journal of Biomolecular Structure & Dynamics, 2024, v. 42, n. 18, p. 9529, doi. 10.1080/07391102.2023.2252088
    By:
    • Almaghrabi, Mohammed;
    • Musa, Arafa;
    • Aljohani, Ahmed K. B.;
    • Ahmed, Hany E. A.;
    • Alsulaimany, Marwa;
    • Miski, Samar F.;
    • Mostafa, Ehab M.;
    • Hussein, Shaimaa;
    • Parambi, Della Grace Thomas;
    • Ghoneim, Mohammed M.;
    • Elgammal, Walid E.;
    • Halawa, Ahmed H.;
    • Hammad, Ali;
    • El-Agrody, Ahmed M.
    Publication type:
    Article
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    The anticancer and EGFR-TK/CDK-9 dual inhibitory potentials of new synthetic pyranopyrazole and pyrazolone derivatives: X-ray crystallography, in vitro, and in silico mechanistic investigations.

    Published in:
    Journal of Biomolecular Structure & Dynamics, 2023, v. 41, n. 21, p. 12411, doi. 10.1080/07391102.2023.2167000
    By:
    • Musa, Arafa;
    • Ihmaid, Saleh K.;
    • Hughes, David L.;
    • Said, Musa A.;
    • Abulkhair, Hamada S.;
    • El-Ghorab, Ahmed H.;
    • Abdelgawad, Mohamed A.;
    • Shalaby, Khaled;
    • Shaker, Mohamed E.;
    • Alharbi, Khalid Saad;
    • Alotaibi, Nasser Hadal;
    • Kays, Deborah L.;
    • Taylor, Laurence J.;
    • Parambi, Della Grace Thomas;
    • Alzarea, Sami I.;
    • Al-Karmalawy, Ahmed A.;
    • Ahmed, Hany E. A.;
    • El-Agrody, Ahmed M.
    Publication type:
    Article
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