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Antimycobacterial activity of novel 1-(5-cyclobutyl-1,3-oxazol-2-yl)-3-(sub)phenyl/pyridylthiourea compounds endowed with high activity toward multidrug-resistant Mycobacterium tuberculosis.
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- Journal of Antimicrobial Chemotherapy (JAC), 2007, v. 59, n. 6, p. 1194, doi. 10.1093/jac/dkm085
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- Article
Design and Development of Mycobacterium tuberculosis Lysine ɛ-Aminotransferase Inhibitors for Latent Tuberculosis Infection.
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- Chemical Biology & Drug Design, 2016, v. 87, n. 2, p. 265, doi. 10.1111/cbdd.12655
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- Article
Targeting NAMPT for Therapeutic Intervention in Cancer.
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- Chemical Biology & Drug Design, 2015, v. 86, n. 4, p. 881, doi. 10.1111/cbdd.12562
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- Article
Design and Biological Evaluation of Furan/Pyrrole/Thiophene-2-carboxamide Derivatives as Efficient DNA GyraseB Inhibitors of Staphylococcus aureus.
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- Chemical Biology & Drug Design, 2015, v. 86, n. 4, p. 918, doi. 10.1111/cbdd.12529
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Discovery and Structure Optimization of a Series of Isatin Derivatives as Mycobacterium tuberculosis Chorismate Mutase Inhibitors.
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- Chemical Biology & Drug Design, 2014, v. 83, n. 4, p. 498, doi. 10.1111/cbdd.12265
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- Article
Discovery of Novel 1,2,4-Triazol-5-Ones as Tumor Necrosis Factor-Alpha Inhibitors for the Treatment of Neuropathic Pain.
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- Chemical Biology & Drug Design, 2012, v. 80, n. 6, p. 961, doi. 10.1111/cbdd.12049
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- Article
Synthesis and Antimycobacterial Evaluation of Novel Phthalazin-4-ylacetamides Against log- and Starved Phase Cultures.
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- Chemical Biology & Drug Design, 2010, v. 75, n. 4, p. 381, doi. 10.1111/j.1747-0285.2010.00947.x
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- Article
Inhibition of lipopolysaccharide (LPS)-induced neuroinflammatory response by polysaccharide fractions of <italic>Khaya grandifoliola</italic> (C.D.C.) stem bark, <italic>Cryptolepis sanguinolenta</italic> (Lindl.) Schltr and <italic>Cymbopogon citratus</italic> Stapf leaves in raw 264.7 macrophages and U87 glioblastoma cells
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- BMC Complementary & Alternative Medicine, 2018, v. 18, p. 1, doi. 10.1186/s12906-018-2156-2
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- Article
Design and Synthesis of New Etodolac‐Pyridazinones as Potent Anticancer Agents Using Pb(OAc)<sub>4</sub> to Assist N‐N Bond Formation.
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- ChemistrySelect, 2018, v. 3, n. 18, p. 5050, doi. 10.1002/slct.201800459
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- Article
Synthesis of new pyrazole-triazole hybrids by click reaction using a green solvent and evaluation of their antitubercular and antibacterial activity.
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- Research on Chemical Intermediates, 2016, v. 42, n. 4, p. 3721, doi. 10.1007/s11164-015-2241-9
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- Article
Structure-based design of diverse inhibitors of Mycobacterium tuberculosis N-acetylglucosamine-1-phosphate uridyltransferase: combined molecular docking, dynamic simulation, and biological activity.
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- Journal of Molecular Modeling, 2015, v. 21, n. 7, p. 174, doi. 10.1007/s00894-015-2704-3
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- Article
Design and synthesis of oxaprozin‐1,3,4‐oxadiazole hybrids as potential anticancer and antibacterial agents.
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- Journal of Heterocyclic Chemistry, 2020, v. 57, n. 3, p. 1071, doi. 10.1002/jhet.3842
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- Article
Heteroaryl-substuted semicarbazones: Synthesis and anticonvulsant activity of N-(3-methylpyridin-2-yl)-substituted semicarbazones.
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- Journal of Heterocyclic Chemistry, 2006, v. 43, n. 5, p. 1287, doi. 10.1002/jhet.5570430522
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- Article
Targeting multiple response regulators of Mycobacterium tuberculosis augments the host immune response to infection.
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- Scientific Reports, 2016, p. 25851, doi. 10.1038/srep25851
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- Article
Design and development of novel inhibitors for the treatment of latent tuberculosis.
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- International Journal of Mycobacteriology, 2016, v. 5, p. S121, doi. 10.1016/j.ijmyco.2016.09.006
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- Article
Benzothiazinone-piperazine derivatives as efficient Mycobacterium tuberculosis DNA gyrase inhibitors.
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- International Journal of Mycobacteriology, 2015, v. 4, n. 2, p. 104, doi. 10.1016/j.ijmyco.2015.02.002
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- Article
Optimization and validation of Mycobacterium marinum-induced adult zebrafish model for evaluation of oral anti-tuberculosis drugs.
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- International Journal of Mycobacteriology, 2014, v. 3, n. 4, p. 259, doi. 10.1016/j.ijmyco.2014.10.001
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- Article
Investigating structure–activity relationship and mechanism of action of antitubercular 1-(4-chlorophenyl)-4-(4-hydroxy-3-methoxy-5-nitrobenzylidene) pyrazolidine-3,5-dione [CD59].
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- International Journal of Mycobacteriology, 2014, v. 3, n. 2, p. 117, doi. 10.1016/j.ijmyco.2014.02.006
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- Article
A Novel, Potent, Small Molecule AKT Inhibitor Exhibits Efficacy against Lung Cancer Cells In Vitro.
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- Cancer Research & Treatment, 2015, v. 47, n. 4, p. 913, doi. 10.4143/crt.2014.057
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- Article
Novel Thiazolidinone-Azole Hybrids: Design, Synthesis and Antimycobacterial Activity Studies.
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- Iranian Journal of Pharmaceutical Research, 2016, v. 15, n. 4, p. 783
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- Article
Synthesis and anti-mycobacterial activity of 4-(4-phenyl-1 H-1,2,3-triazol-1-yl)salicylhydrazones: revitalizing an old drug.
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- Archives of Pharmacal Research, 2017, v. 40, n. 2, p. 168, doi. 10.1007/s12272-016-0882-x
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- Article
Newer N-Phthaloyl GABA Derivatives with Antiallodynic and Antihyperalgesic Activities in Both Sciatic Nerve and Spinal Nerve Ligation Models of Neuropathic Pain.
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- Pharmacology, 2007, v. 81, n. 1, p. 21, doi. 10.1159/000107711
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- Article
Structural Models for the Design of PKMzeta Inhibitors with Neurobiological Indications.
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- Molecular Informatics, 2015, v. 34, n. 10, p. 665, doi. 10.1002/minf.201500003
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- Article
Design of Novel Mycobacterium tuberculosis Pantothenate Synthetase Inhibitors: Virtual Screening, Synthesis and In Vitro Biological Activities.
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- Molecular Informatics, 2015, v. 34, n. 2/3, p. 147, doi. 10.1002/minf.201400120
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- Article
Discovery of Novel Mycobacterial DNA Gyrase B Inhibitors: In Silico and In Vitro Biological Evaluation.
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- Molecular Informatics, 2014, v. 33, n. 9, p. 597, doi. 10.1002/minf.201400058
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- Article
Multiple e-Pharmacophore Modeling Combined with High-Throughput Virtual Screening and Docking to Identify Potential Inhibitors of β-Secretase(BACE1).
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- Molecular Informatics, 2013, v. 32, n. 4, p. 385, doi. 10.1002/minf.201200169
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- Article
Enhanced ranking of PknB Inhibitors using data fusion methods.
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- Journal of Cheminformatics, 2013, v. 5, n. 1, p. 1, doi. 10.1186/1758-2946-5-2
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- Article
Depletion of M. tuberculosis GlmU from Infected Murine Lungs Effects the Clearance of the Pathogen.
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- PLoS Pathogens, 2015, v. 11, n. 10, p. 1, doi. 10.1371/journal.ppat.1005235
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- Article
Synthesis of novel cytotoxic tetracyclic acridone derivatives and study of their molecular docking, ADMET, QSAR, bioactivity and protein binding properties.
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- Scientific Reports, 2020, v. 10, n. 1, p. N.PAG, doi. 10.1038/s41598-020-77590-1
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- Article
Bis-spirochromanones as potent inhibitors of Mycobacterium tuberculosis: synthesis and biological evaluation.
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- Molecular Diversity, 2017, v. 21, n. 4, p. 999, doi. 10.1007/s11030-017-9779-y
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- Article
Cathepsin D inhibitors as potential therapeutics for breast cancer treatment: Molecular docking and bioevaluation against triple-negative and triple-positive breast cancers.
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- Molecular Diversity, 2016, v. 20, n. 2, p. 521, doi. 10.1007/s11030-015-9645-8
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- Article
Deep Learning Classifies Low- and High-Grade Glioma Patients with High Accuracy, Sensitivity, and Specificity Based on Their Brain White Matter Networks Derived from Diffusion Tensor Imaging.
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- Diagnostics (2075-4418), 2022, v. 12, n. 12, p. 3216, doi. 10.3390/diagnostics12123216
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Targeting hexokinase 2 for oral cancer therapy: structure-based design and validation of lead compounds.
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- Frontiers in Pharmacology, 2024, p. 1, doi. 10.3389/fphar.2024.1346270
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- Article
Structure-Guided Discovery of Antitubercular Agents That Target the Gyrase ATPase Domain.
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- ChemMedChem, 2016, v. 11, n. 5, p. 539, doi. 10.1002/cmdc.201500556
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- Article
Structure-Guided Design of Thiazolidine Derivatives as Mycobacterium tuberculosis Pantothenate Synthetase Inhibitors.
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- ChemMedChem, 2014, v. 9, n. 11, p. 2538, doi. 10.1002/cmdc.201402171
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- Article
Gyrase ATPase Domain as an Antitubercular Drug Discovery Platform: Structure-Based Design and Lead Optimization of Nitrothiazolyl Carboxamide Analogues.
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- ChemMedChem, 2014, v. 9, n. 8, p. 1850, doi. 10.1002/cmdc.201402035
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- Article
A small molecule inhibitor of dengue virus type 2 protease inhibits the replication of all four dengue virus serotypes in cell culture.
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- Virology Journal, 2015, v. 12, n. 1, p. 1, doi. 10.1186/s12985-015-0248-x
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- Article
N-methylisatin-beta-thiosemicarbazone derivative (SCH 16) is an inhibitor of Japanese encephalitis virus infection in vitro and in vivo.
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- Virology Journal, 2008, v. 5, p. 1, doi. 10.1186/1743-422X-5-64
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- Article