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Differential maturation and chaperone dependence of the paralogous protein kinases DYRK1A and DYRK1B.
- Published in:
- Scientific Reports, 2022, v. 12, n. 1, p. 1, doi. 10.1038/s41598-022-06423-0
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- Article
Identification of Novel Chemical Scaffolds Inhibiting Trypanothione Synthetase from Pathogenic Trypanosomatids.
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- PLoS Neglected Tropical Diseases, 2016, v. 10, n. 4, p. 1, doi. 10.1371/journal.pntd.0004617
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- Article
The indole motif is essential for the antitrypanosomal activity of N<sup>5</sup>-substituted paullones.
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- PLoS ONE, 2023, v. 18, n. 11, p. 1, doi. 10.1371/journal.pone.0292946
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- Article
Discovery of Antitrypanosomal Indolylacetamides by a Deconstruction–Optimization Strategy Applied to Paullones.
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- ChemMedChem, 2023, v. 18, n. 10, p. 1, doi. 10.1002/cmdc.202300036
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- Article
(E)-5-(Methoxyimino)-1,3,4,5-tetrahydro-2 H -benzo[ b ]azepin-2-one.
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- Molbank, 2021, v. 2021, n. 4, p. M1293, doi. 10.3390/M1293
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- Publication type:
- Article
1-(Imidazo[1,2-a]pyridin-1-ium-1-yl)-2,3,4-trioxocyclobutan-1-ide.
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- Molbank, 2019, v. 2019, n. 3, p. M1072, doi. 10.3390/M1072
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- Publication type:
- Article
2,3,4-Trioxo-1-(1H-pyrrolo[2,3-b]pyridin-7-ium-7yl)-cyclobutan-1-ide.
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- Molbank, 2018, v. 2018, n. 4, p. M1026, doi. 10.3390/M1026
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- Article
(E)-2-(1-Cyano-2-methoxy-2-oxoethylidene)-3,4-dioxo-1-(pyridin-1-ium-1-yl)cyclobutan-1-ide.
- Published in:
- Molbank, 2017, v. 2017, n. 3, p. m953, doi. 10.3390/M953
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- Article
7-Bromo-1-methyl-2-phenyl-1H-indole-3-carbonitrile.
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- Molbank, 2017, v. 2017, n. 2, p. m941, doi. 10.3390/M941
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- Article
3-Chlorokenpaullone.
- Published in:
- Molbank, 2015, v. 2015, n. 2, p. 1, doi. 10.3390/M856
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- Article
7-Iodo-1H-indole-3-carbonitrile.
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- Molbank, 2015, v. 2015, n. 4, p. 1, doi. 10.3390/M869
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- Publication type:
- Article
4,5,6,7-Tetrachloro-2-(1H-imidazol-2-yl)isoindoline-1,3-dione.
- Published in:
- Molbank, 2012, v. 12, n. 4, p. 1, doi. 10.3390/M785
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- Article
2-tert-Butyl-5,6,7,8,9,10-hexahydrocyclohepta[b]indole.
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- Molbank, 2011, v. 11, n. 3, p. 1, doi. 10.3390/M737
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- Article
Synthesis of pyrido[3,4- d] benzazepines.
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- Journal of Heterocyclic Chemistry, 1995, v. 32, n. 3, p. 803, doi. 10.1002/jhet.5570320319
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- Article
Metallkomplexe als Proteinkinase-Hemmstoffe.
- Published in:
- Angewandte Chemie, 2010, v. 122, n. 31, p. 5354, doi. 10.1002/ange.201002062
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- Article
Hierarchical phosphorylation of apical membrane antigen 1 is required for efficient red blood cell invasion by malaria parasites.
- Published in:
- Scientific Reports, 2016, p. 34479, doi. 10.1038/srep34479
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- Publication type:
- Article
Synthesis and Properties of a Selective Inhibitor of Homeodomain–Interacting Protein Kinase 2 (HIPK2).
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- PLoS ONE, 2014, v. 9, n. 2, p. 1, doi. 10.1371/journal.pone.0089176
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- Article
Synthesis of Paullones with Aminoalkyl Side Chains.
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- Archiv der Pharmazie, 2002, v. 335, n. 7, p. 311, doi. 10.1002/1521-4184(200209)335:7<311::AID-ARDP311>3.0.CO;2-F
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- Article
Aryl Rings Are Part of the Darpone Pharmacophore.
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- Archiv der Pharmazie, 2001, v. 334, n. 5, p. 163, doi. 10.1002/1521-4184(200105)334:5<163::AID-ARDP163>3.0.CO;2-3
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- Publication type:
- Article
Synthese von 7,12-Dihydro-indolo[3,2- d][1]benzazepin-6-( 5H)-onen und 6,11-Dihydro-thieno-[3′,2′:2,3]azepino[4,5- b]indol-5(4 H)- on.
- Published in:
- Archiv der Pharmazie, 1992, v. 325, n. 5, p. 297, doi. 10.1002/ardp.19923250509
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- Article
Synthese [ b]-kondensierter azepindione durch dealkoxycarbonylierung.
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- Archiv der Pharmazie, 1991, v. 324, n. 9, p. 579, doi. 10.1002/ardp.2503240910
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- Publication type:
- Article
Additionsreaktionen von β-Ketosulfoxiden und Bis(phenylsulfinyl)methan an Isocyanate.
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- Archiv der Pharmazie, 1985, v. 318, n. 12, p. 1086, doi. 10.1002/ardp.19853181206
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- Publication type:
- Article
2-Sulfinyl-pentan-1,5-dione aus β-Oxosulfoxiden 2-Sulfinyl-pentane-1,5-diones from β-Oxosulfoxides.
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- Archiv der Pharmazie, 1985, v. 318, n. 11, p. 1045, doi. 10.1002/ardp.19853181116
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- Article
Identification of CLK1 Inhibitors by a Fragment-linking Based Virtual Screening.
- Published in:
- Molecular Informatics, 2017, v. 36, n. 4, p. n/a, doi. 10.1002/minf.201600123
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- Article
Identification of Inhibitors of the Tyrosine Kinase c-Met by Structure-Based Virtual Screening.
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- Molecular Informatics, 2011, v. 30, n. 2/3, p. 145, doi. 10.1002/minf.201000138
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- Article
Book Review: Microwaves in Organic and Medicinal Chemistry. Edited by R. Mannhold, H. Kubinyi, G. Folkers.
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- Archiv der Pharmazie, 2006, v. 339, n. 4, p. 217, doi. 10.1002/ardp.200600006
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- Article
Alsterpaullone, a novel cyclin-dependent kinase inhibitor, induces apoptosis by activation of caspase-9 due to perturbation in mitochondrial membrane potential (This article is a US Government work and, as such, is in the public domain in the United States of America.)
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- Molecular Carcinogenesis, 2003, v. 36, n. 4, p. 183, doi. 10.1002/mc.10114
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- Article
Antiplasmodial dihetarylthioethers target the coenzyme A synthesis pathway in Plasmodium falciparum erythrocytic stages.
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- Malaria Journal, 2017, v. 16, p. 1, doi. 10.1186/s12936-017-1839-3
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- Article
Garbage in, garbage out: how reliable training data improved a virtual screening approach against SARS-CoV-2 MPro.
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- Frontiers in Pharmacology, 2023, p. 1, doi. 10.3389/fphar.2023.1193282
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- Article
Synthesis and Antiplasmodial Activity of Bisindolylcyclobutenediones.
- Published in:
- Molecules, 2021, v. 26, n. 16, p. 4739, doi. 10.3390/molecules26164739
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- Article
7-(2-Anilinopyrimidin-4-yl)-1-benzazepin-2-ones Designed by a "Cut and Glue" Strategy Are Dual Aurora A/VEGF-R Kinase Inhibitors.
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- Molecules, 2021, v. 26, n. 6, p. 1611, doi. 10.3390/molecules26061611
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- Article
4-Arylthieno[2,3-b]pyridine-2-carboxamides Are a New Class of Antiplasmodial Agents.
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- Molecules, 2020, v. 25, n. 14, p. 3187, doi. 10.3390/molecules25143187
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- Article
[b]-Annulated Halogen-Substituted Indoles as Potential DYRK1A Inhibitors.
- Published in:
- Molecules, 2019, v. 24, n. 22, p. 4090, doi. 10.3390/molecules24224090
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- Article
Indole-3-Carbonitriles as DYRK1A Inhibitors by Fragment-Based Drug Design.
- Published in:
- Molecules, 2018, v. 23, n. 2, p. 64, doi. 10.3390/molecules23020064
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- Article
Novel 2-Phenoxyanilide Congeners Derived from a Hit Structure of the TCAMS: Synthesis and Evaluation of Their in Vitro Activity against Plasmodium falciparum.
- Published in:
- Molecules, 2016, v. 21, n. 2, p. 223, doi. 10.3390/molecules21020223
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- Article
Structure-Aided Optimization of Kinase Inhibitors Derived from Alsterpaullone.
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- ChemBioChem, 2005, v. 6, n. 3, p. 541, doi. 10.1002/cbic.200400099
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- Article
Molecular structures of cdc2-like kinases in complex with a new inhibitor chemotype.
- Published in:
- PLoS ONE, 2018, v. 13, n. 5, p. 1, doi. 10.1371/journal.pone.0196761
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- Article
Metal Complexes as Protein Kinase Inhibitors.
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- Angewandte Chemie International Edition, 2010, v. 49, n. 31, p. 5226, doi. 10.1002/anie.201002062
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- Publication type:
- Article
Structure–activity relationships in a series of antiplasmodial thieno[2,3-b]pyridines.
- Published in:
- Malaria Journal, 2019, v. 18, n. 1, p. N.PAG, doi. 10.1186/s12936-019-2725-y
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- Publication type:
- Article