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Radiosynthesis and First-In-Human PET/MRI Evaluation with Clinical-Grade [<sup>18</sup>F]FTC-146.
- Published in:
- 2017
- By:
- Publication type:
- journal article
The evaluation of AZ66, an optimized sigma receptor antagonist, against methamphetamine-induced dopaminergic neurotoxicity and memory impairment in mice.
- Published in:
- International Journal of Neuropsychopharmacology, 2013, v. 16, n. 5, p. 1033, doi. 10.1017/S1461145712000831
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- Publication type:
- Article
Effects of the sigma-1 receptor agonist blarcamesine in a murine model of fragile X syndrome: neurobehavioral phenotypes and receptor occupancy.
- Published in:
- Scientific Reports, 2021, v. 11, n. 1, p. 1, doi. 10.1038/s41598-021-94079-7
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- Publication type:
- Article
Editorial: The Pharmacology of Kratom and Its Alkaloids.
- Published in:
- Frontiers in Pharmacology, 2022, v. 13, p. 1, doi. 10.3389/fphar.2022.878376
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- Publication type:
- Article
Searching for a Signal: Self-Reported Kratom Dose-Effect Relationships Among a Sample of US Adults With Regular Kratom Use Histories.
- Published in:
- Frontiers in Pharmacology, 2022, v. 13, p. 1, doi. 10.3389/fphar.2022.765917
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- Publication type:
- Article
Anionic phospholipids control mechanisms of GPCR-G protein recognition.
- Published in:
- Nature Communications, 2023, n. 1, p. 1, doi. 10.1038/s41467-023-36425-z
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- Publication type:
- Article
Abuse liability and therapeutic potential of the Mitragyna speciosa (kratom) alkaloids mitragynine and 7-hydroxymitragynine.
- Published in:
- 2019
- By:
- Publication type:
- journal article
In Vitro and In Vivo Pharmacological Comparison of Mu‐Opioid Receptor Activity of the Kratom (Mitragyna speciosa) Alkaloid Mitragynine and its Metabolite 7‐Hydroxymitragynine.
- Published in:
- Alzheimer's & Dementia: The Journal of the Alzheimer's Association, 2021, v. 17, p. 1, doi. 10.1002/alz.058605
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- Publication type:
- Article
Natural Corynanthe-Type Cholinesterase Inhibitors from Malaysian Uncaria attenuata Korth.: Isolation, Characterization, In Vitro and In Silico Studies.
- Published in:
- Metabolites (2218-1989), 2023, v. 13, n. 3, p. 390, doi. 10.3390/metabo13030390
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- Publication type:
- Article
A unique binding epitope for salvinorin A, a non-nitrogenous kappa opioid receptor agonist.
- Published in:
- FEBS Journal, 2006, v. 273, n. 9, p. 1966, doi. 10.1111/j.1742-4658.2006.05212.x
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- Publication type:
- Article
Health Effects Associated With Kratom (Mitragyna speciosa) and Polysubstance Use: A Narrative Review.
- Published in:
- Substance Abuse: Research & Treatment, 2022, p. 1, doi. 10.1177/11782218221095873
- By:
- Publication type:
- Article
Health Effects Associated With Kratom (Mitragyna speciosa) and Polysubstance Use: A Narrative Review.
- Published in:
- Substance Abuse: Research & Treatment, 2022, v. 16, p. 1, doi. 10.1177/11782218221095873
- By:
- Publication type:
- Article
Successful treatment of chronic knee pain following localization by a sigma-1 receptor radioligand and PET/MRI: a case report.
- Published in:
- Journal of Pain Research, 2018, v. 11, p. 2353, doi. 10.2147/JPR.S167839
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- Publication type:
- Article
Metabolism of Speciociliatine, an Overlooked Kratom Alkaloid for its Potential Pharmacological Effects.
- Published in:
- AAPS Journal, 2022, v. 24, n. 5, p. 1, doi. 10.1208/s12248-022-00736-8
- By:
- Publication type:
- Article
Discovery of a Highly Selective Sigma-2 Receptor Ligand, 1-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-3-methyl-1H-benzo[d]imidazol-2(3H)-one (CM398), with Drug-Like Properties and Antinociceptive Effects In Vivo.
- Published in:
- AAPS Journal, 2020, v. 22, n. 5, p. N.PAG, doi. 10.1208/s12248-020-00472-x
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- Publication type:
- Article
The Journey to AAPS 2020: a Reflection from Strategic Planning to PharmSci 360.
- Published in:
- AAPS Journal, 2019, v. 21, n. 1, p. 1, doi. 10.1208/s12248-018-0273-y
- By:
- Publication type:
- Article
Synthesis and Pharmacological Characterization of a Novel Sigma Receptor Ligand with Improved Metabolic Stability and Antagonistic Effects Against Methamphetamine.
- Published in:
- AAPS Journal, 2012, v. 14, n. 1, p. 43, doi. 10.1208/s12248-011-9311-8
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- Publication type:
- Article
Synthesis and Pharmacological Evaluation of 6-Acetyl-3-(4-(4-(4-fluorophenyl)piperazin-1-yl)butyl)benzo[ d]oxazol-2( 3H)-one (SN79), a Cocaine Antagonist, in Rodents.
- Published in:
- AAPS Journal, 2011, v. 13, n. 3, p. 336, doi. 10.1208/s12248-011-9274-9
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- Publication type:
- Article
Corrigendum: 2007 highlights of advances in the pharmaceutical sciences: An American Association of Pharmaceutical Scientists (AAPS) perspective.
- Published in:
- 2007
- By:
- Publication type:
- Correction Notice
419 A CTS team approach to identifying thematic constructs related to kratom use during pregnancy and breastfeeding: A qualitative analysis of social media posts.
- Published in:
- 2023
- By:
- Publication type:
- Abstract
Effects of Nutrient Fertility on Growth and Alkaloidal Content in Mitragyna speciosa (Kratom).
- Published in:
- Frontiers in Plant Science, 2020, v. 11, p. N.PAG, doi. 10.3389/fpls.2020.597696
- By:
- Publication type:
- Article
Herbal Medicines for the Management of Opioid Addiction.
- Published in:
- CNS Drugs, 2011, v. 25, n. 12, p. 999, doi. 10.2165/11596830-000000000-00000
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- Publication type:
- Article
Herbal medicines for the management of opioid addiction: safe and effective alternatives to conventional pharmacotherapy?
- Published in:
- 2011
- By:
- Publication type:
- journal article
Insight into the Willgerodt-Kindler Reaction of ω-Haloacetophenone Derivatives: Mechanistic Implication.
- Published in:
- Organic Chemistry International, 2014, p. 1, doi. 10.1155/2014/486540
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- Publication type:
- Article
Chiral separation of lobeline analogs using high performance capillary electrophoresis and derivatized cyclodextrins as chiral additives.
- Published in:
- Electrophoresis, 1999, v. 20, n. 1, p. 212, doi. 10.1002/(SICI)1522-2683(19990101)20:1<212::AID-ELPS212>3.0.CO;2-M
- By:
- Publication type:
- Article
Characterization of CM-398, a Novel Selective Sigma-2 Receptor Ligand, as a Potential Therapeutic for Neuropathic Pain.
- Published in:
- Molecules, 2022, v. 27, n. 11, p. 3617, doi. 10.3390/molecules27113617
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- Publication type:
- Article
Ecological Momentary Assessment of Self-Reported Kratom Use, Effects, and Motivations Among US Adults.
- Published in:
- JAMA Network Open, 2024, v. 7, n. 1, p. e2353401, doi. 10.1001/jamanetworkopen.2023.53401
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- Publication type:
- Article
Variations in mitragynine content in the naturally growing Kratom (Mitragyna speciosa) population of Thailand.
- Published in:
- Frontiers in Plant Science, 2022, v. 13, p. 1, doi. 10.3389/fpls.2022.1028547
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- Publication type:
- Article
Mitragynine Reverses Paclitaxel Chemotherapy‐Induced Peripheral Neuropathy and is Mediated via Opioid Receptor Involvement.
- Published in:
- FASEB Journal, 2022, v. 36, p. N.PAG, doi. 10.1096/fasebj.2022.36.S1.0R851
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- Publication type:
- Article
Probing the Activity of Mitragyna Speciosa (Kratom) Alkaloids at Serotonin G Protein‐Coupled Receptors.
- Published in:
- FASEB Journal, 2022, v. 36, p. N.PAG, doi. 10.1096/fasebj.2022.36.S1.R2407
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- Publication type:
- Article
Effects of Mitragynine and its Active Metabolites on the Reinforcing Effects of Remifentanil and Cocaine in Rats Self‐Administering Remifentanil.
- Published in:
- FASEB Journal, 2022, v. 36, p. N.PAG, doi. 10.1096/fasebj.2022.36.S1.R5776
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- Publication type:
- Article
Serotonin 5‐HT<sub>1A</sub> Receptor Activity of Kratom Alkaloids Mitragynine, Paynantheine, and Speciogynine.
- Published in:
- FASEB Journal, 2021, v. 35, p. N.PAG, doi. 10.1096/fasebj.2021.35.S1.04764
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- Publication type:
- Article
Pharmacological Characterization of Mitragynine: Antinociception, Respiratory Depression, Self‐Administration, Drug Discrimination, Tolerance, and withdrawal in Rats.
- Published in:
- FASEB Journal, 2021, v. 35, p. N.PAG, doi. 10.1096/fasebj.2021.35.S1.02725
- By:
- Publication type:
- Article
Mitragynine Attenuates the Development of Tolerance to and Withdrawal from Morphine in Rats.
- Published in:
- FASEB Journal, 2021, v. 35, p. N.PAG, doi. 10.1096/fasebj.2021.35.S1.05506
- By:
- Publication type:
- Article
Assessment of Contribution of 7‐Hydroxymitragynine and Mitragynine Pseudoindoxyl to the MU‐Opioid Activity of Mitragynine.
- Published in:
- FASEB Journal, 2021, v. 35, p. N.PAG, doi. 10.1096/fasebj.2021.35.S1.05475
- By:
- Publication type:
- Article
The Lofexidine‐Like Discriminative Effects of the Primary Kratom Alkaloid Mitragynine in Rats.
- Published in:
- FASEB Journal, 2021, v. 35, p. N.PAG, doi. 10.1096/fasebj.2021.35.S1.04912
- By:
- Publication type:
- Article
The dopamine uptake inhibitor, WIN 35,428, has sigma2 receptor agonist effects that contribute to its self‐administration (848.10).
- Published in:
- FASEB Journal, 2014, v. 28, p. N.PAG, doi. 10.1096/fasebj.28.1_supplement.848.10
- By:
- Publication type:
- Article
Preclinical efficacy of the dual sigma receptor antagonist dopamine uptake inhibitor, CM699, as a medication for stimulant abuse (803.3).
- Published in:
- FASEB Journal, 2014, v. 28, p. N.PAG, doi. 10.1096/fasebj.28.1_supplement.803.3
- By:
- Publication type:
- Article
The journey to AAPS 2020: a reflection from strategic planning to PharmSci 360.
- Published in:
- 2018
- By:
- Publication type:
- Editorial
Highly Specific Sigma Receptor Ligands Exhibit Anti-Viral Properties in SARS-CoV-2 Infected Cells.
- Published in:
- Pathogens, 2021, v. 10, n. 11, p. 1514, doi. 10.3390/pathogens10111514
- By:
- Publication type:
- Article
Brain Magnetic Resonance Imaging of Regular Kratom (Mitragyna speciosa Korth.) Users: A Preliminary Study.
- Published in:
- Malaysian Journal of Medicine & Health Sciences, 2018, v. 14, p. 65
- By:
- Publication type:
- Article
Further validation to support clinical translation of [<sup>18</sup>F]FTC-146 for imaging sigma-1 receptors.
- Published in:
- EJNMMI Research, 2015, v. 5, n. 1, p. 1, doi. 10.1186/s13550-015-0122-2
- By:
- Publication type:
- Article
Further validation to support clinical translation of [F]FTC-146 for imaging sigma-1 receptors.
- Published in:
- EJNMMI Research, 2015, v. 5, n. 1, p. 1, doi. 10.1186/s13550-015-0122-2
- By:
- Publication type:
- Article
Biodistribution and Radiation Dosimetry of 18F-FTC-146 in Humans.
- Published in:
- Journal of Nuclear Medicine, 2017, v. 58, n. 12, p. 2004, doi. 10.2967/jnumed.117.192641
- By:
- Publication type:
- Article
Evaluation of σ-1 Receptor Radioligand <sup>18</sup>F-FTC-146 in Rats and Squirrel Monkeys Using PET.
- Published in:
- Journal of Nuclear Medicine, 2014, v. 55, n. 1, p. 147, doi. 10.2967/jnumed.113.120261
- By:
- Publication type:
- Article
Novel Radioligands for Sigma-1 Receptor Binding Studies.
- Published in:
- FASEB Journal, 2008, v. 22, p. 628, doi. 10.1096/fasebj.22.2_supplement.628
- By:
- Publication type:
- Article
Toward Mycobacterium tuberculosis DXR inhibitor design: homology modeling and molecular dynamics simulations.
- Published in:
- Journal of Computer-Aided Molecular Design, 2007, v. 21, n. 9, p. 511, doi. 10.1007/s10822-007-9132-0
- By:
- Publication type:
- Article
A combined ligand-based and target-based drug design approach for G-protein coupled receptors: application to salvinorin A, a selective kappa opioid receptor agonist.
- Published in:
- Journal of Computer-Aided Molecular Design, 2006, v. 20, n. 7/8, p. 1, doi. 10.1007/s10822-006-9067-x
- By:
- Publication type:
- Article
Development and validation of a UPLC-MS/MS method for the determination of 7-hydroxymitragynine, a μ-opioid agonist, in rat plasma and its application to a pharmacokinetic study.
- Published in:
- Biomedical Chromatography, 2013, v. 27, n. 12, p. 1726, doi. 10.1002/bmc.2986
- By:
- Publication type:
- Article
Ultra-performance liquid chromatography tandem mass spectrometry method for the determination of AZ66, a sigma receptor ligand, in rat plasma and its application to in vivo pharmacokinetics.
- Published in:
- Biomedical Chromatography, 2013, v. 27, n. 8, p. 1034, doi. 10.1002/bmc.2901
- By:
- Publication type:
- Article