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Mutation in the Common Docking Domain Affects MAP Kinase ERK2 Catalysis and Stability.
Published in:
Cancers, 2023, v. 15, n. 11, p. 2938, doi. 10.3390/cancers15112938
By:
- Novak, Leonore;
- Petrosino, Maria;
- Pasquo, Alessandra;
- Chaikuad, Apirat;
- Chiaraluce, Roberta;
- Knapp, Stefan;
- Consalvi, Valerio
Publication type:
Article
Discovery of a Potent and Highly Isoform-Selective Inhibitor of the Neglected Ribosomal Protein S6 Kinase Beta 2 (S6K2).
Published in:
Cancers, 2021, v. 13, n. 20, p. 5133, doi. 10.3390/cancers13205133
By:
- Gerstenecker, Stefan;
- Haarer, Lisa;
- Schröder, Martin;
- Kudolo, Mark;
- Schwalm, Martin P.;
- Wydra, Valentin;
- Serafim, Ricardo A. M.;
- Chaikuad, Apirat;
- Knapp, Stefan;
- Laufer, Stefan;
- Gehringer, Matthias
Publication type:
Article
Furo[3,2‐b]pyridine: A Privileged Scaffold for Highly Selective Kinase Inhibitors and Effective Modulators of the Hedgehog Pathway.
Published in:
Angewandte Chemie International Edition, 2019, v. 58, n. 4, p. 1062, doi. 10.1002/anie.201810312
By:
- Němec, Václav;
- Hylsová, Michaela;
- Maier, Lukáš;
- Flegel, Jana;
- Sievers, Sonja;
- Ziegler, Slava;
- Schröder, Martin;
- Berger, Benedict‐Tilman;
- Chaikuad, Apirat;
- Valčíková, Barbora;
- Uldrijan, Stjepan;
- Drápela, Stanislav;
- Souček, Karel;
- Waldmann, Herbert;
- Knapp, Stefan;
- Paruch, Kamil
Publication type:
Article
Discovery of an MLLT1/3 YEATS Domain Chemical Probe.
Published in:
Angewandte Chemie International Edition, 2018, v. 57, n. 50, p. 16302, doi. 10.1002/anie.201810617
By:
- Moustakim, Moses;
- Christott, Thomas;
- Monteiro, Octovia P.;
- Bennett, James;
- Giroud, Charline;
- Ward, Jennifer;
- Rogers, Catherine M.;
- Smith, Paul;
- Panagakou, Ioanna;
- Díaz‐Sáez, Laura;
- Felce, Suet Ling;
- Gamble, Vicki;
- Gileadi, Carina;
- Halidi, Nadia;
- Heidenreich, David;
- Chaikuad, Apirat;
- Knapp, Stefan;
- Huber, Kilian V. M.;
- Farnie, Gillian;
- Heer, Jag
Publication type:
Article
Halogen–Aromatic π Interactions Modulate Inhibitor Residence Times.
Published in:
Angewandte Chemie International Edition, 2018, v. 57, n. 24, p. 7220, doi. 10.1002/anie.201801666
By:
- Heroven, Christina;
- Georgi, Victoria;
- Ganotra, Gaurav K.;
- Brennan, Paul;
- Wolfreys, Finn;
- Wade, Rebecca C.;
- Fernández‐Montalván, Amaury E.;
- Chaikuad, Apirat;
- Knapp, Stefan
Publication type:
Article
Inside Back Cover: The Cysteinome of Protein Kinases as a Target in Drug Development (Angew. Chem. Int. Ed. 16/2018).
Published in:
Angewandte Chemie International Edition, 2018, v. 57, n. 16, p. 4429, doi. 10.1002/anie.201802502
By:
- Chaikuad, Apirat;
- Koch, Pierre;
- Laufer, Stefan A.;
- Knapp, Stefan
Publication type:
Article
The Cysteinome of Protein Kinases as a Target in Drug Development.
Published in:
Angewandte Chemie International Edition, 2018, v. 57, n. 16, p. 4372, doi. 10.1002/anie.201707875
By:
- Chaikuad, Apirat;
- Koch, Pierre;
- Laufer, Stefan A.;
- Knapp, Stefan
Publication type:
Article
Discovery of a PCAF Bromodomain Chemical Probe.
Published in:
Angewandte Chemie International Edition, 2017, v. 56, n. 3, p. 827, doi. 10.1002/anie.201610816
By:
- Moustakim, Moses;
- Clark, Peter G. K.;
- Trulli, Laura;
- Fuentes de Arriba, Angel L.;
- Ehebauer, Matthias T.;
- Chaikuad, Apirat;
- Murphy, Emma J.;
- Mendez-Johnson, Jacqui;
- Daniels, Danette;
- Hou, Chun-Feng D.;
- Lin, Yu-Hui;
- Walker, John R.;
- Hui, Raymond;
- Yang, Hongbing;
- Dorrell, Lucy;
- Rogers, Catherine M.;
- Monteiro, Octovia P.;
- Fedorov, Oleg;
- Huber, Kilian V. M.;
- Knapp, Stefan
Publication type:
Article
Back Cover: Discovery of a PCAF Bromodomain Chemical Probe (Angew. Chem. Int. Ed. 3/2017).
Published in:
Angewandte Chemie International Edition, 2017, v. 56, n. 3, p. 908, doi. 10.1002/anie.201612063
By:
- Moustakim, Moses;
- Clark, Peter G. K.;
- Trulli, Laura;
- Fuentes de Arriba, Angel L.;
- Ehebauer, Matthias T.;
- Chaikuad, Apirat;
- Murphy, Emma J.;
- Mendez-Johnson, Jacqui;
- Daniels, Danette;
- Hou, Chun-Feng D.;
- Lin, Yu-Hui;
- Walker, John R.;
- Hui, Raymond;
- Yang, Hongbing;
- Dorrell, Lucy;
- Rogers, Catherine M.;
- Monteiro, Octovia P.;
- Fedorov, Oleg;
- Huber, Kilian V. M.;
- Knapp, Stefan
Publication type:
Article
Discovery of Potent and Exquisitely Selective Inhibitors of Kinase CK1 with Tunable Isoform Selectivity.
Published in:
Angewandte Chemie, 2023, v. 135, n. 11, p. 1, doi. 10.1002/ange.202217532
By:
- Němec, Václav;
- Khirsariya, Prashant;
- Janovská, Pavlína;
- Moyano, Paula Martín;
- Maier, Lukáš;
- Procházková, Petra;
- Kebková, Pavlína;
- Gybel', Tomáš;
- Berger, Benedict‐Tilman;
- Chaikuad, Apirat;
- Reinecke, Maria;
- Kuster, Bernhard;
- Knapp, Stefan;
- Bryja, Vítězslav;
- Paruch, Kamil
Publication type:
Article
Controlling the Covalent Reactivity of a Kinase Inhibitor with Light.
Published in:
Angewandte Chemie, 2021, v. 133, n. 37, p. 20340, doi. 10.1002/ange.202103767
By:
- Reynders, Martin;
- Chaikuad, Apirat;
- Berger, Benedict‐Tilman;
- Bauer, Katharina;
- Koch, Pierre;
- Laufer, Stefan;
- Knapp, Stefan;
- Trauner, Dirk
Publication type:
Article
Lessons from LIMK1 enzymology and their impact on inhibitor design.
Published in:
Biochemical Journal, 2019, v. 476, n. 21, p. 3197, doi. 10.1042/BCJ20190517
By:
- Salah, Eidarus;
- Chatterjee, Deep;
- Beltrami, Alessandra;
- Tumber, Anthony;
- Preuss, Franziska;
- Canning, Peter;
- Chaikuad, Apirat;
- Knaus, Petra;
- Knapp, Stefan;
- Bullock, Alex N.;
- Mathea, Sebastian
Publication type:
Article
Conservation of structure, function and inhibitor binding in UNC-51-like kinase 1 and 2 (ULK1/2).
Published in:
Biochemical Journal, 2019, v. 476, n. 5, p. 875, doi. 10.1042/BCJ20190038
By:
- Chaikuad, Apirat;
- Koschade, Sebastian E.;
- Stolz, Alexandra;
- Zivkovic, Katarina;
- Pohl, Christian;
- Shaid, Shabnam;
- Ren, Huiyu;
- Lambert, Lester J.;
- Cosford, Nicholas D. P.;
- Brandts, Christian H.;
- Knapp, Stefan
Publication type:
Article
Structure of cyclin G-associated kinase (GAK) trapped in different conformations using nanobodies.
Published in:
Biochemical Journal, 2014, v. 459, n. 1, p. 59, doi. 10.1042/BJ20131399
By:
- CHAIKUAD, Apirat;
- KEATES, Tracy;
- VINCKE, Cécile;
- KAUFHOLZ, Melanie;
- ZENN, Michael;
- ZIMMERMANN, Bastian;
- GUTIÉRREZ, Carlos;
- Rong-guang ZHANG;
- HATZOS-SKINTGES, Catherine;
- JOACHIMIAK, Andrzej;
- MUYLDERMANS, Serge;
- HERBERG, Friedrich W.;
- KNAPP, Stefan;
- MÜLLER, Susanne
Publication type:
Article
Hepatitis Delta Virus histone mimicry drives the recruitment of chromatin remodelers for viral RNA replication.
Published in:
Nature Communications, 2020, v. 11, n. 1, p. 1, doi. 10.1038/s41467-020-14299-9
By:
- Abeywickrama-Samarakoon, Natali;
- Cortay, Jean-Claude;
- Sureau, Camille;
- Müller, Susanne;
- Alfaiate, Dulce;
- Guerrieri, Francesca;
- Chaikuad, Apirat;
- Schröder, Martin;
- Merle, Philippe;
- Levrero, Massimo;
- Dény, Paul
Publication type:
Article
A Consensus Compound/Bioactivity Dataset for Data-Driven Drug Design and Chemogenomics.
Published in:
Molecules, 2022, v. 27, n. 8, p. N.PAG, doi. 10.3390/molecules27082513
By:
- Isigkeit, Laura;
- Chaikuad, Apirat;
- Merk, Daniel
Publication type:
Article
Image-Based Annotation of Chemogenomic Libraries for Phenotypic Screening.
Published in:
Molecules, 2022, v. 27, n. 4, p. 1439, doi. 10.3390/molecules27041439
By:
- Tjaden, Amelie;
- Chaikuad, Apirat;
- Kowarz, Eric;
- Marschalek, Rolf;
- Knapp, Stefan;
- Schröder, Martin;
- Müller, Susanne
Publication type:
Article
Crystal Structure-Guided Design of Bisubstrate Inhibitors and Photoluminescent Probes for Protein Kinases of the PIM Family.
Published in:
Molecules, 2021, v. 26, n. 14, p. 4353, doi. 10.3390/molecules26144353
By:
- Nonga, Olivier E.;
- Lavogina, Darja;
- Enkvist, Erki;
- Kestav, Katrin;
- Chaikuad, Apirat;
- Dixon-Clarke, Sarah E.;
- Bullock, Alex N.;
- Kopanchuk, Sergei;
- Ivan, Taavi;
- Ekambaram, Ramesh;
- Viht, Kaido;
- Knapp, Stefan;
- Uri, Asko
Publication type:
Article
7-(2-Anilinopyrimidin-4-yl)-1-benzazepin-2-ones Designed by a "Cut and Glue" Strategy Are Dual Aurora A/VEGF-R Kinase Inhibitors.
Published in:
Molecules, 2021, v. 26, n. 6, p. 1611, doi. 10.3390/molecules26061611
By:
- Karatas, Mehmet;
- Chaikuad, Apirat;
- Berger, Bianca;
- Kubbutat, Michael H. G.;
- Totzke, Frank;
- Knapp, Stefan;
- Kunick, Conrad;
- Chiara, Brullo
Publication type:
Article
How to Separate Kinase Inhibition from Undesired Monoamine Oxidase A Inhibition—The Development of the DYRK1A Inhibitor AnnH75 from the Alkaloid Harmine.
Published in:
Molecules, 2020, v. 25, n. 24, p. 5962, doi. 10.3390/molecules25245962
By:
- Wurzlbauer, Anne;
- Rüben, Katharina;
- Gürdal, Ece;
- Chaikuad, Apirat;
- Knapp, Stefan;
- Sippl, Wolfgang;
- Becker, Walter;
- Bracher, Franz;
- Ntie-Kang, Fidele
Publication type:
Article
[b]-Annulated Halogen-Substituted Indoles as Potential DYRK1A Inhibitors.
Published in:
Molecules, 2019, v. 24, n. 22, p. 4090, doi. 10.3390/molecules24224090
By:
- Lechner, Christian;
- Flaßhoff, Maren;
- Falke, Hannes;
- Preu, Lutz;
- Loaëc, Nadége;
- Meijer, Laurent;
- Knapp, Stefan;
- Chaikuad, Apirat;
- Kunick, Conrad;
- Black, David StC
Publication type:
Article
DARPins detect the formation of hetero-tetramers of p63 and p73 in epithelial tissues and in squamous cell carcinoma.
Published in:
Cell Death & Disease, 2023, v. 14, n. 10, p. 1, doi. 10.1038/s41419-023-06213-0
By:
- Strubel, Alexander;
- Münick, Philipp;
- Hartmann, Oliver;
- Chaikuad, Apirat;
- Dreier, Birgit;
- Schaefer, Jonas V.;
- Gebel, Jakob;
- Osterburg, Christian;
- Tuppi, Marcel;
- Schäfer, Birgit;
- Buck, Viktoria;
- Rosenfeldt, Mathias;
- Knapp, Stefan;
- Plückthun, Andreas;
- Diefenbacher, Markus E.;
- Dötsch, Volker
Publication type:
Article
Co-crystal structures of the protein kinase haspin with bisubstrate inhibitors.
Published in:
Acta Crystallographica: Section F, Structural Biology Communications, 2016, v. 72, n. 5, p. 339, doi. 10.1107/S2053230X16004611
By:
- Lavogina, Darja;
- Kestav, Katrin;
- Uri, Asko;
- Chaikuad, Apirat;
- Heroven, Christina;
- Knapp, Stefan
Publication type:
Article
Structural consequences of BMPR2 kinase domain mutations causing pulmonary arterial hypertension.
Published in:
Scientific Reports, 2019, v. 9, n. 1, p. N.PAG, doi. 10.1038/s41598-019-54830-7
By:
- Chaikuad, Apirat;
- Thangaratnarajah, Chancievan;
- von Delft, Frank;
- Bullock, Alex N.
Publication type:
Article
The ins and outs of selective kinase inhibitor development.
Published in:
Nature Chemical Biology, 2015, v. 11, n. 11, p. 818, doi. 10.1038/nchembio.1938
By:
- Müller, Susanne;
- Chaikuad, Apirat;
- Gray, Nathanael S;
- Knapp, Stefan
Publication type:
Article
A unique inhibitor binding site in ERK1/2 is associated with slow binding kinetics.
Published in:
Nature Chemical Biology, 2014, v. 10, n. 10, p. 853, doi. 10.1038/nchembio.1629
By:
- Chaikuad, Apirat;
- M C Tacconi, Eliana;
- Zimmer, Jutta;
- Liang, Yanke;
- Gray, Nathanael S;
- Tarsounas, Madalena;
- Knapp, Stefan
Publication type:
Article
Structure of human aspartyl aminopeptidase complexed with substrate analogue: insight into catalytic mechanism, substrate specificity and M18 peptidase family.
Published in:
BMC Structural Biology, 2012, v. 12, n. 1, p. 14, doi. 10.1186/1472-6807-12-14
By:
- Chaikuad, Apirat;
- Pilka, Ewa S.;
- De Riso, Antonio;
- von Delft, Frank;
- Kavanagh, Kathryn L.;
- V‚nien-Bryan, Catherine;
- Oppermann, Udo;
- Yue, Wyatt W.
Publication type:
Article
Copper is required for oncogenic BRAF signalling and tumorigenesis.
Published in:
Nature, 2014, v. 509, n. 7501, p. 492, doi. 10.1038/nature13180
By:
- Brady, Donita C.;
- Crowe, Matthew S.;
- Turski, Michelle L.;
- Hobbs, G. Aaron;
- Yao, Xiaojie;
- Chaikuad, Apirat;
- Knapp, Stefan;
- Xiao, Kunhong;
- Campbell, Sharon L.;
- Thiele, Dennis J.;
- Counter, Christopher M.
Publication type:
Article
Discovery of Potent and Exquisitely Selective Inhibitors of Kinase CK1 with Tunable Isoform Selectivity.
Published in:
Angewandte Chemie International Edition, 2023, v. 62, n. 11, p. 1, doi. 10.1002/anie.202217532
By:
- Němec, Václav;
- Khirsariya, Prashant;
- Janovská, Pavlína;
- Moyano, Paula Martín;
- Maier, Lukáš;
- Procházková, Petra;
- Kebková, Pavlína;
- Gybel', Tomáš;
- Berger, Benedict‐Tilman;
- Chaikuad, Apirat;
- Reinecke, Maria;
- Kuster, Bernhard;
- Knapp, Stefan;
- Bryja, Vítězslav;
- Paruch, Kamil
Publication type:
Article
Controlling the Covalent Reactivity of a Kinase Inhibitor with Light.
Published in:
Angewandte Chemie International Edition, 2021, v. 60, n. 37, p. 20178, doi. 10.1002/anie.202103767
By:
- Reynders, Martin;
- Chaikuad, Apirat;
- Berger, Benedict‐Tilman;
- Bauer, Katharina;
- Koch, Pierre;
- Laufer, Stefan;
- Knapp, Stefan;
- Trauner, Dirk
Publication type:
Article
The orphan nuclear receptor Nurr1 is responsive to non-steroidal anti-inflammatory drugs.
Published in:
Communications Chemistry, 2020, v. 3, n. 1, p. 1, doi. 10.1038/s42004-020-0331-0
By:
- Willems, Sabine;
- Kilu, Whitney;
- Ni, Xiaomin;
- Chaikuad, Apirat;
- Knapp, Stefan;
- Heering, Jan;
- Merk, Daniel
Publication type:
Article
Modulation of tau tubulin kinases (TTBK1 and TTBK2) impacts ciliogenesis.
Published in:
Scientific Reports, 2023, v. 13, n. 1, p. 1, doi. 10.1038/s41598-023-32854-4
By:
- Bashore, Frances M.;
- Marquez, Ariana B.;
- Chaikuad, Apirat;
- Howell, Stefanie;
- Dunn, Andrea S.;
- Beltran, Alvaro A.;
- Smith, Jeffery L.;
- Drewry, David H.;
- Beltran, Adriana S.;
- Axtman, Alison D.
Publication type:
Article
A New Class of Small Molecule Inhibitor of BMP Signaling.
Published in:
PLoS ONE, 2013, v. 8, n. 4, p. 1, doi. 10.1371/journal.pone.0062721
By:
- Sanvitale, Caroline E.;
- Kerr, Georgina;
- Chaikuad, Apirat;
- Ramel, Marie-Christine;
- Mohedas, Agustin H.;
- Reichert, Sabine;
- Wang, You;
- Triffitt, James T.;
- Cuny, Gregory D.;
- Yu, Paul B.;
- Hill, Caroline S.;
- Bullock, Alex N.
Publication type:
Article
Structural Comparison of Human Mammalian Ste20-Like Kinases.
Published in:
PLoS ONE, 2010, v. 5, n. 8, p. 1, doi. 10.1371/journal.pone.0011905
By:
- Record, Christopher J.;
- Chaikuad, Apirat;
- Rellos, Peter;
- Das, Sanjan;
- Pike, Ashley C. W.;
- Fedorov, Oleg;
- Marsden, Brian D.;
- Knapp, Stefan;
- Wen Hwa Lee
Publication type:
Article
Identification of CLK1 Inhibitors by a Fragment-linking Based Virtual Screening.
Published in:
Molecular Informatics, 2017, v. 36, n. 4, p. n/a, doi. 10.1002/minf.201600123
By:
- Walter, Anne;
- Chaikuad, Apirat;
- Loaëc, Nadège;
- Preu, Lutz;
- Knapp, Stefan;
- Meijer, Laurent;
- Kunick, Conrad;
- Koch, Oliver
Publication type:
Article
Atad2 is a generalist facilitator of chromatin dynamics in embryonic stem cells.
Published in:
Journal of Molecular Cell Biology, 2016, v. 8, n. 4, p. 349, doi. 10.1093/jmcb/mjv060
By:
- Yuichi Morozumi;
- Boussouar, Fayçal;
- Minjia Tan;
- Chaikuad, Apirat;
- Jamshidikia, Mahya;
- Colak, Gozde;
- Huang He;
- Litong Nie;
- Petosa, Carlo;
- de Dieuleveult, Maud;
- Curtet, Sandrine;
- Vitte, Anne-Laure;
- Rabatel, Clothilde;
- Debernardi, Alexandra;
- Cosset, François-Loïc;
- Verhoeyen, Els;
- Emadali, Anouk;
- Schweifer, Norbert;
- Gianni, Davide;
- Gut, Marta
Publication type:
Article
Furo[3,2‐b]pyridine: A Privileged Scaffold for Highly Selective Kinase Inhibitors and Effective Modulators of the Hedgehog Pathway.
Published in:
Angewandte Chemie, 2019, v. 131, n. 4, p. 1074, doi. 10.1002/ange.201810312
By:
- Němec, Václav;
- Hylsová, Michaela;
- Maier, Lukáš;
- Flegel, Jana;
- Sievers, Sonja;
- Ziegler, Slava;
- Schröder, Martin;
- Berger, Benedict‐Tilman;
- Chaikuad, Apirat;
- Valčíková, Barbora;
- Uldrijan, Stjepan;
- Drápela, Stanislav;
- Souček, Karel;
- Waldmann, Herbert;
- Knapp, Stefan;
- Paruch, Kamil
Publication type:
Article
Halogenaromatische π‐Wechselwirkungen modulieren die Verweilzeit von Inhibitoren.
Published in:
Angewandte Chemie, 2018, v. 130, n. 24, p. 7338, doi. 10.1002/ange.201801666
By:
- Heroven, Christina;
- Georgi, Victoria;
- Ganotra, Gaurav K.;
- Brennan, Paul;
- Wolfreys, Finn;
- Wade, Rebecca C.;
- Fernández‐Montalván, Amaury E.;
- Chaikuad, Apirat;
- Knapp, Stefan
Publication type:
Article
Innenrücktitelbild: Das Cysteinom der Proteinkinasen als Zielstruktur in der Arzneistoffentwicklung (Angew. Chem. 16/2018).
Published in:
Angewandte Chemie, 2018, v. 130, n. 16, p. 4517, doi. 10.1002/ange.201802502
By:
- Chaikuad, Apirat;
- Koch, Pierre;
- Laufer, Stefan A.;
- Knapp, Stefan
Publication type:
Article
Das Cysteinom der Proteinkinasen als Zielstruktur in der Arzneistoffentwicklung.
Published in:
Angewandte Chemie, 2018, v. 130, n. 16, p. 4456, doi. 10.1002/ange.201707875
By:
- Chaikuad, Apirat;
- Koch, Pierre;
- Laufer, Stefan A.;
- Knapp, Stefan
Publication type:
Article
Discovery of a PCAF Bromodomain Chemical Probe.
Published in:
Angewandte Chemie, 2017, v. 129, n. 3, p. 845, doi. 10.1002/ange.201610816
By:
- Moustakim, Moses;
- Clark, Peter G. K.;
- Trulli, Laura;
- Fuentes de Arriba, Angel L.;
- Ehebauer, Matthias T.;
- Chaikuad, Apirat;
- Murphy, Emma J.;
- Mendez ‐ Johnson, Jacqui;
- Daniels, Danette;
- Hou, Chun ‐ Feng D.;
- Lin, Yu ‐ Hui;
- Walker, John R.;
- Hui, Raymond;
- Yang, Hongbing;
- Dorrell, Lucy;
- Rogers, Catherine M.;
- Monteiro, Octovia P.;
- Fedorov, Oleg;
- Huber, Kilian V. M.;
- Knapp, Stefan
Publication type:
Article
Rücktitelbild: Discovery of a PCAF Bromodomain Chemical Probe (Angew. Chem. 3/2017).
Published in:
Angewandte Chemie, 2017, v. 129, n. 3, p. 928, doi. 10.1002/ange.201612063
By:
- Moustakim, Moses;
- Clark, Peter G. K.;
- Trulli, Laura;
- Fuentes de Arriba, Angel L.;
- Ehebauer, Matthias T.;
- Chaikuad, Apirat;
- Murphy, Emma J.;
- Mendez ‐ Johnson, Jacqui;
- Daniels, Danette;
- Hou, Chun ‐ Feng D.;
- Lin, Yu ‐ Hui;
- Walker, John R.;
- Hui, Raymond;
- Yang, Hongbing;
- Dorrell, Lucy;
- Rogers, Catherine M.;
- Monteiro, Octovia P.;
- Fedorov, Oleg;
- Huber, Kilian V. M.;
- Knapp, Stefan
Publication type:
Article
A Specific and Covalent JNK-1 Ligand Selected from an Encoded Self-Assembling Chemical Library.
Published in:
Chemistry - A European Journal, 2017, v. 23, n. 34, p. 8152, doi. 10.1002/chem.201701644
By:
- Zimmermann, Gunther;
- Rieder, Ulrike;
- Bajic, Davor;
- Vanetti, Sara;
- Chaikuad, Apirat;
- Knapp, Stefan;
- Scheuermann, Jörg;
- Mattarella, Martin;
- Neri, Dario
Publication type:
Article
Comparative structural analyses and nucleotide-binding characterization of the four KH domains of FUBP1.
Published in:
Scientific Reports, 2020, v. 10, n. 1, p. 1, doi. 10.1038/s41598-020-69832-z
By:
- Ni, Xiaomin;
- Knapp, Stefan;
- Chaikuad, Apirat
Publication type:
Article
Molecular structures of cdc2-like kinases in complex with a new inhibitor chemotype.
Published in:
PLoS ONE, 2018, v. 13, n. 5, p. 1, doi. 10.1371/journal.pone.0196761
By:
- Walter, Anne;
- Chaikuad, Apirat;
- Helmer, Renate;
- Loaëc, Nadège;
- Preu, Lutz;
- Ott, Ingo;
- Knapp, Stefan;
- Meijer, Laurent;
- Kunick, Conrad
Publication type:
Article
Radiolabeled cCPE Peptides for SPECT Imaging of Claudin-4 Overexpression in Pancreatic Cancer.
Published in:
Journal of Nuclear Medicine, 2020, v. 61, n. 12, p. 1, doi. 10.2967/jnumed.120.243113
By:
- Torres, Julia Baguña;
- Mosley, Michael;
- Koustoulidou, Sofia;
- Hopkins, Samantha;
- Knapp, Stefan;
- Chaikuad, Apirat;
- Masuo Kondoh;
- Keisuke Tachibana;
- Kersemans, Veerle;
- Cornelissen, Bart
Publication type:
Article
Radiolabeled cCPE Peptides for SPECT Imaging of Claudin-4 Overexpression in Pancreatic Cancer.
Published in:
Journal of Nuclear Medicine, 2020, v. 61, n. 11, p. 1, doi. 10.2967/jnumed.120.243113
By:
- Torres, Julia Baguña;
- Mosley, Michael;
- Koustoulidou, Sofia;
- Hopkins, Samantha;
- Knapp, Stefan;
- Chaikuad, Apirat;
- Masuo Kondoh;
- Keisuke Tachibana;
- Kersemans, Veerle;
- Cornelissen, Bart
Publication type:
Article
Radiolabeled cCPE Peptides for SPECT Imaging of Claudin-4 Overexpression in Pancreatic Cancer.
Published in:
Journal of Nuclear Medicine, 2020, v. 61, n. 10, p. 1, doi. 10.2967/jnumed.120.243113
By:
- Torres, Julia Baguña;
- Mosley, Michael;
- Koustoulidou, Sofia;
- Hopkins, Samantha;
- Knapp, Stefan;
- Chaikuad, Apirat;
- Kondoh, Masuo;
- Tachibana, Keisuke;
- Kersemans, Veerle;
- Cornelissen, Bart
Publication type:
Article
Radiolabeled cCPE Peptides for SPECT Imaging of Claudin-4 Overexpression in Pancreatic Cancer.
Published in:
Journal of Nuclear Medicine, 2020, v. 61, n. 9, p. 1, doi. 10.2967/jnumed.120.243113
By:
- Baguña Torres, Julia;
- Mosley, Michael;
- Koustoulidou, Sofia;
- Hopkins, Samantha;
- Knapp, Stefan;
- Chaikuad, Apirat;
- Kondoh, Masuo;
- Tachibana, Keisuke;
- Kersemans, Veerle;
- Cornelissen, Bart
Publication type:
Article
Radiolabeled cCPE Peptides for SPECT Imaging of Claudin-4 Overexpression in Pancreatic Cancer.
Published in:
Journal of Nuclear Medicine, 2020, v. 61, n. 7, p. 1, doi. 10.2967/jnumed.120.243113
By:
- Torres, Julia Baguña;
- Mosley, Michael;
- Koustoulidou, Sofia;
- Hopkins, Samantha;
- Knapp, Stefan;
- Chaikuad, Apirat;
- Kondoh, Masuo;
- Tachibana, Keisuke;
- Kersemans, Veerle;
- Cornelissen, Bart
Publication type:
Article

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