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- Title
Synthesis of Indolines and Derivatives by Aza‐Heck Cyclization.
- Authors
Xu, Feiyang; Korch, Katerina M.; Watson, Donald A.
- Abstract
For the first time, an aza‐Heck cyclization that allows the preparation of indoline scaffolds is described. Using N‐hydroxy anilines as electrophiles, which can be easily accessed from the corresponding nitroarenes, this method provides indolines bearing pendant functionality and complex ring topologies. Synthesis of challenging indolines, such as those bearing fully substituted carbon atoms at C2, is also possible using this method.
- Subjects
NITROAROMATIC compounds; ANILINE; INDOLINE; ATOMS; AZA compounds
- Publication
Angewandte Chemie, 2019, Vol 131, Issue 38, p13582
- ISSN
0044-8249
- Publication type
Article
- DOI
10.1002/ange.201907758