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Titelbild: Squalenyl Hydrogen Sulfate Nanoparticles for Simultaneous Delivery of Tobramycin and an Alkylquinolone Quorum Sensing Inhibitor Enable the Eradication of P. aeruginosa Biofilm Infections (Angew. Chem. 26/2020).
- Published in:
- Angewandte Chemie, 2020, v. 132, n. 26, p. 10285, doi. 10.1002/ange.202005838
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- Article
Squalenyl Hydrogen Sulfate Nanoparticles for Simultaneous Delivery of Tobramycin and an Alkylquinolone Quorum Sensing Inhibitor Enable the Eradication of P. aeruginosa Biofilm Infections.
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- Angewandte Chemie, 2020, v. 132, n. 26, p. 10378, doi. 10.1002/ange.202001407
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- Article
Metallfreie meta-selektive Oxyarylierung von Alkinen mit Pyridin- N-oxiden: schnelle Synthese von Metyrapon-Analoga.
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- Angewandte Chemie, 2016, v. 128, n. 49, p. 15650, doi. 10.1002/ange.201607988
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- Article
Platinum(II) complexes interfering with testicular steroid biosynthesis: drugs for the therapy of advanced or recurrent prostate cancers? Preclinical studies.
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- Journal of Cancer Research & Clinical Oncology, 2007, v. 133, n. 3, p. 153, doi. 10.1007/s00432-006-0151-3
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- Article
In-depth Profiling of MvfR-Regulated Small Molecules in Pseudomonas aeruginosa after Quorum Sensing Inhibitor Treatment.
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- Frontiers in Microbiology, 2017, v. 8, p. 1, doi. 10.3389/fmicb.2017.00924
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- Article
Synthesis, Optimization, Antifungal Activity, Selectivity, and CYP51 Binding of New 2-Aryl-3-azolyl-1-indolyl-propan-2-ols.
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- Pharmaceuticals (14248247), 2020, v. 13, n. 8, p. 186, doi. 10.3390/ph13080186
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- Article
Metal-Free meta-Selective Alkyne Oxyarylation with Pyridine N-Oxides: Rapid Assembly of Metyrapone Analogues.
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- Angewandte Chemie International Edition, 2016, v. 55, n. 49, p. 15424, doi. 10.1002/anie.201607988
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- Article
Overcoming the Unexpected Functional Inversion of a PqsR Antagonist in Pseudomonas aeruginosa: An In Vivo Potent Antivirulence Agent Targeting pqs Quorum Sensing.
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- Angewandte Chemie International Edition, 2014, v. 53, n. 4, p. 1109, doi. 10.1002/anie.201307547
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Rule–based regulatory and metabolic model for Quorum sensing in P. aeruginosa.
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- BMC Systems Biology, 2013, v. 7, n. 1, p. 1, doi. 10.1186/1752-0509-7-81
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- Article
Finding New Molecular Targets of Familiar Natural Products Using In Silico Target Prediction.
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- International Journal of Molecular Sciences, 2020, v. 21, n. 19, p. 7102, doi. 10.3390/ijms21197102
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- Article
Recent Progress in Pharmaceutical Therapies for Castration-Resistant Prostate Cancer.
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- International Journal of Molecular Sciences, 2013, v. 14, n. 7, p. 13958, doi. 10.3390/ijms140713958
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- Article
Bacterial RNAP Inhibitors: Synthesis and Evaluation of Prodrugs of Aryl‐ureidothiophene‐carboxylic acids.
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- ChemistrySelect, 2017, v. 2, n. 35, p. 11899, doi. 10.1002/slct.201702574
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- Article
Structure‐Activity Relationship and Mode‐Of‐Action Studies Highlight 1‐(4‐Biphenylylmethyl)‐1H‐imidazole‐Derived Small Molecules as Potent CYP121 Inhibitors.
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- ChemMedChem, 2021, v. 16, n. 18, p. 2786, doi. 10.1002/cmdc.202100283
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- Article
Front Cover: Phosphonate as a Stable Zinc‐Binding Group for "Pathoblocker" Inhibitors of Clostridial Collagenase H (ColH) (ChemMedChem 8/2021).
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- ChemMedChem, 2021, v. 16, n. 8, p. 1198, doi. 10.1002/cmdc.202100229
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- Article
Phosphonate as a Stable Zinc‐Binding Group for "Pathoblocker" Inhibitors of Clostridial Collagenase H (ColH).
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- ChemMedChem, 2021, v. 16, n. 8, p. 1257, doi. 10.1002/cmdc.202000994
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- Article
Overcoming the Unexpected Functional Inversion of a PqsR Antagonist in Pseudomonas aeruginosa: An In Vivo Potent Antivirulence Agent Targeting pqs Quorum Sensing.
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- Angewandte Chemie, 2014, v. 126, n. 4, p. 1127, doi. 10.1002/ange.201307547
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- Article
17β-Hydroxysteroid Dehydrogenase Type 2 Inhibition: Discovery of Selective and Metabolically Stable Compounds Inhibiting Both the Human Enzyme and Its Murine Ortholog.
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- PLoS ONE, 2015, v. 10, n. 7, p. 1, doi. 10.1371/journal.pone.0134754
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- Article
Design and Synthesis of a Library of Lead-Like 2,4-Bisheterocyclic Substituted Thiophenes as Selective Dyrk/Clk Inhibitors.
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- PLoS ONE, 2014, v. 9, n. 3, p. 1, doi. 10.1371/journal.pone.0087851
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- Article
3-Pyridyl Substituted Aliphatic Cycles as CYP11B2 Inhibitors: Aromaticity Abolishment of the Core Significantly Increased Selectivity over CYP1A2.
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- PLoS ONE, 2012, v. 7, n. 11, p. 1, doi. 10.1371/journal.pone.0048048
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- Article
Insights in 17β-HSD1 Enzyme Kinetics and Ligand Binding by Dynamic Motion Investigation.
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- PLoS ONE, 2010, v. 5, n. 8, p. 1, doi. 10.1371/journal.pone.0012026
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- Article
Quantitative analysis of 5α-reductase inhibitors in DU145 cells using matrix-assisted laser desorption/ ionization time-of-flight mass spectrometry and high-performance liquid chromatography/tandem mass spectrometry.
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- Journal of Mass Spectrometry, 2004, v. 39, n. 7, p. 762, doi. 10.1002/jms.647
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- Article
C16 and C17 Substituted Derivatives of Pregnenolone and Progesterone as Inhibitors of 17α-Hydroxylase-C17, 20-lyase: Synthesis and Biological Evaluation.
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- Archiv der Pharmazie, 2002, v. 335, n. 11/12, p. 526, doi. 10.1002/ardp.200290006
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- Article
Inhibition of CYP 17, a New Strategy for the Treatment of Prostate Cancer.
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- Archiv der Pharmazie, 2002, v. 335, n. 4, p. 119, doi. 10.1002/1521-4184(200204)335:4<119::AID-ARDP119>3.0.CO;2-#
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- Article
Synthesis and Biological Evaluation of 4-(4-(Alkyl-and Phenylaminocarbonyl)benzoyl)benzoic Acid Derivatives as Non-steroidal Inhibitors of Steroid 5α-Reductase Isozymes 1 and 2.
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- Archiv der Pharmazie, 2002, v. 335, n. 2/3, p. 83, doi. 10.1002/1521-4184(200203)335:2/3<83::AID-ARDP83>3.0.CO;2-3
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- Article
Novel steroidal pyrimidyl inhibitors of P450 17 (17α-hydroxylase/C17-20-lyase).
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- Archiv der Pharmazie, 2001, v. 334, n. 12, p. 373, doi. 10.1002/1521-4184(200112)334:12<373::AID-ARDP373>3.0.CO;2-X
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- Article
1-(2,6-Dichloro-4-hydroxyphenyl)-2-phenylethanes - New Biological Response Modifiers for the Therapy of Breast Cancer. Synthesis and Evaluation of Estrogenic/Antiestrogenic Properties.
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- Archiv der Pharmazie, 2001, v. 334, n. 4, p. 125, doi. 10.1002/1521-4184(200104)334:4<125::AID-ARDP125>3.0.CO;2-D
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- Article
Synthesis and Evaluation of Steroidal Hydroxamic Acids as Inhibitors of P450 17 (17α-Hydroxylase/C17-20-Lyase).
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- Archiv der Pharmazie, 2001, v. 334, n. 4, p. 138, doi. 10.1002/1521-4184(200104)334:4<138::AID-ARDP138>3.0.CO;2-Y
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- Article
5α-Reductase in Intact DU145 Cells: Evidence for Isozyme I and Evaluation of Novel Inhibitors.
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- Archiv der Pharmazie, 2000, v. 333, n. 7, p. 201, doi. 10.1002/1521-4184(20007)333:7<201::AID-ARDP201>3.0.CO;2-D
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New Nonsteroidal Steroid 5α-Reductase Inhibitors. Syntheses and Structure-Activity Studies on Carboxamide Phenylalkyl-Substituted Pyridones and Piperidones.
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- Archiv der Pharmazie, 2000, v. 333, n. 5, p. 145, doi. 10.1002/(SICI)1521-4184(20005)333:5<145::AID-ARDP145>3.0.CO;2-Q
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- Article
Synthesis of 2-[2-(1-Imidazolyl)ethyl]-4-phenylcycloalka[ g]phthalazin-1(2 H)-ones as Thromboxane A<sub>2</sub> Synthase Inhibitors.
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- Archiv der Pharmazie, 1999, v. 332, n. 11, p. 408, doi. 10.1002/(SICI)1521-4184(199911)332:11<408::AID-ARDP408>3.0.CO;2-P
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- Article
1-Imidazolylcarbonyloxy-substituted Tetrahydroquinolines and Pyridines: Synthesis and Evaluation of P450 TxA2 Inhibition.
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- Archiv der Pharmazie, 1999, v. 332, n. 10, p. 358, doi. 10.1002/(SICI)1521-4184(199910)332:10<358::AID-ARDP358>3.0.CO;2-D
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- Article
Synthesis and Evaluation of Azole-substituted 2-Aryl-6-methoxy-3,4-dihydronaphthalenes and -naphthalenes as Inhibitors of 17α-Hydroxylase-C17,20-Lyase (P450 17.
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- Archiv der Pharmazie, 1999, v. 332, n. 1, p. 25, doi. 10.1002/(SICI)1521-4184(19991)332:1<25::AID-ARDP25>3.0.CO;2-7
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- Article
Spectrofluorimetric Quantification of Malondialdehyde for Evaluation of Cyclooxygenase-1/Thromboxane Synthase Inhibition.
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- Archiv der Pharmazie, 1998, v. 331, n. 11, p. 359, doi. 10.1002/(SICI)1521-4184(199811)331:11<359::AID-ARDP359>3.0.CO;2-B
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- Publication type:
- Article
Synthesis of Novel Oximes of 2-Aryl-6-methoxy-3,4-dihydronaphthalene and Their Evaluation as Inhibitors of 17α-Hydroxylase-C17,20-Lyase (P450 17).
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- Archiv der Pharmazie, 1998, v. 331, n. 1, p. 36, doi. 10.1002/(SICI)1521-4184(199801)331:1<36::AID-ARDP36>3.0.CO;2-0
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- Publication type:
- Article
Novel Highly Active Thromboxane A<sub>2</sub> Synthase Inhibitors Devoid of Carboxylic Groups.
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- Archiv der Pharmazie, 1997, v. 330, n. 1/2, p. 1, doi. 10.1002/ardp.19973300102
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- Article
Synthesis and In Vitro Evaluation of 3-(1-Azolylmethyl)-1 H-indoles and 3-(1-Azolyl-1-phenylmethyl)-1 H-indoles as Inhibitors of P450 arom.
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- Archiv der Pharmazie, 1997, v. 330, n. 5, p. 141, doi. 10.1002/ardp.19973300506
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- Article
Synthesis of Z- and E-1-Methyl-2-(1-hydroximinoethyl)-6-methoxy-3,4-dihydronaphthalene and Evaluation as Inhibitors of 17α-Hydroxylase-C17,20-Lyase (P450 17).
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- Archiv der Pharmazie, 1997, v. 330, n. 11, p. 359, doi. 10.1002/ardp.19973301108
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- Article
Synthesis and Evaluation of Azole-Substituted Tetrahydronaphthalenes as Inhibitors of P450 arom, P450 17, and P450 TxA<sub>2</sub>.
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- Archiv der Pharmazie, 1996, v. 329, n. 5, p. 251, doi. 10.1002/ardp.19963290506
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- Article
Editorial.
- Published in:
- Archiv der Pharmazie, 1996, v. 329, n. 1, p. 1, doi. 10.1002/ardp.19963290102
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- Article
4,5-Dihydro-3-(2-pyrazinyl)naphtho[1,2- c]pyrazole: A Potent and Selective Inhibitor of Steroid-17α-Hydroxylase-C17,20-Lyase (P450 17).
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- Archiv der Pharmazie, 1995, v. 328, n. 7/8, p. 573, doi. 10.1002/ardp.19953280703
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- Article
Synthesis and Biochemical Evaluation of (Carbamoylalkenyl)phenyloxy Carboxylic Acid Derivatives as Non-steroidal 5α-Reductase Inhibitors.
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- Archiv der Pharmazie, 1995, v. 328, n. 3, p. 239, doi. 10.1002/ardp.19953280307
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- Article
Synthesis and Evaluation of Sulfur-Containing Glutethimide Derivatives for Aromatase and Desmolase Inhibitory Activity.
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- Archiv der Pharmazie, 1993, v. 326, n. 7, p. 391, doi. 10.1002/ardp.19933260704
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- Article
Neue Hemmstoffe der Aromatase: Synthese und biologische Aktivität pyridyl-substituierter Phenanthrenonderivate.
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- Archiv der Pharmazie, 1991, v. 324, n. 11, p. 833, doi. 10.1002/ardp.2503241102
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- Article
Pyridyl-Substituierte Tetralonderivate: Eine Neue Klasse Nichtsteroidaler Aromatase-Inhibitoren.
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- Archiv der Pharmazie, 1991, v. 324, n. 10, p. 815, doi. 10.1002/ardp.2503241008
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- Publication type:
- Article
Potentielle Antiöstrogene vom Typ des 1,2-Diphenyl-1-pyridyl-but-1-ens. Teil 2: Biologische Prüfung.
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- Archiv der Pharmazie, 1991, v. 324, n. 4, p. 231, doi. 10.1002/ardp.19913240408
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- Article
Potentielle Antiöstrogene vom Typ des 1,2-Diphenyl-1-pyridyl-but-1-ens Teil 1: Synthese.
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- Archiv der Pharmazie, 1991, v. 324, n. 4, p. 223, doi. 10.1002/ardp.19913240407
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- Article
Antiestrogene N-(4-Hydroxyphenyl)-N-(1,1,1-trifluor-2-propyl)-4-hydroxybenzamide: Beeinflussung der Wirkung durch hydrophobe Reste in ortho-Position des Benzamidfragments.
- Published in:
- Archiv der Pharmazie, 1990, v. 323, n. 2, p. 73, doi. 10.1002/ardp.19903230204
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- Publication type:
- Article
Cytotoxic Ester Derivatives of the Mammary Tumor Inhibiting Antiestrogen 2,3-Bis(2-fluoro-4-hydroxyphenyl)-2,3-dimethylbutane.
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- Archiv der Pharmazie, 1990, v. 323, n. 2, p. 121, doi. 10.1002/ardp.19903230213
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- Publication type:
- Article
N-(4-Hydroxyphenyl)-N-(1,1,1-trifluor-2-propyl)-4-hydroxybenzamid: Synthese und pharmakologische Bewertung eines neues Antiestrogens.
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- Archiv der Pharmazie, 1988, v. 321, n. 8, p. 497, doi. 10.1002/ardp.19883210814
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- Article
Hemmstoffe der Aromatase. Synthese und pharmakologische Bewertung von potentiellen mammatumorhemmenden 4-Alkyl-3-(4-aminophenyl)-3-ethylpiperidin-2,6-dionen.
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- Archiv der Pharmazie, 1987, v. 320, n. 1, p. 51, doi. 10.1002/ardp.19873200109
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- Article